ATE191218T1 - Rapamycin-derivate als immunosuppressoren - Google Patents

Rapamycin-derivate als immunosuppressoren

Info

Publication number
ATE191218T1
ATE191218T1 AT95903810T AT95903810T ATE191218T1 AT E191218 T1 ATE191218 T1 AT E191218T1 AT 95903810 T AT95903810 T AT 95903810T AT 95903810 T AT95903810 T AT 95903810T AT E191218 T1 ATE191218 T1 AT E191218T1
Authority
AT
Austria
Prior art keywords
pct
immunosuppressors
rapamycin derivatives
date jun
sec
Prior art date
Application number
AT95903810T
Other languages
English (en)
Inventor
Sylvain Cottens
Richard Sedrani
Original Assignee
Novartis Ag
Novartis Erfind Verwalt Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB939325800A external-priority patent/GB9325800D0/en
Priority claimed from GB939325802A external-priority patent/GB9325802D0/en
Priority claimed from GB9407138A external-priority patent/GB9407138D0/en
Priority claimed from GB9421982A external-priority patent/GB9421982D0/en
Application filed by Novartis Ag, Novartis Erfind Verwalt Gmbh filed Critical Novartis Ag
Application granted granted Critical
Publication of ATE191218T1 publication Critical patent/ATE191218T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/18—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1804—Compounds having Si-O-C linkages

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Immunology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Transplantation (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
AT95903810T 1993-12-17 1994-12-16 Rapamycin-derivate als immunosuppressoren ATE191218T1 (de)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
GB939325800A GB9325800D0 (en) 1993-12-17 1993-12-17 Organic compounds
GB939325802A GB9325802D0 (en) 1993-12-17 1993-12-17 Organic compounds
GB9407138A GB9407138D0 (en) 1994-04-11 1994-04-11 Organic compounds
GB9421982A GB9421982D0 (en) 1994-11-01 1994-11-01 Organic compounds
PCT/EP1994/004191 WO1995016691A1 (en) 1993-12-17 1994-12-16 Rapamycin derivatives useful as immunosuppressants

Publications (1)

Publication Number Publication Date
ATE191218T1 true ATE191218T1 (de) 2000-04-15

Family

ID=27451097

Family Applications (1)

Application Number Title Priority Date Filing Date
AT95903810T ATE191218T1 (de) 1993-12-17 1994-12-16 Rapamycin-derivate als immunosuppressoren

Country Status (21)

Country Link
US (1) US5912253A (de)
EP (1) EP0734389B1 (de)
JP (1) JP3745772B2 (de)
CN (1) CN1046944C (de)
AT (1) ATE191218T1 (de)
AU (1) AU687491B2 (de)
BR (1) BR9408323A (de)
CZ (1) CZ284650B6 (de)
DE (1) DE69423781T2 (de)
DK (1) DK0734389T3 (de)
ES (1) ES2146741T3 (de)
FI (1) FI962487A (de)
GR (1) GR3033545T3 (de)
HU (1) HUT74686A (de)
NO (1) NO962540L (de)
NZ (1) NZ277498A (de)
PL (1) PL314238A1 (de)
PT (1) PT734389E (de)
SG (1) SG64372A1 (de)
SK (1) SK78196A3 (de)
WO (1) WO1995016691A1 (de)

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