ATE425973T1 - Depsipeptid-derivat, verfahren zu dessen herstellung und zwischenprodukt dafur - Google Patents
Depsipeptid-derivat, verfahren zu dessen herstellung und zwischenprodukt dafurInfo
- Publication number
- ATE425973T1 ATE425973T1 AT96918897T AT96918897T ATE425973T1 AT E425973 T1 ATE425973 T1 AT E425973T1 AT 96918897 T AT96918897 T AT 96918897T AT 96918897 T AT96918897 T AT 96918897T AT E425973 T1 ATE425973 T1 AT E425973T1
- Authority
- AT
- Austria
- Prior art keywords
- production
- depsipeptide derivative
- depsipeptide
- derivative
- chem
- Prior art date
Links
- 238000004519 manufacturing process Methods 0.000 title abstract 2
- OHRURASPPZQGQM-GCCNXGTGSA-N romidepsin Chemical class O1C(=O)[C@H](C(C)C)NC(=O)C(=C/C)/NC(=O)[C@H]2CSSCC\C=C\[C@@H]1CC(=O)N[C@H](C(C)C)C(=O)N2 OHRURASPPZQGQM-GCCNXGTGSA-N 0.000 title abstract 2
- 230000000507 anthelmentic effect Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D273/00—Heterocyclic compounds containing rings having nitrogen and oxygen atoms as the only ring hetero atoms, not provided for by groups C07D261/00 - C07D271/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Peptides Or Proteins (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Micro-Organisms Or Cultivation Processes Thereof (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP18788995 | 1995-06-30 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE425973T1 true ATE425973T1 (de) | 2009-04-15 |
Family
ID=16213973
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT96918897T ATE425973T1 (de) | 1995-06-30 | 1996-06-24 | Depsipeptid-derivat, verfahren zu dessen herstellung und zwischenprodukt dafur |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US5856436A (de) |
| EP (1) | EP0872481B1 (de) |
| JP (1) | JP3985050B2 (de) |
| CN (2) | CN1071323C (de) |
| AT (1) | ATE425973T1 (de) |
| DE (1) | DE69637876D1 (de) |
| ES (1) | ES2322678T3 (de) |
| PT (1) | PT872481E (de) |
| WO (1) | WO1997002256A1 (de) |
Families Citing this family (25)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6262058B1 (en) * | 1996-03-11 | 2001-07-17 | Syngenta Crop Protection, Inc. | Pyrimidin-4-one derivatives as pesticide |
| PT953563E (pt) | 1996-10-07 | 2003-08-29 | Fujisawa Pharmaceutical Co | Processo para a preparacao de derivados de depsipeptidos e novos compostos intermediarios para essa preparacao |
| ATE221055T1 (de) * | 1997-11-10 | 2002-08-15 | Fujisawa Pharmaceutical Co | Kristall eines depsipeptid-derivates und verfahren zu seiner herstellung |
| DE19962147A1 (de) * | 1999-12-22 | 2001-06-28 | Bayer Ag | Schädlingsbekämpfungsmittel / PF 1022-221 |
| DE10031044A1 (de) * | 2000-06-26 | 2002-01-03 | Bayer Ag | Endoparasitizide Mittel zur freiwilligen oralen Aufnahme durch Tiere |
| DE10104362A1 (de) * | 2001-02-01 | 2002-08-08 | Bayer Ag | Kristallmodifikation eines cyclischen Depsipeptids mit besserer Wirksamkeit |
| CN1315837C (zh) * | 2002-11-04 | 2007-05-16 | 杭州博大药物研究所 | 藤黄酸类化合物的盐,其制备方法和以该盐为活性成份的药物组合物 |
| DE102004055316A1 (de) * | 2004-11-16 | 2006-05-18 | Bayer Healthcare Ag | Verhinderung vertikaler Endoparasiten-Infektionen |
| JP2008520682A (ja) * | 2004-11-17 | 2008-06-19 | ザ ユニヴァーシティー オヴ シカゴ | ヒストンデアセチラーゼ阻害剤およびその使用方法 |
| DE102008022520A1 (de) | 2008-05-07 | 2009-11-12 | Bayer Animal Health Gmbh | Feste Arzneimittelformulierung mit verzögerter Freisetzung |
| DE102008030764A1 (de) | 2008-06-28 | 2009-12-31 | Bayer Animal Health Gmbh | Kombination von Amidin-Derivaten mit cyclischen Depsipeptiden |
| DE102008031284A1 (de) * | 2008-07-02 | 2010-01-07 | Bayer Schering Pharma Aktiengesellschaft | Neue Bekämpfungsmöglichkeit der Giardiose |
| DE102008031283A1 (de) | 2008-07-02 | 2010-01-07 | Bayer Schering Pharma Aktiengesellschaft | Neue Bekämpfungsmöglichkeit von durch Trichomonadida hervorgerufenen Krankheiten |
| DE102009012423A1 (de) | 2009-03-10 | 2010-09-16 | Bayer Animal Health Gmbh | Zubereitung auf Ölbasis |
| DE102010064245A1 (de) | 2010-12-28 | 2012-06-28 | Bayer Animal Health Gmbh | Makrocylischen Lactone und deren Verwendung und deren Kombinationen mit anderen Wirkstoffen |
| WO2012028556A1 (en) | 2010-08-31 | 2012-03-08 | Bayer Animal Health Gmbh | Macrocyclic lactones and their use and their combinations with other active substances |
| CN107835818B (zh) | 2015-05-20 | 2022-04-29 | 勃林格殷格翰动物保健美国公司 | 驱虫缩酚酸肽化合物 |
| CN105613526A (zh) * | 2016-02-24 | 2016-06-01 | 燕素琴 | 一种防治林业害虫杨树天牛的药膏 |
| EP3541789A1 (de) | 2016-11-16 | 2019-09-25 | Boehringer Ingelheim Animal Health USA Inc. | Anthelmintische depsipeptidverbindungen |
| JP7164608B2 (ja) | 2017-11-29 | 2022-11-01 | ゾエティス・サービシーズ・エルエルシー | 内部寄生性デプシペプチド |
| EP3790876B1 (de) | 2018-05-10 | 2025-04-30 | Zoetis Services LLC | Endoparasitische depsipeptide |
| CN114195732A (zh) * | 2022-01-04 | 2022-03-18 | 丽珠集团福州福兴医药有限公司 | 一种艾默德斯的单晶型iii及其制备方法 |
| CN114262303A (zh) * | 2022-01-04 | 2022-04-01 | 丽珠集团福州福兴医药有限公司 | 一种艾默德斯的单晶型ii及其制备方法 |
| CN115010680A (zh) * | 2022-07-13 | 2022-09-06 | 丽珠集团福州福兴医药有限公司 | 单晶型i的艾默德斯及其制备方法 |
| CN114989110A (zh) * | 2022-07-13 | 2022-09-02 | 丽珠集团福州福兴医药有限公司 | 单晶型ⅳ的艾默德斯及其制备方法 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2132199C (en) * | 1992-03-17 | 2000-01-18 | Hitoshi Nishiyama | Depsipeptide derivative, production thereof and use thereof |
| CN1073560C (zh) * | 1993-02-19 | 2001-10-24 | 明治制果株式会社 | 环缩酚酸肽pf1022衍生物 |
| US5646244A (en) * | 1993-09-06 | 1997-07-08 | Fujisawa Pharmaceutical Co., Ltd. | Cyclodepsipeptide compound |
| JPH07233068A (ja) * | 1993-12-27 | 1995-09-05 | Meiji Seika Kaisha Ltd | 高コレステロール血症、高脂血症又は動脈硬化症の治療薬 |
-
1996
- 1996-06-24 CN CN96195073A patent/CN1071323C/zh not_active Expired - Lifetime
- 1996-06-24 DE DE69637876T patent/DE69637876D1/de not_active Expired - Lifetime
- 1996-06-24 US US08/973,718 patent/US5856436A/en not_active Expired - Lifetime
- 1996-06-24 EP EP96918897A patent/EP0872481B1/de not_active Expired - Lifetime
- 1996-06-24 PT PT96918897T patent/PT872481E/pt unknown
- 1996-06-24 ES ES96918897T patent/ES2322678T3/es not_active Expired - Lifetime
- 1996-06-24 AT AT96918897T patent/ATE425973T1/de not_active IP Right Cessation
- 1996-06-24 WO PCT/JP1996/001748 patent/WO1997002256A1/ja not_active Ceased
- 1996-06-24 JP JP50497997A patent/JP3985050B2/ja not_active Expired - Lifetime
- 1996-06-24 CN CNB001353926A patent/CN1162409C/zh not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| EP0872481B1 (de) | 2009-03-18 |
| EP0872481A1 (de) | 1998-10-21 |
| CN1189159A (zh) | 1998-07-29 |
| DE69637876D1 (de) | 2009-04-30 |
| EP0872481A4 (de) | 2001-04-11 |
| US5856436A (en) | 1999-01-05 |
| PT872481E (pt) | 2009-05-20 |
| WO1997002256A1 (en) | 1997-01-23 |
| JP3985050B2 (ja) | 2007-10-03 |
| ES2322678T3 (es) | 2009-06-24 |
| CN1162409C (zh) | 2004-08-18 |
| CN1309124A (zh) | 2001-08-22 |
| CN1071323C (zh) | 2001-09-19 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |