KR20000036066A - 압출성형에 의한 고상 제형의 제조 방법 - Google Patents
압출성형에 의한 고상 제형의 제조 방법 Download PDFInfo
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- KR20000036066A KR20000036066A KR1019997002072A KR19997002072A KR20000036066A KR 20000036066 A KR20000036066 A KR 20000036066A KR 1019997002072 A KR1019997002072 A KR 1019997002072A KR 19997002072 A KR19997002072 A KR 19997002072A KR 20000036066 A KR20000036066 A KR 20000036066A
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- MYPYJXKWCTUITO-LYRMYLQWSA-N vancomycin Chemical compound O([C@@H]1[C@@H](O)[C@H](O)[C@@H](CO)O[C@H]1OC1=C2C=C3C=C1OC1=CC=C(C=C1Cl)[C@@H](O)[C@H](C(N[C@@H](CC(N)=O)C(=O)N[C@H]3C(=O)N[C@H]1C(=O)N[C@H](C(N[C@@H](C3=CC(O)=CC(O)=C3C=3C(O)=CC=C1C=3)C(O)=O)=O)[C@H](O)C1=CC=C(C(=C1)Cl)O2)=O)NC(=O)[C@@H](CC(C)C)NC)[C@H]1C[C@](C)(N)[C@H](O)[C@H](C)O1 MYPYJXKWCTUITO-LYRMYLQWSA-N 0.000 description 1
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61J—CONTAINERS SPECIALLY ADAPTED FOR MEDICAL OR PHARMACEUTICAL PURPOSES; DEVICES OR METHODS SPECIALLY ADAPTED FOR BRINGING PHARMACEUTICAL PRODUCTS INTO PARTICULAR PHYSICAL OR ADMINISTERING FORMS; DEVICES FOR ADMINISTERING FOOD OR MEDICINES ORALLY; BABY COMFORTERS; DEVICES FOR RECEIVING SPITTLE
- A61J3/00—Devices or methods specially adapted for bringing pharmaceutical products into particular physical or administering forms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2095—Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19637479A DE19637479A1 (de) | 1996-09-13 | 1996-09-13 | Verfahren zur Herstellung fester pharmazeutischer Formen |
| DE19637479.0 | 1996-09-13 | ||
| DE19734011.3 | 1997-08-06 | ||
| DE19734011A DE19734011A1 (de) | 1997-08-06 | 1997-08-06 | Verfahren zur Herstellung fester pharmazeutischer Formen |
Publications (1)
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| KR20000036066A true KR20000036066A (ko) | 2000-06-26 |
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| EP (1) | EP0930875B1 (enExample) |
| JP (1) | JP4975894B2 (enExample) |
| KR (1) | KR20000036066A (enExample) |
| CN (1) | CN1230109A (enExample) |
| AT (1) | ATE239452T1 (enExample) |
| AU (1) | AU720535B2 (enExample) |
| BR (1) | BR9711777A (enExample) |
| CA (1) | CA2265532C (enExample) |
| CZ (1) | CZ82999A3 (enExample) |
| DE (1) | DE59710059D1 (enExample) |
| DK (1) | DK0930875T3 (enExample) |
| ES (1) | ES2199373T3 (enExample) |
| HR (1) | HRP970485A2 (enExample) |
| IL (1) | IL128672A0 (enExample) |
| SK (1) | SK26099A3 (enExample) |
| TR (1) | TR199900563T2 (enExample) |
| TW (1) | TW474824B (enExample) |
| WO (1) | WO1998010752A2 (enExample) |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| KR101417892B1 (ko) * | 2006-03-10 | 2014-07-16 | 아비에 도이치란트 게엠베하 운트 콤파니 카게 | 활성 성분의 고체 분산체를 제조하는 방법 |
| KR102757752B1 (ko) | 2024-01-31 | 2025-01-21 | (주) 제이아리 | 강성재질 성형틀 기반의 고형 제형 흡습제 제조 장비 |
| KR20250119038A (ko) | 2024-01-31 | 2025-08-07 | 주식회사 이엔케이글로벌 | 신축성재질 성형틀 기반의 고흡수성 고형 제형 흡습제 제조 장비 |
| KR20250120088A (ko) | 2024-02-01 | 2025-08-08 | (주) 제이아리 | 고흡수성 고형 제형 흡습제 제조 장비 |
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| US20040185099A1 (en) * | 2000-01-20 | 2004-09-23 | Biovail Laboratories, Inc. | Multiparticulate bisoprolol formulation |
| EP1284729A4 (en) * | 2000-04-13 | 2007-12-19 | Mayo Foundation | A- (BETA) -42 DECREASING MEDICINAL PRODUCTS |
| DE10026698A1 (de) * | 2000-05-30 | 2001-12-06 | Basf Ag | Selbstemulgierende Wirkstoffformulierung und Verwendung dieser Formulierung |
| GB0106469D0 (en) * | 2001-03-15 | 2001-05-02 | Syngenta Ltd | Solid formulation |
| FR2823974B1 (fr) * | 2001-04-25 | 2004-10-15 | Pf Medicament | Pastille medicamenteuse a liberation lente du principe actif |
| GB0113841D0 (en) * | 2001-06-07 | 2001-08-01 | Boots Co Plc | Therapeutic agents |
| WO2003000235A1 (en) * | 2001-06-22 | 2003-01-03 | Pfizer Products Inc. | Pharmaceutical compositions of dispersions of drugs and neutral polymers |
| US20030091633A1 (en) * | 2001-11-15 | 2003-05-15 | John Kelly | Methods and compositions for use of (S)-bisoprolol |
| US20030118652A1 (en) * | 2001-11-15 | 2003-06-26 | John Kelly | Methods and compositions for use of (S)-bisoprolol |
| WO2004071431A2 (en) * | 2003-02-05 | 2004-08-26 | Myriad Genetics, Inc. | Method and composition for treating neurodegenerative disorders |
| EP1624859A4 (en) * | 2003-05-06 | 2010-06-23 | Bpsi Holdings Inc | METHOD FOR PRODUCING THERMOFORMED COMPOSITIONS WITH ACRYLIC POLYMER BINDERS, PHARMACEUTICAL DOSAGE FORMS, AND METHOD FOR THE PRODUCTION THEREOF |
| CA2532207A1 (en) * | 2003-07-11 | 2005-07-21 | Myriad Genetics, Inc. | Pharmaceutical methods, dosing regimes and dosage forms for the treatment of alzheimer's disease |
| US8025899B2 (en) | 2003-08-28 | 2011-09-27 | Abbott Laboratories | Solid pharmaceutical dosage form |
| US8377952B2 (en) | 2003-08-28 | 2013-02-19 | Abbott Laboratories | Solid pharmaceutical dosage formulation |
| JP2007513147A (ja) * | 2003-12-04 | 2007-05-24 | ファイザー・プロダクツ・インク | 押し出し機を使用して、好ましくはポロキサマーとグリセリドを含有する多粒子結晶性医薬組成物を製造するための噴霧凝結方法 |
| WO2005053639A2 (en) * | 2003-12-04 | 2005-06-16 | Pfizer Products Inc. | Controlled release multiparticulates formed with dissolution enhancers |
| WO2005053652A1 (en) | 2003-12-04 | 2005-06-16 | Pfizer Products Inc. | Multiparticulate crystalline drug compositions containing a poloxamer and a glyceride |
| DE602004014805D1 (de) * | 2003-12-04 | 2008-08-14 | Pfizer Prod Inc | Verfahren zur herstellung von pharmazeutischen multiteilchenförmigen produkten |
| US6984403B2 (en) * | 2003-12-04 | 2006-01-10 | Pfizer Inc. | Azithromycin dosage forms with reduced side effects |
| CA2547597A1 (en) * | 2003-12-04 | 2005-06-16 | Pfizer Products Inc. | Multiparticulate compositions with improved stability |
| KR20080064209A (ko) * | 2003-12-04 | 2008-07-08 | 화이자 프로덕츠 인코포레이티드 | 바람직하게는 폴록사머와 글리세라이드를 함유하는다미립자 아지트로마이신 조성물의 제조를 위해 압출기를사용하는 분무응결 방법 |
| CN1889933A (zh) * | 2003-12-04 | 2007-01-03 | 辉瑞产品公司 | 由基于液体的工艺制备的阿奇霉素多颗粒剂型 |
| WO2006001877A2 (en) * | 2004-04-13 | 2006-01-05 | Myriad Genetics, Inc. | Combination treatment for neurodegenerative disorders comprising r-flurbiprofen |
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| WO2006020852A2 (en) * | 2004-08-11 | 2006-02-23 | Myriad Genetics, Inc. | Pharmaceutical composition and method for treating neurodegenerative disorders |
| WO2006020850A2 (en) * | 2004-08-11 | 2006-02-23 | Myriad Genetics, Inc. | Pharmaceutical composition and method for treating neurodegenerative disorders |
| BRPI0514303A (pt) * | 2004-08-11 | 2008-06-10 | Myriad Genetics Inc | composição farmacêutica e método para tratar distúrbios neurodegenerativos |
| US7799744B2 (en) * | 2005-03-09 | 2010-09-21 | Halliburton Energy Services, Inc. | Polymer coated particulates |
| JP5232644B2 (ja) * | 2005-07-05 | 2013-07-10 | アボット ゲーエムベーハー ウント コンパニー カーゲー | 固形又は半固形マトリックスを含む組成物及び剤形 |
| CA2615063A1 (en) * | 2005-07-22 | 2007-02-01 | Myriad Genetics, Inc. | High drug load formulations and dosage forms |
| WO2008006099A2 (en) * | 2006-07-07 | 2008-01-10 | Myriad Genetics, Inc. | Treatment of psychiatric disorders |
| AU2007287793A1 (en) * | 2006-08-23 | 2008-02-28 | Bayer Cropscience Ag | Formulations for the controlled release of agrochemical active agents |
| US8399007B2 (en) * | 2006-12-05 | 2013-03-19 | Landec Corporation | Method for formulating a controlled-release pharmaceutical formulation |
| US20090269403A1 (en) * | 2008-04-24 | 2009-10-29 | Shaked Ze Ev | Oral contraceptive dosage forms and methods of making such dosage forms |
| US20160113906A1 (en) | 2014-09-19 | 2016-04-28 | Board Of Regents, The University Of Texas System | Methods of preparing extrudates |
| CN108421497A (zh) * | 2018-04-03 | 2018-08-21 | 杨高品 | 药物连续化制粒的生产工艺和设备 |
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-
1997
- 1997-09-10 HR HR19734011.3A patent/HRP970485A2/xx not_active Application Discontinuation
- 1997-09-10 TW TW086113103A patent/TW474824B/zh active
- 1997-09-11 CA CA002265532A patent/CA2265532C/en not_active Expired - Lifetime
- 1997-09-11 CZ CZ99829A patent/CZ82999A3/cs unknown
- 1997-09-11 BR BR9711777A patent/BR9711777A/pt not_active Application Discontinuation
- 1997-09-11 AU AU43846/97A patent/AU720535B2/en not_active Ceased
- 1997-09-11 US US09/254,558 patent/US6221368B1/en not_active Expired - Lifetime
- 1997-09-11 KR KR1019997002072A patent/KR20000036066A/ko not_active Withdrawn
- 1997-09-11 CN CN97197941A patent/CN1230109A/zh active Pending
- 1997-09-11 DE DE59710059T patent/DE59710059D1/de not_active Expired - Lifetime
- 1997-09-11 EP EP97942022A patent/EP0930875B1/de not_active Expired - Lifetime
- 1997-09-11 WO PCT/EP1997/004984 patent/WO1998010752A2/de not_active Ceased
- 1997-09-11 ES ES97942022T patent/ES2199373T3/es not_active Expired - Lifetime
- 1997-09-11 SK SK260-99A patent/SK26099A3/sk unknown
- 1997-09-11 AT AT97942022T patent/ATE239452T1/de active
- 1997-09-11 JP JP51302098A patent/JP4975894B2/ja not_active Expired - Fee Related
- 1997-09-11 TR TR1999/00563T patent/TR199900563T2/xx unknown
- 1997-09-11 DK DK97942022T patent/DK0930875T3/da active
- 1997-09-11 IL IL12867297A patent/IL128672A0/xx unknown
Cited By (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR101417892B1 (ko) * | 2006-03-10 | 2014-07-16 | 아비에 도이치란트 게엠베하 운트 콤파니 카게 | 활성 성분의 고체 분산체를 제조하는 방법 |
| KR101453399B1 (ko) * | 2006-03-10 | 2014-10-22 | 아비에 도이치란트 게엠베하 운트 콤파니 카게 | 활성 성분의 고체 분산체를 제조하는 개선된 방법 |
| US9205027B2 (en) | 2006-03-10 | 2015-12-08 | Abbvie Deutschland Gmbh & Co Kg | Process for producing a solid dispersion of an active ingredient |
| US9414992B2 (en) | 2006-03-10 | 2016-08-16 | Abbvie Deutschland Gmbh & Co Kg | Process for producing a solid dispersion of an active ingredient |
| KR102757752B1 (ko) | 2024-01-31 | 2025-01-21 | (주) 제이아리 | 강성재질 성형틀 기반의 고형 제형 흡습제 제조 장비 |
| KR20250119038A (ko) | 2024-01-31 | 2025-08-07 | 주식회사 이엔케이글로벌 | 신축성재질 성형틀 기반의 고흡수성 고형 제형 흡습제 제조 장비 |
| KR20250120088A (ko) | 2024-02-01 | 2025-08-08 | (주) 제이아리 | 고흡수성 고형 제형 흡습제 제조 장비 |
Also Published As
| Publication number | Publication date |
|---|---|
| EP0930875A2 (de) | 1999-07-28 |
| JP4975894B2 (ja) | 2012-07-11 |
| JP2001500130A (ja) | 2001-01-09 |
| ES2199373T3 (es) | 2004-02-16 |
| TW474824B (en) | 2002-02-01 |
| WO1998010752A2 (de) | 1998-03-19 |
| WO1998010752A3 (de) | 1998-06-18 |
| HRP970485A2 (en) | 1998-08-31 |
| SK26099A3 (en) | 2000-03-13 |
| AU720535B2 (en) | 2000-06-01 |
| BR9711777A (pt) | 1999-08-24 |
| ATE239452T1 (de) | 2003-05-15 |
| US6221368B1 (en) | 2001-04-24 |
| CA2265532C (en) | 2006-04-04 |
| CA2265532A1 (en) | 1998-03-19 |
| AU4384697A (en) | 1998-04-02 |
| TR199900563T2 (xx) | 1999-07-21 |
| DE59710059D1 (de) | 2003-06-12 |
| IL128672A0 (en) | 2000-01-31 |
| DK0930875T3 (da) | 2003-09-01 |
| CN1230109A (zh) | 1999-09-29 |
| EP0930875B1 (de) | 2003-05-07 |
| CZ82999A3 (cs) | 1999-06-16 |
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