KR101379967B1 - 임의로 2-치환된1,6-디히드로-6-옥소-4-피리미딘카르복시산의 제조 방법 - Google Patents

임의로 2-치환된1,6-디히드로-6-옥소-4-피리미딘카르복시산의 제조 방법 Download PDF

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KR101379967B1
KR101379967B1 KR1020077025602A KR20077025602A KR101379967B1 KR 101379967 B1 KR101379967 B1 KR 101379967B1 KR 1020077025602 A KR1020077025602 A KR 1020077025602A KR 20077025602 A KR20077025602 A KR 20077025602A KR 101379967 B1 KR101379967 B1 KR 101379967B1
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formula
compound
unsubstituted
substituted
acid
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KR20080006576A (ko
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라파엘 샤피로
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이 아이 듀폰 디 네모아 앤드 캄파니
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
KR1020077025602A 2005-05-06 2006-04-28 임의로 2-치환된1,6-디히드로-6-옥소-4-피리미딘카르복시산의 제조 방법 Active KR101379967B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US67826405P 2005-05-06 2005-05-06
US60/678,264 2005-05-06
PCT/US2006/016340 WO2006121648A2 (en) 2005-05-06 2006-04-28 Method for preparation of optionally 2-substituted 1,6-dihydro-6-oxo-4-pyrimidinecarboxylic acids

Publications (2)

Publication Number Publication Date
KR20080006576A KR20080006576A (ko) 2008-01-16
KR101379967B1 true KR101379967B1 (ko) 2014-04-01

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KR1020077025602A Active KR101379967B1 (ko) 2005-05-06 2006-04-28 임의로 2-치환된1,6-디히드로-6-옥소-4-피리미딘카르복시산의 제조 방법

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US (2) US8198442B2 (enExample)
EP (1) EP1877384B1 (enExample)
JP (1) JP5161764B2 (enExample)
KR (1) KR101379967B1 (enExample)
CN (2) CN101171237B (enExample)
AT (1) ATE506352T1 (enExample)
AU (1) AU2006246374B2 (enExample)
BR (1) BRPI0612475B8 (enExample)
CA (1) CA2607934C (enExample)
DE (1) DE602006021411D1 (enExample)
DK (1) DK1877384T3 (enExample)
EG (1) EG25480A (enExample)
ES (1) ES2362005T3 (enExample)
GE (1) GEP20105099B (enExample)
IL (2) IL185885A (enExample)
MA (1) MA29464B1 (enExample)
ME (1) ME00498B (enExample)
MX (1) MX2007013424A (enExample)
NZ (1) NZ561399A (enExample)
PL (1) PL1877384T3 (enExample)
RS (2) RS20070434A (enExample)
TN (1) TNSN07403A1 (enExample)
UA (1) UA92171C2 (enExample)
WO (1) WO2006121648A2 (enExample)
ZA (1) ZA200707975B (enExample)

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ATE465999T1 (de) * 2005-05-16 2010-05-15 Du Pont Verfahren zur herstellung substituierter pyrimidine
BRPI0616647B1 (pt) * 2005-09-29 2016-04-12 Dsm Ip Assets Bv sal de ácido metano-sulfônico, processo para esterificação de dihidro-fenil-glicina ou fenil-glicina no metil éster correspondente e uso de sal de ácido metano-sulfônico de metil éster de dihidro-fenil-glicina ou metil éster de fenil-glicina
ES2401348T3 (es) 2007-08-13 2013-04-18 Dow Agrosciences, Llc 2-(Fenil 2-fluoro-substituido)-6-amino-5-cloro-4-pirimidinacarboxilatos y su uso como herbicidas
BR122016003312B8 (pt) 2007-10-02 2022-06-28 Dow Agrosciences Llc Ácidos 2-substituído-6-amino-5-alquil, alquenil ou alquinil-4-pirimidinacarboxílicos e ácidos 6-substituído-4-amino-3-alquil, alquenil ou alquinil picolínicos, composição herbicida que os compreende e método de controlar vegetação indesejável
PL2279178T3 (pl) * 2008-04-18 2015-10-30 Dow Agrosciences Llc 2-(podstawione-fenylo)-6-hydroksy- lub alkoksy-5-podstawione-4 pirymidynokarboksylany i ich zastosowanie jako herbicydów
TWI596088B (zh) * 2011-01-25 2017-08-21 陶氏農業科學公司 ４－胺基－６－（經取代的苯基）吡啶甲酸酯及６－胺基－２－（經取代的苯基）－４－嘧啶羧酸酯之芳烷酯以及其等作為除草劑之用途
PL2736897T3 (pl) * 2011-07-27 2016-04-29 Bayer Ip Gmbh Podstawione kwasy pikolinowe i kwasy pirymidyno-4-karboksylowe, sposób ich otrzymywania i ich zastosowanie jako herbicydy i regulatory wzrostu roślin
US9113629B2 (en) * 2013-03-15 2015-08-25 Dow Agrosciences Llc 4-amino-6-(4-substituted-phenyl)-picolinates and 6-amino-2-(4-substituted-phenyl)-pyrimidine-4-carboxylates and their use as herbicides
US9637505B2 (en) 2013-03-15 2017-05-02 Dow Agrosciences Llc 4-amino-6-(heterocyclic)picolinates and 6-amino-2-(heterocyclic)pyrimidine-4-carboxylates and their use as herbicides
RU2672584C2 (ru) * 2013-03-15 2018-11-16 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи 4-амино-6-(гетероциклил)пиколинаты и 6-амино-2-(гетероциклил)пиримидин-4-карбоксилаты и их применение в качестве гербицидов
EP3193607A4 (en) 2014-09-15 2018-05-02 Dow AgroSciences LLC Synergistic weed control from applications of pyridine carboxylic acid herbicides and photosystem ii inhibitors
TWI689251B (zh) 2014-09-15 2020-04-01 美商陶氏農業科學公司 源自於施用吡啶羧酸除草劑與合成生長素除草劑及/或生長素轉運抑制劑的協同性雜草控制
TWI694770B (zh) 2014-09-15 2020-06-01 美商陶氏農業科學公司 包含吡啶羧酸除草劑之安全的除草組成物（二）
TWI689252B (zh) 2014-09-15 2020-04-01 美商陶氏農業科學公司 源自於施用吡啶羧酸除草劑與乙醯乳酸合成酶（ａｌｓ）抑制劑的協同性雜草控制
TWI685302B (zh) 2014-09-15 2020-02-21 美商陶氏農業科學公司 包含吡啶羧酸除草劑之安全的除草組成物
WO2026028053A2 (en) 2024-07-27 2026-02-05 Assia Chemical Industries Ltd. Process for the preparation of tovorafenib

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CA207185A (en) 1921-01-04 C. Wagner Virgil Warming plate
JPS60100559A (ja) * 1983-11-05 1985-06-04 Morishita Seiyaku Kk ２−アニリノ−１，６−ジヒドロ−６−オキソ−５−ピリミジンカルボン酸誘導体，その製法及び該化合物を含有する抗アレルギ−剤
JPH0331267A (ja) 1989-06-28 1991-02-12 Morishita Pharmaceut Co Ltd ２―アニリノ―１，６―ジヒドロ―６―オキソ―４―ピリミジンカルボン酸誘導体
JPH0341071A (ja) 1989-07-06 1991-02-21 Morishita Pharmaceut Co Ltd １，６―ジヒドロ―６―オキソ―２―フェノキシアルキルチオ―５―ピリミジンカルボン酸類
DE3935277A1 (de) 1989-10-24 1991-05-02 Hoechst Ag Sulfonierte heterocyclische carboxamide, verfahren zu ihrer herstellung, sie enthaltende mittel und ihre verwendung als herbizide oder wachstumsregulatoren
US5637618A (en) 1990-06-01 1997-06-10 Bioresearch, Inc. Specific eatable taste modifiers
DE4029654A1 (de) 1990-09-19 1992-04-02 Hoechst Ag 2-phenyl-pyrimidine, verfahren zu ihrer herstellung, sie enthaltende mittel und ihre verwendung als fungizide
DE4131924A1 (de) 1991-09-25 1993-07-08 Hoechst Ag Substituierte 4-alkoxypyrimidine, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
DE4408404A1 (de) 1994-03-12 1995-09-14 Huels Chemische Werke Ag Verfahren zur Herstellung von Chlorpyrimidinen
BR9908004A (pt) 1998-02-17 2001-12-18 Tularik Inc Composto, composição e método para prevençãoou supressão de uma infecção viral
US6281358B1 (en) 1999-04-15 2001-08-28 American Cyanamid Company Process for the preparation of substituted pyrimidines
SK285728B6 (sk) 1999-04-15 2007-07-06 Basf Aktiengesellschaft Spôsob prípravy substituovaných pyrimidínov
AU2002258400A1 (en) 2001-02-16 2002-08-28 Tularik Inc. Methods of using pyrimidine-based antiviral agents
EP1646615B1 (en) 2003-06-06 2009-08-26 Vertex Pharmaceuticals Incorporated Pyrimidine derivatives as modulators of atp-binding cassette transporters
TWI355894B (en) * 2003-12-19 2012-01-11 Du Pont Herbicidal pyrimidines
WO2006083012A1 (ja) 2005-02-02 2006-08-10 Ajinomoto Co., Inc. ピリミジン化合物の製造方法
DE102005027150A1 (de) 2005-03-12 2006-09-28 Bayer Healthcare Ag Pyrimidincarbonsäure-Derivate und ihre Verwendung
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Also Published As

Publication number Publication date
DK1877384T3 (da) 2011-08-15
IL185885A0 (en) 2008-01-06
IL185885A (en) 2012-10-31
ATE506352T1 (de) 2011-05-15
JP5161764B2 (ja) 2013-03-13
DE602006021411D1 (de) 2011-06-01
CN102153516B (zh) 2013-02-06
NZ561399A (en) 2009-11-27
CA2607934A1 (en) 2006-11-16
US20090043098A1 (en) 2009-02-12
IL222041A (en) 2016-10-31
KR20080006576A (ko) 2008-01-16
CN102153516A (zh) 2011-08-17
CN101171237B (zh) 2011-04-20
BRPI0612475B1 (pt) 2020-03-10
JP2008540414A (ja) 2008-11-20
WO2006121648A3 (en) 2006-12-28
GEP20105099B (en) 2010-10-25
EP1877384A2 (en) 2008-01-16
AU2006246374A1 (en) 2006-11-16
ES2362005T3 (es) 2011-06-27
BRPI0612475A2 (pt) 2010-11-23
EP1877384B1 (en) 2011-04-20
AU2006246374B2 (en) 2012-03-29
EG25480A (en) 2012-01-15
US20120232271A1 (en) 2012-09-13
MX2007013424A (es) 2008-01-16
RS51804B (sr) 2011-12-31
RS20070434A (sr) 2009-01-22
UA92171C2 (ru) 2010-10-11
MA29464B1 (fr) 2008-05-02
US8198442B2 (en) 2012-06-12
ME00498B (me) 2011-10-10
BRPI0612475B8 (pt) 2022-12-06
TNSN07403A1 (en) 2009-03-17
CA2607934C (en) 2013-10-01
ZA200707975B (en) 2008-11-26
PL1877384T3 (pl) 2011-09-30
WO2006121648A2 (en) 2006-11-16
CN101171237A (zh) 2008-04-30

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