ATE284703T1 - Kristallmodifikation eines cyclischen depsipeptids mit besserer wirksamkeit - Google Patents

Kristallmodifikation eines cyclischen depsipeptids mit besserer wirksamkeit

Info

Publication number
ATE284703T1
ATE284703T1 AT02716073T AT02716073T ATE284703T1 AT E284703 T1 ATE284703 T1 AT E284703T1 AT 02716073 T AT02716073 T AT 02716073T AT 02716073 T AT02716073 T AT 02716073T AT E284703 T1 ATE284703 T1 AT E284703T1
Authority
AT
Austria
Prior art keywords
cyclic depsipeptide
crystal modification
better effectiveness
effectiveness
better
Prior art date
Application number
AT02716073T
Other languages
German (de)
English (en)
Inventor
Jochen Kalbe
Michael Traeubel
Achim Harder
Samson-Himmelstjerna Georg Von
Original Assignee
Bayer Healthcare Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Healthcare Ag filed Critical Bayer Healthcare Ag
Application granted granted Critical
Publication of ATE284703T1 publication Critical patent/ATE284703T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K11/00Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K11/02Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof cyclic, e.g. valinomycins ; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/15Depsipeptides; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Organic Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Engineering & Computer Science (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Immunology (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
AT02716073T 2001-02-01 2002-01-21 Kristallmodifikation eines cyclischen depsipeptids mit besserer wirksamkeit ATE284703T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10104362A DE10104362A1 (de) 2001-02-01 2001-02-01 Kristallmodifikation eines cyclischen Depsipeptids mit besserer Wirksamkeit
PCT/EP2002/000541 WO2002066048A1 (de) 2001-02-01 2002-01-21 Kristallmodifikation eines cyclischen depsipeptids mit besserer wirksamkeit

Publications (1)

Publication Number Publication Date
ATE284703T1 true ATE284703T1 (de) 2005-01-15

Family

ID=7672376

Family Applications (1)

Application Number Title Priority Date Filing Date
AT02716073T ATE284703T1 (de) 2001-02-01 2002-01-21 Kristallmodifikation eines cyclischen depsipeptids mit besserer wirksamkeit

Country Status (27)

Country Link
US (1) US20040115483A1 (https=)
EP (1) EP1357932B1 (https=)
JP (1) JP2004525111A (https=)
KR (2) KR20030081378A (https=)
CN (1) CN1278735C (https=)
AT (1) ATE284703T1 (https=)
AU (1) AU2002226415B2 (https=)
BR (1) BRPI0206841B8 (https=)
CA (1) CA2436832C (https=)
CR (1) CR7039A (https=)
CZ (1) CZ299564B6 (https=)
DE (2) DE10104362A1 (https=)
EE (1) EE05490B1 (https=)
ES (1) ES2233805T3 (https=)
HR (1) HRP20030635A2 (https=)
HU (1) HU229229B1 (https=)
IL (2) IL157026A0 (https=)
MX (1) MXPA03006866A (https=)
NO (1) NO331289B1 (https=)
NZ (1) NZ527230A (https=)
PL (1) PL213106B1 (https=)
PT (1) PT1357932E (https=)
RU (1) RU2300390C2 (https=)
SK (1) SK286280B6 (https=)
UA (1) UA74623C2 (https=)
WO (1) WO2002066048A1 (https=)
ZA (1) ZA200305864B (https=)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20080003546A1 (en) * 2006-06-29 2008-01-03 Dunbar Kimberly L Animated digital charted yarncraft instruction
LT3298027T (lt) 2015-05-20 2021-08-10 Boehringer Ingelheim Animal Health USA Inc. Antihelmintiniai depsipeptido junginiai
RU2715556C2 (ru) 2015-12-28 2020-03-02 Мериал, Инк. Противогельминтные депсипептидные соединения
CA3044038A1 (en) 2016-11-16 2018-05-24 Boehringer Ingelheim Animal Health USA Inc. Anthelmintic depsipeptide compounds
CN114262303A (zh) * 2022-01-04 2022-04-01 丽珠集团福州福兴医药有限公司 一种艾默德斯的单晶型ii及其制备方法
CN114195732A (zh) * 2022-01-04 2022-03-18 丽珠集团福州福兴医药有限公司 一种艾默德斯的单晶型iii及其制备方法
CN114989110A (zh) * 2022-07-13 2022-09-02 丽珠集团福州福兴医药有限公司 单晶型ⅳ的艾默德斯及其制备方法
CN115010680A (zh) * 2022-07-13 2022-09-06 丽珠集团福州福兴医药有限公司 单晶型i的艾默德斯及其制备方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2096907A (en) * 1981-04-22 1982-10-27 Exxon Research Engineering Co Distillation column with steam stripping
ES2166359T3 (es) * 1992-03-17 2002-04-16 Fujisawa Pharmaceutical Co Derivado de depsipeptido, su produccion y uso.
DE4317458A1 (de) * 1992-06-11 1993-12-16 Bayer Ag Verwendung von cyclischen Depsipeptiden mit 18 Ringatomen zur Bekämpfung von Endoparasiten, neue cyclische Depsipeptide mit 18 Ringatomen und Verfahren zu ihrer Herstellung
DE4400464A1 (de) * 1994-01-11 1995-07-13 Bayer Ag Endoparasitizide Mittel
WO1997002256A1 (en) * 1995-06-30 1997-01-23 Fujisawa Pharmaceutical Co., Ltd. Depsipeptide derivative, process for production thereof, and novel intermediate therefor
KR19990063676A (ko) * 1995-09-22 1999-07-26 빌프리더 하이더 신규한 환상 데프시펩티드 pf1022 유도체
BR9815292A (pt) * 1997-11-10 2000-10-24 Fujisawa Pharmaceutical Co Cristal de derivado de despsipeptìdeo e método para a sua produção
DE10008128A1 (de) * 2000-02-22 2001-08-23 Bayer Ag Endoparasitizide Mittel
DE10031044A1 (de) * 2000-06-26 2002-01-03 Bayer Ag Endoparasitizide Mittel zur freiwilligen oralen Aufnahme durch Tiere

Also Published As

Publication number Publication date
BRPI0206841B1 (pt) 2018-02-14
PL362389A1 (en) 2004-11-02
KR20030081378A (ko) 2003-10-17
MXPA03006866A (es) 2004-05-31
PT1357932E (pt) 2005-04-29
NO20033413L (no) 2003-09-26
RU2300390C2 (ru) 2007-06-10
US20040115483A1 (en) 2004-06-17
UA74623C2 (en) 2006-01-16
AU2002226415B2 (en) 2007-03-22
CZ299564B6 (cs) 2008-09-03
EE05490B1 (et) 2011-12-15
HUP0302880A3 (en) 2005-05-30
CZ20032063A3 (cs) 2003-11-12
EP1357932B1 (de) 2004-12-15
CN1592631A (zh) 2005-03-09
CR7039A (es) 2004-06-08
NZ527230A (en) 2005-04-29
BR0206841A (pt) 2004-02-25
CN1278735C (zh) 2006-10-11
WO2002066048A1 (de) 2002-08-29
PL213106B1 (pl) 2013-01-31
BRPI0206841B8 (pt) 2021-05-25
NO331289B1 (no) 2011-11-21
WO2002066048A8 (de) 2003-11-20
HUP0302880A2 (hu) 2003-12-29
DE10104362A1 (de) 2002-08-08
JP2004525111A (ja) 2004-08-19
SK286280B6 (sk) 2008-06-06
IL157026A (en) 2010-11-30
SK9882003A3 (en) 2003-12-02
HU229229B1 (en) 2013-09-30
ES2233805T3 (es) 2005-06-16
CA2436832A1 (en) 2002-08-29
HK1075013A1 (en) 2005-12-02
EP1357932A1 (de) 2003-11-05
DE50201777D1 (de) 2005-01-20
NO20033413D0 (no) 2003-07-30
CA2436832C (en) 2013-06-11
KR20090041451A (ko) 2009-04-28
IL157026A0 (en) 2004-02-08
RU2003126589A (ru) 2005-02-27
HRP20030635A2 (en) 2005-10-31
EE200300365A (et) 2003-10-15
ZA200305864B (en) 2004-08-27

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