KR101811997B1 - 1­클로로­4­(베타­d­글루코피라노스­1­일)­2­(4­((s)­테트라하이드로푸란­3­일옥시)벤질)벤젠의 결정형의 제조방법 - Google Patents

1­클로로­4­(베타­d­글루코피라노스­1­일)­2­(4­((s)­테트라하이드로푸란­3­일옥시)벤질)벤젠의 결정형의 제조방법 Download PDF

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KR101811997B1
KR101811997B1 KR1020127008069A KR20127008069A KR101811997B1 KR 101811997 B1 KR101811997 B1 KR 101811997B1 KR 1020127008069 A KR1020127008069 A KR 1020127008069A KR 20127008069 A KR20127008069 A KR 20127008069A KR 101811997 B1 KR101811997 B1 KR 101811997B1
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solvent
compound
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crystalline form
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KR20120091024A (ko
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디르크 베버
스페냐 레너
토비아스 피들러
지모네 오를리흐
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베링거 인겔하임 인터내셔날 게엠베하
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    • C07D407/02Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
    • C07D407/10Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings linked by a carbon chain containing aromatic rings
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    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
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    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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    • A61P9/00Drugs for disorders of the cardiovascular system
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P9/12Antihypertensives
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    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H7/00Compounds containing non-saccharide radicals linked to saccharide radicals by a carbon-to-carbon bond
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  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
KR1020127008069A 2009-09-30 2010-09-24 1­클로로­4­(베타­d­글루코피라노스­1­일)­2­(4­((s)­테트라하이드로푸란­3­일옥시)벤질)벤젠의 결정형의 제조방법 Active KR101811997B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP09171847.8 2009-09-30
EP09171847 2009-09-30
PCT/EP2010/064117 WO2011039107A1 (en) 2009-09-30 2010-09-24 Method for the preparation of a crystalline form of 1-chloro-4- (beta-d-glucopyranos-1-yl)-2-(4-((s)-tetrahydrofuran-3-yloxy)benzyl)benzene

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KR20120091024A KR20120091024A (ko) 2012-08-17
KR101811997B1 true KR101811997B1 (ko) 2017-12-26

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US (1) US8802842B2 (enExample)
EP (1) EP2483286B1 (enExample)
JP (1) JP5736377B2 (enExample)
KR (1) KR101811997B1 (enExample)
CN (1) CN102549005B (enExample)
AR (1) AR078475A1 (enExample)
AU (1) AU2010303123B2 (enExample)
BR (1) BR112012007092B1 (enExample)
CA (1) CA2775961C (enExample)
CL (1) CL2012000810A1 (enExample)
DK (1) DK2483286T3 (enExample)
EA (1) EA020798B1 (enExample)
ES (1) ES2596202T3 (enExample)
HU (1) HUE029381T2 (enExample)
IL (1) IL218102B (enExample)
IN (1) IN2012DN02756A (enExample)
MX (1) MX2012002942A (enExample)
NZ (1) NZ598318A (enExample)
PH (1) PH12012500633B1 (enExample)
PL (1) PL2483286T3 (enExample)
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* Cited by examiner, † Cited by third party
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KR102111248B1 (ko) * 2019-12-30 2020-05-14 유니셀랩 주식회사 새로운 엠파글리플로진의 공결정

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AU2010303123A1 (en) 2012-03-15
EA201200506A1 (ru) 2012-11-30
EP2483286A1 (en) 2012-08-08
AU2010303123B2 (en) 2014-02-27
DK2483286T3 (en) 2016-09-19
BR112012007092A2 (pt) 2016-08-23
CN102549005A (zh) 2012-07-04
JP5736377B2 (ja) 2015-06-17
EP2483286B1 (en) 2016-07-13
HUE029381T2 (en) 2017-02-28
US8802842B2 (en) 2014-08-12
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AR078475A1 (es) 2011-11-09
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IL218102B (en) 2020-06-30
BR112012007092B1 (pt) 2020-03-31
KR20120091024A (ko) 2012-08-17
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PL2483286T3 (pl) 2017-04-28

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