KR20030081378A - 강도가 개선된 사이클릭 뎁시펩타이드의 결정 변형체 - Google Patents
강도가 개선된 사이클릭 뎁시펩타이드의 결정 변형체 Download PDFInfo
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- KR20030081378A KR20030081378A KR10-2003-7009110A KR20037009110A KR20030081378A KR 20030081378 A KR20030081378 A KR 20030081378A KR 20037009110 A KR20037009110 A KR 20037009110A KR 20030081378 A KR20030081378 A KR 20030081378A
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- ZPWFUIUNWDIYCJ-UHFFFAOYSA-N propan-2-yl octadecanoate Chemical compound CCCCCCCCCCCCCCCCCC(=O)OC(C)C ZPWFUIUNWDIYCJ-UHFFFAOYSA-N 0.000 description 1
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K11/00—Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K11/02—Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof cyclic, e.g. valinomycins ; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/15—Depsipeptides; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Organic Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Tropical Medicine & Parasitology (AREA)
- Engineering & Computer Science (AREA)
- Gastroenterology & Hepatology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Immunology (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biochemistry (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10104362.7 | 2001-02-01 | ||
| DE10104362A DE10104362A1 (de) | 2001-02-01 | 2001-02-01 | Kristallmodifikation eines cyclischen Depsipeptids mit besserer Wirksamkeit |
| PCT/EP2002/000541 WO2002066048A1 (de) | 2001-02-01 | 2002-01-21 | Kristallmodifikation eines cyclischen depsipeptids mit besserer wirksamkeit |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020097006790A Division KR20090041451A (ko) | 2001-02-01 | 2002-01-21 | 강도가 개선된 사이클릭 뎁시펩타이드의 결정 변형체 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| KR20030081378A true KR20030081378A (ko) | 2003-10-17 |
Family
ID=7672376
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR10-2003-7009110A Ceased KR20030081378A (ko) | 2001-02-01 | 2002-01-21 | 강도가 개선된 사이클릭 뎁시펩타이드의 결정 변형체 |
| KR1020097006790A Ceased KR20090041451A (ko) | 2001-02-01 | 2002-01-21 | 강도가 개선된 사이클릭 뎁시펩타이드의 결정 변형체 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020097006790A Ceased KR20090041451A (ko) | 2001-02-01 | 2002-01-21 | 강도가 개선된 사이클릭 뎁시펩타이드의 결정 변형체 |
Country Status (27)
| Country | Link |
|---|---|
| US (1) | US20040115483A1 (https=) |
| EP (1) | EP1357932B1 (https=) |
| JP (1) | JP2004525111A (https=) |
| KR (2) | KR20030081378A (https=) |
| CN (1) | CN1278735C (https=) |
| AT (1) | ATE284703T1 (https=) |
| AU (1) | AU2002226415B2 (https=) |
| BR (1) | BRPI0206841B8 (https=) |
| CA (1) | CA2436832C (https=) |
| CR (1) | CR7039A (https=) |
| CZ (1) | CZ299564B6 (https=) |
| DE (2) | DE10104362A1 (https=) |
| EE (1) | EE05490B1 (https=) |
| ES (1) | ES2233805T3 (https=) |
| HR (1) | HRP20030635A2 (https=) |
| HU (1) | HU229229B1 (https=) |
| IL (2) | IL157026A0 (https=) |
| MX (1) | MXPA03006866A (https=) |
| NO (1) | NO331289B1 (https=) |
| NZ (1) | NZ527230A (https=) |
| PL (1) | PL213106B1 (https=) |
| PT (1) | PT1357932E (https=) |
| RU (1) | RU2300390C2 (https=) |
| SK (1) | SK286280B6 (https=) |
| UA (1) | UA74623C2 (https=) |
| WO (1) | WO2002066048A1 (https=) |
| ZA (1) | ZA200305864B (https=) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20080003546A1 (en) * | 2006-06-29 | 2008-01-03 | Dunbar Kimberly L | Animated digital charted yarncraft instruction |
| LT3298027T (lt) | 2015-05-20 | 2021-08-10 | Boehringer Ingelheim Animal Health USA Inc. | Antihelmintiniai depsipeptido junginiai |
| RU2715556C2 (ru) | 2015-12-28 | 2020-03-02 | Мериал, Инк. | Противогельминтные депсипептидные соединения |
| CA3044038A1 (en) | 2016-11-16 | 2018-05-24 | Boehringer Ingelheim Animal Health USA Inc. | Anthelmintic depsipeptide compounds |
| CN114262303A (zh) * | 2022-01-04 | 2022-04-01 | 丽珠集团福州福兴医药有限公司 | 一种艾默德斯的单晶型ii及其制备方法 |
| CN114195732A (zh) * | 2022-01-04 | 2022-03-18 | 丽珠集团福州福兴医药有限公司 | 一种艾默德斯的单晶型iii及其制备方法 |
| CN114989110A (zh) * | 2022-07-13 | 2022-09-02 | 丽珠集团福州福兴医药有限公司 | 单晶型ⅳ的艾默德斯及其制备方法 |
| CN115010680A (zh) * | 2022-07-13 | 2022-09-06 | 丽珠集团福州福兴医药有限公司 | 单晶型i的艾默德斯及其制备方法 |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB2096907A (en) * | 1981-04-22 | 1982-10-27 | Exxon Research Engineering Co | Distillation column with steam stripping |
| ES2166359T3 (es) * | 1992-03-17 | 2002-04-16 | Fujisawa Pharmaceutical Co | Derivado de depsipeptido, su produccion y uso. |
| DE4317458A1 (de) * | 1992-06-11 | 1993-12-16 | Bayer Ag | Verwendung von cyclischen Depsipeptiden mit 18 Ringatomen zur Bekämpfung von Endoparasiten, neue cyclische Depsipeptide mit 18 Ringatomen und Verfahren zu ihrer Herstellung |
| DE4400464A1 (de) * | 1994-01-11 | 1995-07-13 | Bayer Ag | Endoparasitizide Mittel |
| WO1997002256A1 (en) * | 1995-06-30 | 1997-01-23 | Fujisawa Pharmaceutical Co., Ltd. | Depsipeptide derivative, process for production thereof, and novel intermediate therefor |
| KR19990063676A (ko) * | 1995-09-22 | 1999-07-26 | 빌프리더 하이더 | 신규한 환상 데프시펩티드 pf1022 유도체 |
| BR9815292A (pt) * | 1997-11-10 | 2000-10-24 | Fujisawa Pharmaceutical Co | Cristal de derivado de despsipeptìdeo e método para a sua produção |
| DE10008128A1 (de) * | 2000-02-22 | 2001-08-23 | Bayer Ag | Endoparasitizide Mittel |
| DE10031044A1 (de) * | 2000-06-26 | 2002-01-03 | Bayer Ag | Endoparasitizide Mittel zur freiwilligen oralen Aufnahme durch Tiere |
-
2001
- 2001-02-01 DE DE10104362A patent/DE10104362A1/de not_active Withdrawn
-
2002
- 2002-01-21 JP JP2002565606A patent/JP2004525111A/ja active Pending
- 2002-01-21 HR HR20030635A patent/HRP20030635A2/hr not_active Application Discontinuation
- 2002-01-21 MX MXPA03006866A patent/MXPA03006866A/es active IP Right Grant
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