LU92433I2 - Olodatérol, ses isomères optiques individuels, mélanges d'énantiomères individuels ou de racémates, ses sels d'addition d'acide avec des acides pharmaceutiquement acceptables, ainsi que ses solvates et/ou ses hydrates, en particulier l'olodatérol et le chlorhydrate d'olodatérol - Google Patents

Olodatérol, ses isomères optiques individuels, mélanges d'énantiomères individuels ou de racémates, ses sels d'addition d'acide avec des acides pharmaceutiquement acceptables, ainsi que ses solvates et/ou ses hydrates, en particulier l'olodatérol et le chlorhydrate d'olodatérol

Info

Publication number
LU92433I2
LU92433I2 LU92433C LU92433C LU92433I2 LU 92433 I2 LU92433 I2 LU 92433I2 LU 92433 C LU92433 C LU 92433C LU 92433 C LU92433 C LU 92433C LU 92433 I2 LU92433 I2 LU 92433I2
Authority
LU
Luxembourg
Prior art keywords
olodaterol
olodatérol
racemates
solvates
hydrates
Prior art date
Application number
LU92433C
Other languages
English (en)
French (fr)
Original Assignee
Boehringer Ingelheim Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=32185709&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=LU92433(I2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma
Publication of LU92433I2 publication Critical patent/LU92433I2/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/538—1,4-Oxazines, e.g. morpholine ortho- or peri-condensed with carbocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/34—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings
    • C07D265/36—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings condensed with one six-membered ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicinal Preparation (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
LU92433C 2002-11-15 2014-04-22 Olodatérol, ses isomères optiques individuels, mélanges d'énantiomères individuels ou de racémates, ses sels d'addition d'acide avec des acides pharmaceutiquement acceptables, ainsi que ses solvates et/ou ses hydrates, en particulier l'olodatérol et le chlorhydrate d'olodatérol LU92433I2 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE10253282A DE10253282A1 (de) 2002-11-15 2002-11-15 Neue Arzneimittel zur Behandlung von chronisch obstruktiver Lungenerkrankung

Publications (1)

Publication Number Publication Date
LU92433I2 true LU92433I2 (fr) 2014-06-24

Family

ID=32185709

Family Applications (1)

Application Number Title Priority Date Filing Date
LU92433C LU92433I2 (fr) 2002-11-15 2014-04-22 Olodatérol, ses isomères optiques individuels, mélanges d'énantiomères individuels ou de racémates, ses sels d'addition d'acide avec des acides pharmaceutiquement acceptables, ainsi que ses solvates et/ou ses hydrates, en particulier l'olodatérol et le chlorhydrate d'olodatérol

Country Status (38)

Country Link
EP (2) EP1562603B3 (show.php)
JP (1) JP4317138B2 (show.php)
KR (1) KR101092247B1 (show.php)
CN (3) CN101735166A (show.php)
AR (2) AR041969A1 (show.php)
AT (1) ATE430569T1 (show.php)
AU (1) AU2003285326B2 (show.php)
BE (1) BE2014C016I2 (show.php)
BR (1) BRPI0316264B8 (show.php)
CA (1) CA2506082C (show.php)
CO (1) CO5570670A2 (show.php)
CY (2) CY1110500T1 (show.php)
DE (2) DE10253282A1 (show.php)
DK (1) DK1562603T3 (show.php)
EA (1) EA008665B1 (show.php)
EC (1) ECSP055774A (show.php)
ES (1) ES2326878T7 (show.php)
FR (1) FR14C0049I2 (show.php)
HR (1) HRP20050432B1 (show.php)
HU (1) HUS1400011I1 (show.php)
IL (1) IL167900A (show.php)
LT (1) LTC1562603I2 (show.php)
LU (1) LU92433I2 (show.php)
ME (1) ME00354B (show.php)
MX (1) MXPA05005081A (show.php)
MY (1) MY136034A (show.php)
NL (1) NL300650I2 (show.php)
NO (2) NO334314B1 (show.php)
NZ (1) NZ540661A (show.php)
PE (1) PE20040694A1 (show.php)
PL (1) PL212238B1 (show.php)
PT (1) PT1562603E (show.php)
RS (1) RS51607B (show.php)
SI (1) SI1562603T1 (show.php)
TW (1) TWI343812B (show.php)
UA (1) UA81276C2 (show.php)
WO (1) WO2004045618A2 (show.php)
ZA (1) ZA200502246B (show.php)

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HRP20050432B1 (en) 2012-01-31
JP2006508140A (ja) 2006-03-09
HUS1400011I1 (hu) 2022-02-28
TWI343812B (en) 2011-06-21
EP1562603B1 (de) 2009-05-06
RS51607B (sr) 2011-08-31
PL212238B1 (pl) 2012-08-31
PL375270A1 (en) 2005-11-28
EA008665B1 (ru) 2007-06-29
BRPI0316264B8 (pt) 2021-05-25
ME00354B (me) 2011-10-10
WO2004045618A2 (de) 2004-06-03
KR20050075013A (ko) 2005-07-19
LTC1562603I2 (lt) 2016-12-12
CA2506082C (en) 2011-06-21
SI1562603T1 (sl) 2009-10-31
AR087241A2 (es) 2014-03-12
FR14C0049I1 (show.php) 2014-08-08
NL300650I2 (nl) 2017-11-02
NO20052883L (no) 2005-06-14
CN1713914A (zh) 2005-12-28
KR101092247B1 (ko) 2011-12-12
CY2014032I2 (el) 2015-12-09
CN101735166A (zh) 2010-06-16
ATE430569T1 (de) 2009-05-15
EP1562603A2 (de) 2005-08-17
FR14C0049I2 (fr) 2015-07-24
UA81276C2 (en) 2007-12-25
JP4317138B2 (ja) 2009-08-19
BRPI0316264B1 (pt) 2019-04-09
CY2014032I1 (el) 2015-12-09
DE10253282A1 (de) 2004-05-27
HRP20050432A2 (en) 2006-06-30
CY1110500T1 (el) 2015-04-29
EP2025338A1 (de) 2009-02-18
IL167900A (en) 2013-06-27
TW200423943A (en) 2004-11-16
EA200500715A1 (ru) 2005-12-29
PT1562603E (pt) 2009-06-18
NZ540661A (en) 2007-12-21
EP1562603B3 (de) 2014-01-08
ECSP055774A (es) 2005-11-22
ES2326878T3 (es) 2009-10-21
DE50311502D1 (de) 2009-06-18
NO334314B1 (no) 2014-02-03
NO2014005I1 (no) 2014-03-10
WO2004045618A3 (de) 2004-09-30
ES2326878T7 (es) 2014-03-11
AU2003285326A1 (en) 2004-06-15
ZA200502246B (en) 2006-01-25
MEP53608A (en) 2011-05-10
AU2003285326B2 (en) 2009-06-04
CN101817800A (zh) 2010-09-01
BE2014C016I2 (show.php) 2023-03-07
CO5570670A2 (es) 2005-10-31
MXPA05005081A (es) 2005-07-01
BR0316264A (pt) 2005-10-11
AR041969A1 (es) 2005-06-01
PE20040694A1 (es) 2004-11-23
DK1562603T3 (da) 2009-09-07
MY136034A (en) 2008-07-31
CA2506082A1 (en) 2004-06-03
RS20050361A (sr) 2007-04-10

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