US4232027A
(en)
|
1979-01-29 |
1980-11-04 |
E. R. Squibb & Sons, Inc. |
1,2-Dihydro-2-oxo-4-phenyl-3-quinolinecarbonitrile derivatives
|
GB2116183B
(en)
|
1982-03-03 |
1985-06-05 |
Genentech Inc |
Human antithrombin iii dna sequences therefore expression vehicles and cloning vectors containing such sequences and cell cultures transformed thereby a process for expressing human antithrombin iii and pharmaceutical compositions comprising it
|
GB8827305D0
(en)
|
1988-11-23 |
1988-12-29 |
British Bio Technology |
Compounds
|
JP2762522B2
(ja)
|
1989-03-06 |
1998-06-04 |
藤沢薬品工業株式会社 |
血管新生阻害剤
|
GB8912336D0
(en)
|
1989-05-30 |
1989-07-12 |
Smithkline Beckman Intercredit |
Compounds
|
US5112946A
(en)
|
1989-07-06 |
1992-05-12 |
Repligen Corporation |
Modified pf4 compositions and methods of use
|
PT98990A
(pt)
|
1990-09-19 |
1992-08-31 |
American Home Prod |
Processo para a preparacao de esteres de acidos carboxilicos de rapamicina
|
US5892112A
(en)
|
1990-11-21 |
1999-04-06 |
Glycomed Incorporated |
Process for preparing synthetic matrix metalloprotease inhibitors
|
US5120842A
(en)
|
1991-04-01 |
1992-06-09 |
American Home Products Corporation |
Silyl ethers of rapamycin
|
US5100883A
(en)
|
1991-04-08 |
1992-03-31 |
American Home Products Corporation |
Fluorinated esters of rapamycin
|
US5118678A
(en)
|
1991-04-17 |
1992-06-02 |
American Home Products Corporation |
Carbamates of rapamycin
|
CA2066898A1
(fr)
|
1991-04-29 |
1992-10-30 |
Chuan Shih |
Composes pharmaceutiques
|
SG64322A1
(en)
|
1991-05-10 |
1999-04-27 |
Rhone Poulenc Rorer Int |
Bis mono and bicyclic aryl and heteroaryl compounds which inhibit egf and/or pdgf receptor tyrosine kinase
|
US5118677A
(en)
|
1991-05-20 |
1992-06-02 |
American Home Products Corporation |
Amide esters of rapamycin
|
NZ243082A
(en)
|
1991-06-28 |
1995-02-24 |
Ici Plc |
4-anilino-quinazoline derivatives; pharmaceutical compositions, preparatory processes, and use thereof
|
US5151413A
(en)
|
1991-11-06 |
1992-09-29 |
American Home Products Corporation |
Rapamycin acetals as immunosuppressant and antifungal agents
|
GB9125660D0
(en)
|
1991-12-03 |
1992-01-29 |
Smithkline Beecham Plc |
Novel compound
|
GB9300059D0
(en)
|
1992-01-20 |
1993-03-03 |
Zeneca Ltd |
Quinazoline derivatives
|
US5521184A
(en)
|
1992-04-03 |
1996-05-28 |
Ciba-Geigy Corporation |
Pyrimidine derivatives and processes for the preparation thereof
|
ZA935111B
(en)
|
1992-07-17 |
1994-02-04 |
Smithkline Beecham Corp |
Rapamycin derivatives
|
ZA935112B
(en)
|
1992-07-17 |
1994-02-08 |
Smithkline Beecham Corp |
Rapamycin derivatives
|
US5256790A
(en)
|
1992-08-13 |
1993-10-26 |
American Home Products Corporation |
27-hydroxyrapamycin and derivatives thereof
|
GB9221220D0
(en)
|
1992-10-09 |
1992-11-25 |
Sandoz Ag |
Organic componds
|
US5258389A
(en)
|
1992-11-09 |
1993-11-02 |
Merck & Co., Inc. |
O-aryl, O-alkyl, O-alkenyl and O-alkynylrapamycin derivatives
|
ES2279508T3
(es)
|
1992-11-13 |
2007-08-16 |
Immunex Corporation |
Ligando elk, una citoquina.
|
US5455258A
(en)
|
1993-01-06 |
1995-10-03 |
Ciba-Geigy Corporation |
Arylsulfonamido-substituted hydroxamic acids
|
US5629327A
(en)
|
1993-03-01 |
1997-05-13 |
Childrens Hospital Medical Center Corp. |
Methods and compositions for inhibition of angiogenesis
|
US5516658A
(en)
|
1993-08-20 |
1996-05-14 |
Immunex Corporation |
DNA encoding cytokines that bind the cell surface receptor hek
|
JPH08503971A
(ja)
|
1993-10-01 |
1996-04-30 |
チバ−ガイギー アクチェンゲゼルシャフト |
ピリミジンアミン誘導体及びその調製のための方法
|
US5656643A
(en)
|
1993-11-08 |
1997-08-12 |
Rhone-Poulenc Rorer Pharmaceuticals Inc. |
Bis mono-and bicyclic aryl and heteroaryl compounds which inhibit EGF and/or PDGF receptor tyrosine kinase
|
CA2175215C
(fr)
|
1993-11-19 |
2008-06-03 |
Yat Sun Or |
Analogues semi-synthetiques de rapamycine (macrolides) utilises comme immunomodulateurs
|
ATE191218T1
(de)
|
1993-12-17 |
2000-04-15 |
Novartis Ag |
Rapamycin-derivate als immunosuppressoren
|
US5700823A
(en)
|
1994-01-07 |
1997-12-23 |
Sugen, Inc. |
Treatment of platelet derived growth factor related disorders such as cancers
|
IL112249A
(en)
|
1994-01-25 |
2001-11-25 |
Warner Lambert Co |
Pharmaceutical compositions containing di and tricyclic pyrimidine derivatives for inhibiting tyrosine kinases of the epidermal growth factor receptor family and some new such compounds
|
IL112248A0
(en)
|
1994-01-25 |
1995-03-30 |
Warner Lambert Co |
Tricyclic heteroaromatic compounds and pharmaceutical compositions containing them
|
AU2096895A
(en)
|
1994-03-07 |
1995-09-25 |
Sugen, Incorporated |
Receptor tyrosine kinase inhibitors for inhibiting cell proliferative disorders and compositions thereof
|
WO1995028484A1
(fr)
|
1994-04-15 |
1995-10-26 |
Amgen Inc. |
Nouvelles proteines tyrosine kinases receptrices analogues a l'eph, du type hek5, hek7, hek8, hek11
|
DK0682027T3
(da)
|
1994-05-03 |
1998-05-04 |
Ciba Geigy Ag |
Pyrrolopyrimidinderivater med antiproliferativ virkning
|
US6303769B1
(en)
|
1994-07-08 |
2001-10-16 |
Immunex Corporation |
Lerk-5 dna
|
US5919905A
(en)
|
1994-10-05 |
1999-07-06 |
Immunex Corporation |
Cytokine designated LERK-6
|
US6057124A
(en)
|
1995-01-27 |
2000-05-02 |
Amgen Inc. |
Nucleic acids encoding ligands for HEK4 receptors
|
US5863949A
(en)
|
1995-03-08 |
1999-01-26 |
Pfizer Inc |
Arylsulfonylamino hydroxamic acid derivatives
|
ES2332984T3
(es)
|
1995-03-30 |
2010-02-16 |
Pfizer Products Inc. |
Derivados de quinazolinas.
|
ES2150113T3
(es)
|
1995-04-03 |
2000-11-16 |
Novartis Ag |
Derivados de pirazol y procedimientos para la preparacion de los mismos.
|
MX9708026A
(es)
|
1995-04-20 |
1997-11-29 |
Pfizer |
Derivados del acido arislfulfonil hidroxamico, composiciones que los contienen y uso de los mismos.
|
GB9508538D0
(en)
|
1995-04-27 |
1995-06-14 |
Zeneca Ltd |
Quinazoline derivatives
|
US5747498A
(en)
|
1996-05-28 |
1998-05-05 |
Pfizer Inc. |
Alkynyl and azido-substituted 4-anilinoquinazolines
|
US5650415A
(en)
|
1995-06-07 |
1997-07-22 |
Sugen, Inc. |
Quinoline compounds
|
US5880141A
(en)
|
1995-06-07 |
1999-03-09 |
Sugen, Inc. |
Benzylidene-Z-indoline compounds for the treatment of disease
|
PT833828E
(pt)
|
1995-06-09 |
2003-02-28 |
Novartis Ag |
Derivados de rapamicina
|
PT836605E
(pt)
|
1995-07-06 |
2002-07-31 |
Novartis Ag |
Pirrolopirimidinas e processos para a sua preparacao
|
US5573001A
(en)
|
1995-09-08 |
1996-11-12 |
Acuson Corporation |
Ultrasonic receive beamformer with phased sub-arrays
|
DE19534177A1
(de)
|
1995-09-15 |
1997-03-20 |
Merck Patent Gmbh |
Cyclische Adhäsionsinhibitoren
|
AR004010A1
(es)
|
1995-10-11 |
1998-09-30 |
Glaxo Group Ltd |
Compuestos heterociclicos
|
GB9523675D0
(en)
|
1995-11-20 |
1996-01-24 |
Celltech Therapeutics Ltd |
Chemical compounds
|
ATE225343T1
(de)
|
1995-12-20 |
2002-10-15 |
Hoffmann La Roche |
Matrix-metalloprotease inhibitoren
|
AU1441497A
(en)
|
1996-01-23 |
1997-08-20 |
Novartis Ag |
Pyrrolopyrimidines and processes for their preparation
|
JP3406763B2
(ja)
|
1996-01-30 |
2003-05-12 |
東レ・ダウコーニング・シリコーン株式会社 |
シリコーンゴム組成物
|
GB9603095D0
(en)
|
1996-02-14 |
1996-04-10 |
Zeneca Ltd |
Quinazoline derivatives
|
GB9603097D0
(en)
|
1996-02-14 |
1996-04-10 |
Zeneca Ltd |
Quinazoline compounds
|
DE19608588A1
(de)
|
1996-03-06 |
1997-09-11 |
Thomae Gmbh Dr K |
Pyrimido [5,4-d]pyrimidine, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung
|
DE19629652A1
(de)
|
1996-03-06 |
1998-01-29 |
Thomae Gmbh Dr K |
4-Amino-pyrimidin-Derivate, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung
|
US6051577A
(en)
|
1996-03-15 |
2000-04-18 |
Novartis Ag |
N-7-heterocyclyl pyrrolo[2,3-D]pyrimidines and the use thereof
|
AU725533B2
(en)
|
1996-04-12 |
2000-10-12 |
Warner-Lambert Company |
Irreversible inhibitors of tyrosine kinases
|
GB9607729D0
(en)
|
1996-04-13 |
1996-06-19 |
Zeneca Ltd |
Quinazoline derivatives
|
AU2912997A
(en)
|
1996-06-24 |
1998-01-14 |
Pfizer Inc. |
Phenylamino-substituted tricyclic derivatives for treatment of hyperproliferative diseases
|
EP0818442A3
(fr)
|
1996-07-12 |
1998-12-30 |
Pfizer Inc. |
Dérivés cycliques de sulfones comme inhibiteurs de métalloprotéinase et de la production du facteur de nécrose des tumeurs
|
WO1998002441A2
(fr)
|
1996-07-12 |
1998-01-22 |
Ariad Pharmaceuticals, Inc. |
Elements et procedes pour traiter ou prevenir les mycoses pathogènes
|
HRP970371A2
(en)
|
1996-07-13 |
1998-08-31 |
Kathryn Jane Smith |
Heterocyclic compounds
|
ID19609A
(id)
|
1996-07-13 |
1998-07-23 |
Glaxo Group Ltd |
Senyawa-senyawa heterosiklik
|
JP2000515136A
(ja)
|
1996-07-13 |
2000-11-14 |
グラクソ、グループ、リミテッド |
プロテインチロシンキナーゼ阻害剤としての二環式ヘテロ芳香族化合物
|
JP3299975B2
(ja)
|
1996-07-18 |
2002-07-08 |
ファイザー・インク |
マトリックスメタロプロテアーゼのホスフィン酸塩ベース阻害薬
|
US6111090A
(en)
|
1996-08-16 |
2000-08-29 |
Schering Corporation |
Mammalian cell surface antigens; related reagents
|
AU4055697A
(en)
|
1996-08-16 |
1998-03-06 |
Schering Corporation |
Mammalian cell surface antigens; related reagents
|
AU720429B2
(en)
|
1996-08-23 |
2000-06-01 |
Novartis Ag |
Substituted pyrrolopyrimidines and processes for their preparation
|
EP0922030A1
(fr)
|
1996-08-23 |
1999-06-16 |
Pfizer Inc. |
Derives de l'acide arylsulfonylamino hydroxamique
|
ID18494A
(id)
|
1996-10-02 |
1998-04-16 |
Novartis Ag |
Turunan pirazola leburan dan proses pembuatannya
|
WO1998014449A1
(fr)
|
1996-10-02 |
1998-04-09 |
Novartis Ag |
Derives de pyrazole condenses et procedes pour leur preparation
|
ES2239779T3
(es)
|
1996-10-02 |
2005-10-01 |
Novartis Ag |
Derivados de pirimidina y procedimientos para la preparacion de los mismos.
|
EP0837063A1
(fr)
|
1996-10-17 |
1998-04-22 |
Pfizer Inc. |
Dérivés de 4-aminoquinazoline
|
GB9621757D0
(en)
|
1996-10-18 |
1996-12-11 |
Ciba Geigy Ag |
Phenyl-substituted bicyclic heterocyclyl derivatives and their use
|
US6077864A
(en)
|
1997-01-06 |
2000-06-20 |
Pfizer Inc. |
Cyclic sulfone derivatives
|
DK0977733T3
(da)
|
1997-02-03 |
2003-11-24 |
Pfizer Prod Inc |
Arylsulfonylaminohydroxamsyrederivater
|
JP2001509805A
(ja)
|
1997-02-05 |
2001-07-24 |
ワーナー−ランバート・コンパニー |
細胞増殖阻害剤としてのピリド〔2,3−d〕ピリミジンおよび4−アミノピリミジン
|
JP2000507975A
(ja)
|
1997-02-07 |
2000-06-27 |
ファイザー・インク |
N−ヒドロキシ−β−スルホニルプロピオンアミド誘導体類及びそれらのマトリックスメタロプロテイナーゼ阻害薬としての使用
|
CA2280151C
(fr)
|
1997-02-11 |
2005-12-13 |
Pfizer Inc. |
Derives de l'acide arylsulfonylhydroxamique
|
CO4950519A1
(es)
|
1997-02-13 |
2000-09-01 |
Novartis Ag |
Ftalazinas, preparaciones farmaceuticas que las comprenden y proceso para su preparacion
|
US6150395A
(en)
|
1997-05-30 |
2000-11-21 |
The Regents Of The University Of California |
Indole-3-carbinol (I3C) derivatives and methods
|
WO1999007701A1
(fr)
|
1997-08-05 |
1999-02-18 |
Sugen, Inc. |
Derives de quinoxaline tricyclique utiles en tant qu'inhibiteurs de proteine tyrosine kinase
|
JP3448275B2
(ja)
|
1997-08-08 |
2003-09-22 |
ファイザー・プロダクツ・インク |
アリールオキシアリールスルホニルアミノヒドロキサム酸誘導体
|
CA2308114A1
(fr)
|
1997-10-21 |
1999-04-29 |
Human Genome Sciences, Inc. |
Proteines tr11, tr11sv1 et tr11sv2 de type recepteur du facteur de necrose tumorale humain
|
GB9725782D0
(en)
|
1997-12-05 |
1998-02-04 |
Pfizer Ltd |
Therapeutic agents
|
GB9800569D0
(en)
|
1998-01-12 |
1998-03-11 |
Glaxo Group Ltd |
Heterocyclic compounds
|
GB9800575D0
(en)
|
1998-01-12 |
1998-03-11 |
Glaxo Group Ltd |
Heterocyclic compounds
|
GB9801690D0
(en)
|
1998-01-27 |
1998-03-25 |
Pfizer Ltd |
Therapeutic agents
|
IL137409A0
(en)
|
1998-02-09 |
2001-07-24 |
Genentech Inc |
Novel tumor necrosis factor receptor homolog and nucleic acids encoding the same
|
ATE430149T1
(de)
|
1998-03-04 |
2009-05-15 |
Bristol Myers Squibb Co |
Heterocyclen substituierte imidazopyrazine als protein- tyrosin-kinase-inhibitoren
|
PA8469501A1
(es)
|
1998-04-10 |
2000-09-29 |
Pfizer Prod Inc |
Hidroxamidas del acido (4-arilsulfonilamino)-tetrahidropiran-4-carboxilico
|
PA8469401A1
(es)
|
1998-04-10 |
2000-05-24 |
Pfizer Prod Inc |
Derivados biciclicos del acido hidroxamico
|
IL139934A
(en)
|
1998-05-29 |
2007-10-31 |
Sugen Inc |
History 2 - Indulinone converted to pyrrole and pharmaceutical preparations containing them
|
UA60365C2
(uk)
|
1998-06-04 |
2003-10-15 |
Пфайзер Продактс Інк. |
Похідні ізотіазолу, спосіб їх одержання, фармацевтична композиція та спосіб лікування гіперпроліферативного захворювання у ссавця
|
AU747427B2
(en)
|
1998-07-10 |
2002-05-16 |
Merck & Co., Inc. |
Novel angiogenesis inhibitors
|
EP1109555A4
(fr)
|
1998-08-31 |
2001-11-21 |
Merck & Co Inc |
Nouveaux inhibiteurs d'angiogenese
|
ES2213985T3
(es)
|
1998-11-05 |
2004-09-01 |
Pfizer Products Inc. |
Derivados de hidroxiamida de acido 5-oxo-pirrolidin-2-carboxilico.
|
ES2384160T3
(es)
|
1999-01-13 |
2012-07-02 |
Bayer Healthcare Llc |
Difenil ureas sustituidas con omega-carboxi arilo como agentes inhibidores de la cinasa p38
|
AU766081B2
(en)
|
1999-03-30 |
2003-10-09 |
Novartis Ag |
Phthalazine derivatives for treating inflammatory diseases
|
GB9912961D0
(en)
|
1999-06-03 |
1999-08-04 |
Pfizer Ltd |
Metalloprotease inhibitors
|
WO2000075323A1
(fr)
|
1999-06-07 |
2000-12-14 |
Immunex Corporation |
Antagonistes tek
|
US6521424B2
(en)
|
1999-06-07 |
2003-02-18 |
Immunex Corporation |
Recombinant expression of Tek antagonists
|
WO2001003720A2
(fr)
|
1999-07-12 |
2001-01-18 |
Genentech, Inc. |
Stimulation ou inhibition de l'angiogenese et de la cardiovascularisation avec des homologues de ligands et de recepteurs du facteur de necrose tumorale
|
ATE264863T1
(de)
|
1999-08-24 |
2004-05-15 |
Ariad Gene Therapeutics Inc |
28-epirapaloge
|
JP3522727B2
(ja)
|
1999-11-05 |
2004-04-26 |
アストラゼネカ アクチボラグ |
Vegf阻害剤としてのキナゾリン誘導体
|
ES2367007T3
(es)
|
1999-11-24 |
2011-10-27 |
Sugen, Inc. |
Derivados de indolinona ionizables y su uso como ligandos de ptk.
|
US6515004B1
(en)
|
1999-12-15 |
2003-02-04 |
Bristol-Myers Squibb Company |
N-[5-[[[5-alkyl-2-oxazolyl]methyl]thio]-2-thiazolyl]-carboxamide inhibitors of cyclin dependent kinases
|
US6727225B2
(en)
|
1999-12-20 |
2004-04-27 |
Immunex Corporation |
TWEAK receptor
|
AU4721901A
(en)
|
2000-02-25 |
2001-09-03 |
Immunex Corp |
Integrin antagonists
|
WO2002006213A2
(fr)
|
2000-07-19 |
2002-01-24 |
Warner-Lambert Company |
Esters oxygenes d'acides 4-iodophenylamino benzhydroxamiques
|
US6630500B2
(en)
|
2000-08-25 |
2003-10-07 |
Cephalon, Inc. |
Selected fused pyrrolocarbazoles
|
WO2002059110A1
(fr)
|
2000-12-21 |
2002-08-01 |
Glaxo Group Limited |
Composes chimiques
|
US20020147198A1
(en)
|
2001-01-12 |
2002-10-10 |
Guoqing Chen |
Substituted arylamine derivatives and methods of use
|
US6995162B2
(en)
|
2001-01-12 |
2006-02-07 |
Amgen Inc. |
Substituted alkylamine derivatives and methods of use
|
US7105682B2
(en)
|
2001-01-12 |
2006-09-12 |
Amgen Inc. |
Substituted amine derivatives and methods of use
|
US7102009B2
(en)
|
2001-01-12 |
2006-09-05 |
Amgen Inc. |
Substituted amine derivatives and methods of use
|
US6878714B2
(en)
|
2001-01-12 |
2005-04-12 |
Amgen Inc. |
Substituted alkylamine derivatives and methods of use
|
US20050026868A1
(en)
|
2003-07-11 |
2005-02-03 |
Metcalf Chester A. |
Phosphorus-containing macrocycles
|
US7307088B2
(en)
|
2002-07-09 |
2007-12-11 |
Amgen Inc. |
Substituted anthranilic amide derivatives and methods of use
|
TWI329112B
(en)
|
2002-07-19 |
2010-08-21 |
Bristol Myers Squibb Co |
Novel inhibitors of kinases
|
WO2004063195A1
(fr)
|
2003-01-03 |
2004-07-29 |
Sloan-Kettering Institute For Cancer Research |
Inhibiteurs de kinases a base de pyridopyrimidine
|
KR20060052681A
(ko)
|
2003-05-23 |
2006-05-19 |
와이어쓰 |
Gitr 리간드, gitr 리간드-연관 분자, 항체 및그의 용도
|
MXPA06000117A
(es)
|
2003-07-08 |
2006-04-27 |
Novartis Ag |
Uso de rapamicina y derivados de rapamicina para el tratamiento de perdida osea.
|
WO2005007190A1
(fr)
|
2003-07-11 |
2005-01-27 |
Schering Corporation |
Agonistes ou antagonistes du recepteur du facteur de necrose tumorale induit par les glucocorticoides (gitr) ou de son ligand utilises dans le traitement des troubles immuns, des infections et du cancer
|
AR045134A1
(es)
|
2003-07-29 |
2005-10-19 |
Smithkline Beecham Plc |
Compuesto de 1h - imidazo [4,5-c] piridin-ilo, composicion farmaceutica que lo comprende, proceso para prepararla, su uso para preparar dicha composicion farmaceutica, combinacion farmaceutica, uso de la combinacion farmaceutica para la preparacion de un medicamento, procedimientos para preparar dic
|
JP2007503388A
(ja)
|
2003-08-22 |
2007-02-22 |
アバニール・ファーマシューティカルズ |
マクロファージ遊走阻止因子の阻害剤としての置換ナフチリジン誘導体、およびヒト疾患の治療におけるそれらの使用
|
WO2005055808A2
(fr)
|
2003-12-02 |
2005-06-23 |
Genzyme Corporation |
Compositions et methodes pour le diagnostic et le traitement du cancer du poumon
|
GB0409799D0
(en)
|
2004-04-30 |
2004-06-09 |
Isis Innovation |
Method of generating improved immune response
|
EP1765402A2
(fr)
|
2004-06-04 |
2007-03-28 |
Duke University |
Methodes et compositions ameliorant l'immunite par depletion in vivo de l'activite cellulaire immunosuppressive
|
CA2578066C
(fr)
|
2004-08-26 |
2011-10-11 |
Pfizer Inc. |
Composes d'aminoheteroaryle enantiomeriquement purs utilises comme inhibiteurs de proteine kinase
|
WO2006044453A1
(fr)
|
2004-10-13 |
2006-04-27 |
Wyeth |
Analogues de la 17-hydroxywortmannine employés en tant qu’inhibiteurs de pi3k
|
US7354944B2
(en)
|
2004-10-18 |
2008-04-08 |
Amgen Inc. |
Thiadiazole compounds and methods of use
|
PT2343320T
(pt)
|
2005-03-25 |
2018-01-23 |
Gitr Inc |
Anticorpos anti-gitr e as suas utilizações
|
CA3151350A1
(fr)
|
2005-05-09 |
2006-11-16 |
E. R. Squibb & Sons, L.L.C. |
Anticorps monoclonaux humains pour mort programmee 1 (mp-1) et procedes pour traiter le cancer en utilisant des anticorps anti-mp-1 seuls ou associes a d'autres immunotherapies
|
GB0510390D0
(en)
|
2005-05-20 |
2005-06-29 |
Novartis Ag |
Organic compounds
|
BRPI0616202A2
(pt)
|
2005-09-20 |
2011-06-14 |
Pfizer Prod Inc |
formas de dosagem e uso de um inibidor da tirosina quinase
|
EA200801716A1
(ru)
|
2006-01-18 |
2009-04-28 |
Амген Инк. |
Тиазольные соединения и их применение
|
EP1981969A4
(fr)
|
2006-01-19 |
2009-06-03 |
Genzyme Corp |
Anticorps anti-gitr destines au traitement du cancer
|
EP2518074B1
(fr)
|
2006-12-07 |
2015-07-22 |
F.Hoffmann-La Roche Ag |
Composés inhibiteurs de phosphoinositide 3-kinase et procédés d'utilisation
|
AU2008231385B2
(en)
|
2007-03-23 |
2012-02-02 |
Amgen Inc. |
Delta3- substituted quinoline or quinoxaline derivatives and their use as phosphatidylinositol 3-kinase ( PI3K) inhibitors
|
HUE028954T2
(en)
|
2007-03-23 |
2017-01-30 |
Amgen Inc |
Heterocyclic compounds and their use
|
WO2008118454A2
(fr)
|
2007-03-23 |
2008-10-02 |
Amgen Inc. |
Composés hétérocycliques et leurs utilisations
|
US8557830B2
(en)
|
2007-06-07 |
2013-10-15 |
Amgen Inc. |
RAF kinase modulators and methods of use
|
CA2693677C
(fr)
|
2007-07-12 |
2018-02-13 |
Tolerx, Inc. |
Therapies combinees utilisant des molecules de liaison au gitr
|
AU2008276512A1
(en)
|
2007-07-17 |
2009-01-22 |
Amgen Inc. |
Thiadiazole modulators of PKB
|
AU2008276521B2
(en)
|
2007-07-17 |
2011-11-03 |
Amgen Inc. |
Heterocyclic modulators of PKB
|
TW200911798A
(en)
|
2007-08-02 |
2009-03-16 |
Amgen Inc |
PI3 kinase modulators and methods of use
|
TWI471134B
(zh)
|
2007-09-12 |
2015-02-01 |
Genentech Inc |
肌醇磷脂3-激酶抑制劑化合物及化療劑之組合及使用方法
|
JP5348725B2
(ja)
|
2007-10-25 |
2013-11-20 |
ジェネンテック, インコーポレイテッド |
チエノピリミジン化合物の製造方法
|
NZ586069A
(en)
|
2007-12-19 |
2012-05-25 |
Amgen Inc |
Fused pyridine, pyrimidine and triazine compounds as cell cycle inhibitors
|
AU2008343813B2
(en)
|
2007-12-19 |
2012-04-12 |
Amgen Inc. |
Inhibitors of PI3 kinase
|
CA2719538C
(fr)
|
2008-04-07 |
2014-03-18 |
Amgen Inc. |
Pyridines/pyrimidines amino spirocycliques et disubstituees par gem en tant qu'inhibiteurs de cycle cellulaire
|
AU2009260447B2
(en)
|
2008-05-30 |
2012-03-29 |
Amgen Inc. |
Inhibitors of PI3 kinase
|
AU2009266873A1
(en)
|
2008-07-02 |
2010-01-07 |
Emergent Product Development Seattle, Llc |
TGF-beta antagonist multi-target binding proteins
|
US8586023B2
(en)
|
2008-09-12 |
2013-11-19 |
Mie University |
Cell capable of expressing exogenous GITR ligand
|
EP2387570A1
(fr)
|
2009-01-15 |
2011-11-23 |
Amgen, Inc |
Thiazoles substitués par fluoroisoquinoléine et leurs méthodes d'application
|
EP2398791A1
(fr)
|
2009-02-18 |
2011-12-28 |
Amgen, Inc |
Composés d'indole ou benzimidazole convenant comme inhibiteurs de la kinase mtor
|
WO2010108074A2
(fr)
|
2009-03-20 |
2010-09-23 |
Amgen Inc. |
Inhibiteurs de pi3 kinase
|
UY32582A
(es)
|
2009-04-28 |
2010-11-30 |
Amgen Inc |
Inhibidores de fosfoinositida 3 cinasa y/u objetivo mamífero
|
MX2011012037A
(es)
|
2009-05-13 |
2012-02-28 |
Amgen Inc |
Compuestos de heteroarilo como inhibidores de pikk.
|
WO2010151735A2
(fr)
|
2009-06-25 |
2010-12-29 |
Amgen Inc. |
Composés hétérocycliques et leurs utilisations
|
BRPI1016150A2
(pt)
|
2009-06-25 |
2016-04-19 |
Amgen Inc |
compostos heterocíclicos e seus usos.
|
TW201111376A
(en)
|
2009-06-25 |
2011-04-01 |
Amgen Inc |
Heterocyclic compounds and their uses
|
MX2011013667A
(es)
|
2009-06-25 |
2012-03-06 |
Amgen Inc |
Compuestos heterociclicos y sus usos.
|
EP2266984A1
(fr)
|
2009-06-26 |
2010-12-29 |
Deutsches Krebsforschungszentrum Stiftung des öffentlichen Rechts |
Pyrido[2,3-d]pyrimidines en tant qu' antagoniste du Wnt pour le traitement du cancer et de l'arthrite
|
CA2772613C
(fr)
|
2009-09-03 |
2020-03-10 |
Schering Corporation |
Anticorps anti-gitr
|
NZ598758A
(en)
|
2009-09-11 |
2013-12-20 |
Amgen Inc |
N-4 (-((3-(2-amino-4 pyrimidinyl)-2-pyridinyl)oxy)phenyl)-4-(4-methyl-2-thienyl)-1-phthalazinamine for use in the treatment of antimitotic agent resistant cancer
|
GB0919054D0
(en)
|
2009-10-30 |
2009-12-16 |
Isis Innovation |
Treatment of obesity
|
EA022984B1
(ru)
|
2009-12-29 |
2016-04-29 |
Эмерджент Продакт Дивелопмент Сиэтл, Ллс |
Конструкты, связывающиеся с ron, и способы их использования
|
US9133164B2
(en)
|
2011-04-13 |
2015-09-15 |
Innov88 Llc |
MIF inhibitors and their uses
|
WO2013039954A1
(fr)
|
2011-09-14 |
2013-03-21 |
Sanofi |
Anticorps anti-gitr
|
WO2013155223A1
(fr)
|
2012-04-10 |
2013-10-17 |
The Regents Of The University Of California |
Compositions et méthodes pour le traitement du cancer
|
JP6374384B2
(ja)
|
2012-08-07 |
2018-08-15 |
メルク パテント ゲゼルシャフト ミット ベシュレンクテル ハフツングMerck Patent Gesellschaft mit beschraenkter Haftung |
プロテインキナーゼ阻害剤としてのピリドピリミジン誘導体
|
WO2014143659A1
(fr)
|
2013-03-15 |
2014-09-18 |
Araxes Pharma Llc |
Inhibiteurs covalents irréversibles de la gtpase k-ras g12c
|
UY35464A
(es)
|
2013-03-15 |
2014-10-31 |
Araxes Pharma Llc |
Inhibidores covalentes de kras g12c.
|
WO2014152588A1
(fr)
|
2013-03-15 |
2014-09-25 |
Araxes Pharma Llc |
Inhibiteurs covalents de k-ras g12c
|
GB201312059D0
(en)
|
2013-07-05 |
2013-08-21 |
Univ Leuven Kath |
Novel GAK modulators
|
UA119971C2
(uk)
|
2013-10-10 |
2019-09-10 |
Араксіс Фарма Ллк |
Інгібітори g12c kras
|
JO3805B1
(ar)
|
2013-10-10 |
2021-01-31 |
Araxes Pharma Llc |
مثبطات كراس جي12سي
|
GB201320729D0
(en)
|
2013-11-25 |
2014-01-08 |
Cancer Rec Tech Ltd |
Therapeutic compounds and their use
|
SG11201605699QA
(en)
|
2014-01-20 |
2016-08-30 |
Cleave Biosciences Inc |
FUSED PYRIMIDINES AS INHIBITORS OF p97 COMPLEX
|
WO2016035008A1
(fr)
|
2014-09-04 |
2016-03-10 |
Lupin Limited |
Dérivés de pyridopyrimidine utilisés comme inhibiteurs de mek
|
JO3556B1
(ar)
|
2014-09-18 |
2020-07-05 |
Araxes Pharma Llc |
علاجات مدمجة لمعالجة السرطان
|
WO2016049565A1
(fr)
|
2014-09-25 |
2016-03-31 |
Araxes Pharma Llc |
Compositions et procédés pour inhiber la ras
|
US10011600B2
(en)
|
2014-09-25 |
2018-07-03 |
Araxes Pharma Llc |
Methods and compositions for inhibition of Ras
|
ES2826443T3
(es)
|
2014-09-25 |
2021-05-18 |
Araxes Pharma Llc |
Inhibidores de proteínas mutantes KRAS G12C
|
EA201792214A1
(ru)
|
2015-04-10 |
2018-01-31 |
Араксис Фарма Ллк |
Соединения замещенного хиназолина
|
US10428064B2
(en)
|
2015-04-15 |
2019-10-01 |
Araxes Pharma Llc |
Fused-tricyclic inhibitors of KRAS and methods of use thereof
|
CA2993013A1
(fr)
|
2015-07-22 |
2017-01-26 |
Araxes Pharma Llc |
Composes de quinazoline substitues et leur utilisation en tant qu'inhibiteurs de proteines kras, hras et/ou nras mutantes g12c
|
WO2017058805A1
(fr)
|
2015-09-28 |
2017-04-06 |
Araxes Pharma Llc |
Inhibiteurs de protéines kras portant la mutation g12c
|
EP3356339A1
(fr)
|
2015-09-28 |
2018-08-08 |
Araxes Pharma LLC |
Inhibiteurs de protéines mutantes kras g12c
|
EP3356353A1
(fr)
|
2015-09-28 |
2018-08-08 |
Araxes Pharma LLC |
Inhibiteurs de protéines kras portant la mutation g12c
|
US10882847B2
(en)
|
2015-09-28 |
2021-01-05 |
Araxes Pharma Llc |
Inhibitors of KRAS G12C mutant proteins
|
EP3356351A1
(fr)
|
2015-09-28 |
2018-08-08 |
Araxes Pharma LLC |
Inhibiteurs de protéines kras portant la mutation g12c
|
WO2017058807A1
(fr)
|
2015-09-28 |
2017-04-06 |
Araxes Pharma Llc |
Inhibiteurs de protéines kras portant la mutation g12c
|
US10975071B2
(en)
|
2015-09-28 |
2021-04-13 |
Araxes Pharma Llc |
Inhibitors of KRAS G12C mutant proteins
|
TW201726656A
(zh)
|
2015-11-16 |
2017-08-01 |
亞瑞克西斯製藥公司 |
包含經取代雜環基團之2-經取代喹唑啉化合物及其使用方法
|
WO2017100546A1
(fr)
|
2015-12-09 |
2017-06-15 |
Araxes Pharma Llc |
Procédés de préparation de dérivés de quinazoléine
|
US10822312B2
(en)
|
2016-03-30 |
2020-11-03 |
Araxes Pharma Llc |
Substituted quinazoline compounds and methods of use
|
CN109843856B
(zh)
|
2016-05-18 |
2023-05-02 |
米拉蒂治疗股份有限公司 |
Kras g12c抑制剂
|
US10646488B2
(en)
|
2016-07-13 |
2020-05-12 |
Araxes Pharma Llc |
Conjugates of cereblon binding compounds and G12C mutant KRAS, HRAS or NRAS protein modulating compounds and methods of use thereof
|
US10280172B2
(en)
|
2016-09-29 |
2019-05-07 |
Araxes Pharma Llc |
Inhibitors of KRAS G12C mutant proteins
|
EP3523289A1
(fr)
|
2016-10-07 |
2019-08-14 |
Araxes Pharma LLC |
Composés hétérocycliques en tant qu'inhibiteurs de ras et leurs procédés d'utilisation
|
SG10201913491PA
(en)
|
2016-12-22 |
2020-03-30 |
Amgen Inc |
Benzisothiazole, isothiazolo[3,4-b]pyridine, quinazoline, phthalazine, pyrido[2,3-d]pyridazine and pyrido[2,3-d]pyrimidine derivatives as kras g12c inhibitors for treating lung, pancreatic or colorectal cancer
|
JP2020505395A
(ja)
|
2017-01-26 |
2020-02-20 |
アラクセス ファーマ エルエルシー |
縮合n−複素環式化合物およびその使用方法
|
JOP20190272A1
(ar)
*
|
2017-05-22 |
2019-11-21 |
Amgen Inc |
مثبطات kras g12c وطرق لاستخدامها
|
CN110831933A
(zh)
|
2017-05-25 |
2020-02-21 |
亚瑞克西斯制药公司 |
喹唑啉衍生物作为突变kras、hras或nras的调节剂
|
MA50077A
(fr)
|
2017-09-08 |
2020-07-15 |
Amgen Inc |
Inhibiteurs de kras g12c et leurs procédés d'utilisation
|
JP7266043B2
(ja)
|
2018-05-04 |
2023-04-27 |
アムジエン・インコーポレーテツド |
KRas G12C阻害剤及びそれを使用する方法
|
WO2019213526A1
(fr)
|
2018-05-04 |
2019-11-07 |
Amgen Inc. |
Inhibiteurs de kras g12c et leurs procédés d'utilisation
|
CA3099045A1
(fr)
|
2018-05-10 |
2019-11-14 |
Amgen Inc. |
Inhibiteurs de kras g12c pour le traitement du cancer
|
MX2020012731A
(es)
|
2018-06-01 |
2021-02-22 |
Amgen Inc |
Inhibidores de kras g12c y metodos para su uso.
|
US20190375749A1
(en)
|
2018-06-11 |
2019-12-12 |
Amgen Inc. |
Kras g12c inhibitors and methods of using the same
|
WO2020050890A2
(fr)
|
2018-06-12 |
2020-03-12 |
Amgen Inc. |
Inhibiteurs de kras g12c et leurs procédés d'utilisation
|
EP3810608B1
(fr)
|
2018-06-21 |
2022-08-10 |
Janssen Pharmaceutica NV |
Composés pyrrolopyridines comme des inhibiteurs de oga
|
JP2021528404A
(ja)
|
2018-06-21 |
2021-10-21 |
ヤンセン ファーマシューティカ エヌ.ベー. |
Oga阻害剤化合物
|
JP7516029B2
(ja)
|
2018-11-16 |
2024-07-16 |
アムジエン・インコーポレーテツド |
Kras g12c阻害剤化合物の重要な中間体の改良合成法
|
AU2019384118A1
(en)
|
2018-11-19 |
2021-05-27 |
Amgen Inc. |
KRAS G12C inhibitors and methods of using the same
|
JP7377679B2
(ja)
|
2018-11-19 |
2023-11-10 |
アムジエン・インコーポレーテツド |
がん治療のためのkrasg12c阻害剤及び1種以上の薬学的に活性な追加の薬剤を含む併用療法
|
EP3738593A1
(fr)
|
2019-05-14 |
2020-11-18 |
Amgen, Inc |
Dosage d'inhibiteur de kras pour le traitement de cancers
|
US20220235045A1
(en)
|
2019-05-21 |
2022-07-28 |
Amgen Inc. |
Solid state forms
|
US11236091B2
(en)
|
2019-05-21 |
2022-02-01 |
Amgen Inc. |
Solid state forms
|
JP2022552873A
(ja)
|
2019-10-24 |
2022-12-20 |
アムジエン・インコーポレーテツド |
がんの治療におけるkras g12c及びkras g12d阻害剤として有用なピリドピリミジン誘導体
|
KR20220101125A
(ko)
|
2019-11-14 |
2022-07-19 |
암젠 인크 |
Kras g12c 억제제 화합물의 개선된 합성
|
WO2021097207A1
(fr)
|
2019-11-14 |
2021-05-20 |
Amgen Inc. |
Synthèse améliorée de composés inhibiteurs de kras g12c
|
WO2021126816A1
(fr)
|
2019-12-16 |
2021-06-24 |
Amgen Inc. |
Schéma posologique d'un inhibiteur du kras g12c
|
EP4153588A1
(fr)
|
2020-05-20 |
2023-03-29 |
Teva Pharmaceuticals International GmbH |
Formes solides d'amg-510 et leur procédé de préparation
|