CA2587926A1 - Bicyclic inhibitors or rho kinase - Google Patents
Bicyclic inhibitors or rho kinase Download PDFInfo
- Publication number
- CA2587926A1 CA2587926A1 CA002587926A CA2587926A CA2587926A1 CA 2587926 A1 CA2587926 A1 CA 2587926A1 CA 002587926 A CA002587926 A CA 002587926A CA 2587926 A CA2587926 A CA 2587926A CA 2587926 A1 CA2587926 A1 CA 2587926A1
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- agent
- aliphatic
- disease
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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Landscapes
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US63011504P | 2004-11-22 | 2004-11-22 | |
| US60/630,115 | 2004-11-22 | ||
| PCT/US2005/042537 WO2006058120A1 (en) | 2004-11-22 | 2005-11-22 | Bicyclic inhibitors or rho kinase |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2587926A1 true CA2587926A1 (en) | 2006-06-01 |
Family
ID=35953926
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA002587894A Abandoned CA2587894A1 (en) | 2004-11-22 | 2005-11-22 | Pyrrolopyrazines and pyrazolopyrazines useful as inhibitors of protein kinases |
| CA002587926A Abandoned CA2587926A1 (en) | 2004-11-22 | 2005-11-22 | Bicyclic inhibitors or rho kinase |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA002587894A Abandoned CA2587894A1 (en) | 2004-11-22 | 2005-11-22 | Pyrrolopyrazines and pyrazolopyrazines useful as inhibitors of protein kinases |
Country Status (14)
| Country | Link |
|---|---|
| US (3) | US7795259B2 (enExample) |
| EP (3) | EP1814883A1 (enExample) |
| JP (3) | JP2008520738A (enExample) |
| KR (1) | KR20070089201A (enExample) |
| CN (1) | CN101098872B (enExample) |
| AU (2) | AU2005309616A1 (enExample) |
| CA (2) | CA2587894A1 (enExample) |
| IL (1) | IL183318A0 (enExample) |
| MX (1) | MX2007006103A (enExample) |
| NO (1) | NO20073140L (enExample) |
| NZ (1) | NZ555566A (enExample) |
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| ZA (1) | ZA200704888B (enExample) |
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| TW202304459A (zh) | 2021-04-12 | 2023-02-01 | 美商英塞特公司 | 包含ｆｇｆｒ抑制劑及ｎｅｃｔｉｎ－４靶向劑之組合療法 |
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| MC2096A1 (fr) * | 1989-02-23 | 1991-02-15 | Hoffmann La Roche | Pyrroles substitues |
| JP2648372B2 (ja) * | 1989-09-18 | 1997-08-27 | キヤノン株式会社 | インクジェット記録装置 |
| AU782775B2 (en) * | 2000-02-05 | 2005-08-25 | Vertex Pharmaceuticals Incorporated | Pyrazole compositions useful as inhibitors of ERK |
| MY130778A (en) * | 2001-02-09 | 2007-07-31 | Vertex Pharma | Heterocyclic inhibitiors of erk2 and uses thereof |
| GB0115109D0 (en) * | 2001-06-21 | 2001-08-15 | Aventis Pharma Ltd | Chemical compounds |
| WO2003000588A1 (de) | 2001-06-22 | 2003-01-03 | Basf Aktiengesellschaft | Stäbchenförmige apatitkristalle mit einem bestimmten länge-zu-breite-verhältnis |
| US7101884B2 (en) * | 2001-09-14 | 2006-09-05 | Merck & Co., Inc. | Tyrosine kinase inhibitors |
| GB0206860D0 (en) * | 2002-03-22 | 2002-05-01 | Glaxo Group Ltd | Compounds |
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| CA2504320A1 (en) * | 2002-10-30 | 2004-05-21 | Vertex Pharmaceuticals Incorporated | Compositions useful as inhibitors of rock and other protein kinases |
| CA2501365C (en) * | 2002-10-30 | 2011-05-31 | Merck & Co., Inc. | Inhibitors of akt activity |
| TWI339206B (en) * | 2003-09-04 | 2011-03-21 | Vertex Pharma | Compositions useful as inhibitors of protein kinases |
| JP2007523938A (ja) * | 2004-02-27 | 2007-08-23 | エフ．ホフマン−ラ ロシュ アーゲー | ピラゾールの縮合誘導体 |
| EP1720878A1 (en) * | 2004-02-27 | 2006-11-15 | F.Hoffmann-La Roche Ag | Heteroaryl-fused pyrazolo derivatives |
| US7763843B2 (en) | 2004-03-01 | 2010-07-27 | Stanton Magnetics, Inc. | Optical navigation system for rotary control based non-contact controller |
| AU2005236002A1 (en) * | 2004-04-02 | 2005-11-03 | Vertex Pharmaceuticals Incorporated | Azaindoles useful as inhibitors of rock and other protein kinases |
| CN101389626A (zh) * | 2004-07-27 | 2009-03-18 | Sgx药物公司 | 稠环杂环激酶调节剂 |
| CA2573573A1 (en) * | 2004-07-27 | 2006-02-09 | Sgx Pharmaceuticals, Inc. | Fused ring heterocycle kinase modulators |
-
2005
- 2005-11-22 CN CN2005800460428A patent/CN101098872B/zh not_active Expired - Fee Related
- 2005-11-22 KR KR1020077014367A patent/KR20070089201A/ko not_active Withdrawn
- 2005-11-22 RU RU2007123360/04A patent/RU2394825C2/ru not_active IP Right Cessation
- 2005-11-22 EP EP05825542A patent/EP1814883A1/en not_active Withdrawn
- 2005-11-22 ZA ZA200704888A patent/ZA200704888B/xx unknown
- 2005-11-22 EP EP05825395A patent/EP1814882A1/en not_active Withdrawn
- 2005-11-22 WO PCT/US2005/042455 patent/WO2006058074A1/en not_active Ceased
- 2005-11-22 JP JP2007543441A patent/JP2008520738A/ja active Pending
- 2005-11-22 JP JP2007543468A patent/JP2008520745A/ja active Pending
- 2005-11-22 EP EP10185488A patent/EP2316835A1/en not_active Withdrawn
- 2005-11-22 US US11/285,497 patent/US7795259B2/en not_active Expired - Fee Related
- 2005-11-22 AU AU2005309616A patent/AU2005309616A1/en not_active Abandoned
- 2005-11-22 AU AU2005309566A patent/AU2005309566A1/en not_active Abandoned
- 2005-11-22 CA CA002587894A patent/CA2587894A1/en not_active Abandoned
- 2005-11-22 CA CA002587926A patent/CA2587926A1/en not_active Abandoned
- 2005-11-22 WO PCT/US2005/042537 patent/WO2006058120A1/en not_active Ceased
- 2005-11-22 US US11/285,516 patent/US20060122185A1/en not_active Abandoned
- 2005-11-22 NZ NZ555566A patent/NZ555566A/en not_active IP Right Cessation
- 2005-11-22 MX MX2007006103A patent/MX2007006103A/es active IP Right Grant
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2007
- 2007-05-20 IL IL183318A patent/IL183318A0/en unknown
- 2007-06-20 NO NO20073140A patent/NO20073140L/no not_active Application Discontinuation
-
2008
- 2008-09-12 JP JP2008235263A patent/JP2009024024A/ja active Pending
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2010
- 2010-07-30 US US12/847,136 patent/US8372835B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| EP1814882A1 (en) | 2007-08-08 |
| US20060122185A1 (en) | 2006-06-08 |
| JP2008520738A (ja) | 2008-06-19 |
| US20110081364A1 (en) | 2011-04-07 |
| ZA200704888B (en) | 2009-02-25 |
| US7795259B2 (en) | 2010-09-14 |
| CA2587894A1 (en) | 2006-06-01 |
| AU2005309566A1 (en) | 2006-06-01 |
| NO20073140L (no) | 2007-06-20 |
| CN101098872B (zh) | 2012-09-05 |
| RU2394825C2 (ru) | 2010-07-20 |
| NZ555566A (en) | 2009-12-24 |
| US8372835B2 (en) | 2013-02-12 |
| IL183318A0 (en) | 2007-09-20 |
| WO2006058074A1 (en) | 2006-06-01 |
| WO2006058120A1 (en) | 2006-06-01 |
| EP2316835A1 (en) | 2011-05-04 |
| KR20070089201A (ko) | 2007-08-30 |
| CN101098872A (zh) | 2008-01-02 |
| MX2007006103A (es) | 2007-07-20 |
| US20060258662A1 (en) | 2006-11-16 |
| JP2008520745A (ja) | 2008-06-19 |
| AU2005309616A1 (en) | 2006-06-01 |
| JP2009024024A (ja) | 2009-02-05 |
| EP1814883A1 (en) | 2007-08-08 |
| RU2007123360A (ru) | 2009-01-27 |
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