AU2006246374B2 - Method for preparation of optionally 2-substituted 1,6-dihydro-6-oxo-4-pyrimidinecarboxylic acids - Google Patents

Method for preparation of optionally 2-substituted 1,6-dihydro-6-oxo-4-pyrimidinecarboxylic acids Download PDF

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Publication number
AU2006246374B2
AU2006246374B2 AU2006246374A AU2006246374A AU2006246374B2 AU 2006246374 B2 AU2006246374 B2 AU 2006246374B2 AU 2006246374 A AU2006246374 A AU 2006246374A AU 2006246374 A AU2006246374 A AU 2006246374A AU 2006246374 B2 AU2006246374 B2 AU 2006246374B2
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AU
Australia
Prior art keywords
formula
compound
acid
optionally substituted
water
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
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AU2006246374A
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English (en)
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AU2006246374A1 (en
Inventor
Rafael Shapiro
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Corteva Agriscience LLC
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Corteva Agriscience LLC
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Assigned to CORTEVA AGRISCIENCE LLC reassignment CORTEVA AGRISCIENCE LLC Request for Assignment Assignors: E. I. DU PONT DE NEMOURS AND COMPANY
Anticipated expiration legal-status Critical
Expired legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AU2006246374A 2005-05-06 2006-04-28 Method for preparation of optionally 2-substituted 1,6-dihydro-6-oxo-4-pyrimidinecarboxylic acids Expired AU2006246374B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US67826405P 2005-05-06 2005-05-06
US60/678,264 2005-05-06
PCT/US2006/016340 WO2006121648A2 (en) 2005-05-06 2006-04-28 Method for preparation of optionally 2-substituted 1,6-dihydro-6-oxo-4-pyrimidinecarboxylic acids

Publications (2)

Publication Number Publication Date
AU2006246374A1 AU2006246374A1 (en) 2006-11-16
AU2006246374B2 true AU2006246374B2 (en) 2012-03-29

Family

ID=36952291

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2006246374A Expired AU2006246374B2 (en) 2005-05-06 2006-04-28 Method for preparation of optionally 2-substituted 1,6-dihydro-6-oxo-4-pyrimidinecarboxylic acids

Country Status (25)

Country Link
US (2) US8198442B2 (enExample)
EP (1) EP1877384B1 (enExample)
JP (1) JP5161764B2 (enExample)
KR (1) KR101379967B1 (enExample)
CN (2) CN101171237B (enExample)
AT (1) ATE506352T1 (enExample)
AU (1) AU2006246374B2 (enExample)
BR (1) BRPI0612475B8 (enExample)
CA (1) CA2607934C (enExample)
DE (1) DE602006021411D1 (enExample)
DK (1) DK1877384T3 (enExample)
EG (1) EG25480A (enExample)
ES (1) ES2362005T3 (enExample)
GE (1) GEP20105099B (enExample)
IL (2) IL185885A (enExample)
MA (1) MA29464B1 (enExample)
ME (1) ME00498B (enExample)
MX (1) MX2007013424A (enExample)
NZ (1) NZ561399A (enExample)
PL (1) PL1877384T3 (enExample)
RS (2) RS20070434A (enExample)
TN (1) TNSN07403A1 (enExample)
UA (1) UA92171C2 (enExample)
WO (1) WO2006121648A2 (enExample)
ZA (1) ZA200707975B (enExample)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE465999T1 (de) * 2005-05-16 2010-05-15 Du Pont Verfahren zur herstellung substituierter pyrimidine
EP1931619B1 (en) * 2005-09-29 2015-06-24 DSM Sinochem Pharmaceuticals Netherlands B.V. Methanesulphonic acid salt of dihydrophenylglycine methyl ester or of phenylglycine methyl ester
EP2311815B1 (en) * 2007-08-13 2012-12-19 Dow AgroSciences LLC 2-(2-Fluoro-substituted phenyl)-6-amino-5-chloro-4-pyrimidinecarboxylates and their use as herbicides
PL2327694T3 (pl) 2007-10-02 2013-12-31 Dow Agrosciences Llc Podstawione kwasy 4-aminopikolinowe i ich zastosowanie jako herbicydów
MX2010011468A (es) * 2008-04-18 2010-12-14 Dow Agrosciences Llc 2-(fenil substituido)-6-hidroxi o alcoxi-5-substituido-4-pirimidin carboxilatos y sus usos como herbicidas.
TWI596088B (zh) * 2011-01-25 2017-08-21 陶氏農業科學公司 ４－胺基－６－（經取代的苯基）吡啶甲酸酯及６－胺基－２－（經取代的苯基）－４－嘧啶羧酸酯之芳烷酯以及其等作為除草劑之用途
HUE028580T2 (en) * 2011-07-27 2016-12-28 Bayer Ip Gmbh Substituted Picolinic Acids and Pyrimidine Carboxylic Acids, Process for their Preparation and Use as Herbicides and Plant Growth Regulators
US9113629B2 (en) * 2013-03-15 2015-08-25 Dow Agrosciences Llc 4-amino-6-(4-substituted-phenyl)-picolinates and 6-amino-2-(4-substituted-phenyl)-pyrimidine-4-carboxylates and their use as herbicides
US9637505B2 (en) 2013-03-15 2017-05-02 Dow Agrosciences Llc 4-amino-6-(heterocyclic)picolinates and 6-amino-2-(heterocyclic)pyrimidine-4-carboxylates and their use as herbicides
WO2014151008A1 (en) * 2013-03-15 2014-09-25 Dow Agrosciences Llc 4-amino-6-(heterocyclic)picolinates and 6-amino-2-(heterocyclic)pyrimidine-4-carboxylates and their use as herbicides
TWI689252B (zh) 2014-09-15 2020-04-01 美商陶氏農業科學公司 源自於施用吡啶羧酸除草劑與乙醯乳酸合成酶（ａｌｓ）抑制劑的協同性雜草控制
TWI685302B (zh) 2014-09-15 2020-02-21 美商陶氏農業科學公司 包含吡啶羧酸除草劑之安全的除草組成物
TWI689251B (zh) 2014-09-15 2020-04-01 美商陶氏農業科學公司 源自於施用吡啶羧酸除草劑與合成生長素除草劑及/或生長素轉運抑制劑的協同性雜草控制
AR101858A1 (es) 2014-09-15 2017-01-18 Dow Agrosciences Llc Composiciones herbicidas protegidas que comprenden un herbicida de ácido piridincarboxílico
EP3193607A4 (en) 2014-09-15 2018-05-02 Dow AgroSciences LLC Synergistic weed control from applications of pyridine carboxylic acid herbicides and photosystem ii inhibitors
WO2026028053A2 (en) 2024-07-27 2026-02-05 Assia Chemical Industries Ltd. Process for the preparation of tovorafenib

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Publication number Priority date Publication date Assignee Title
CA207185A (en) 1921-01-04 C. Wagner Virgil Warming plate
JPS60100559A (ja) * 1983-11-05 1985-06-04 Morishita Seiyaku Kk ２−アニリノ−１，６−ジヒドロ−６−オキソ−５−ピリミジンカルボン酸誘導体，その製法及び該化合物を含有する抗アレルギ−剤
JPH0331267A (ja) 1989-06-28 1991-02-12 Morishita Pharmaceut Co Ltd ２―アニリノ―１，６―ジヒドロ―６―オキソ―４―ピリミジンカルボン酸誘導体
JPH0341071A (ja) 1989-07-06 1991-02-21 Morishita Pharmaceut Co Ltd １，６―ジヒドロ―６―オキソ―２―フェノキシアルキルチオ―５―ピリミジンカルボン酸類
DE3935277A1 (de) 1989-10-24 1991-05-02 Hoechst Ag Sulfonierte heterocyclische carboxamide, verfahren zu ihrer herstellung, sie enthaltende mittel und ihre verwendung als herbizide oder wachstumsregulatoren
US5637618A (en) 1990-06-01 1997-06-10 Bioresearch, Inc. Specific eatable taste modifiers
DE4029654A1 (de) 1990-09-19 1992-04-02 Hoechst Ag 2-phenyl-pyrimidine, verfahren zu ihrer herstellung, sie enthaltende mittel und ihre verwendung als fungizide
DE4131924A1 (de) 1991-09-25 1993-07-08 Hoechst Ag Substituierte 4-alkoxypyrimidine, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
DE4408404A1 (de) 1994-03-12 1995-09-14 Huels Chemische Werke Ag Verfahren zur Herstellung von Chlorpyrimidinen
JP2002503662A (ja) 1998-02-17 2002-02-05 テュラリク インコーポレイテッド 抗ウイルス性ピリミジン誘導体
US6281358B1 (en) 1999-04-15 2001-08-28 American Cyanamid Company Process for the preparation of substituted pyrimidines
MXPA01010390A (es) 1999-04-15 2002-03-27 Basf Ag Proceso para la preparacion de pirimidinas sustituidas.
WO2002064096A2 (en) 2001-02-16 2002-08-22 Tularik Inc. Methods of using pyrimidine-based antiviral agents
ATE440825T1 (de) 2003-06-06 2009-09-15 Vertex Pharma Pyrimidin-derivate zur verwendung als modulatoren von atp-bindende kassette transportern
TWI355894B (en) * 2003-12-19 2012-01-11 Du Pont Herbicidal pyrimidines
EP1849765A4 (en) 2005-02-02 2010-05-05 Ajinomoto Kk PROCESS FOR PREPARING A PYRIMIDINE COMPOUND
DE102005027150A1 (de) 2005-03-12 2006-09-28 Bayer Healthcare Ag Pyrimidincarbonsäure-Derivate und ihre Verwendung
ATE465999T1 (de) 2005-05-16 2010-05-15 Du Pont Verfahren zur herstellung substituierter pyrimidine

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
J. Org. Chem., vol 26, 1961, p2755-2763 *

Also Published As

Publication number Publication date
ES2362005T3 (es) 2011-06-27
IL185885A0 (en) 2008-01-06
US20120232271A1 (en) 2012-09-13
JP5161764B2 (ja) 2013-03-13
TNSN07403A1 (en) 2009-03-17
ME00498B (me) 2011-10-10
CN102153516A (zh) 2011-08-17
US8198442B2 (en) 2012-06-12
IL185885A (en) 2012-10-31
EG25480A (en) 2012-01-15
ATE506352T1 (de) 2011-05-15
EP1877384A2 (en) 2008-01-16
BRPI0612475B1 (pt) 2020-03-10
IL222041A (en) 2016-10-31
MA29464B1 (fr) 2008-05-02
BRPI0612475A2 (pt) 2010-11-23
ZA200707975B (en) 2008-11-26
CN101171237A (zh) 2008-04-30
CN102153516B (zh) 2013-02-06
PL1877384T3 (pl) 2011-09-30
EP1877384B1 (en) 2011-04-20
BRPI0612475B8 (pt) 2022-12-06
CN101171237B (zh) 2011-04-20
RS20070434A (sr) 2009-01-22
CA2607934C (en) 2013-10-01
CA2607934A1 (en) 2006-11-16
US20090043098A1 (en) 2009-02-12
GEP20105099B (en) 2010-10-25
JP2008540414A (ja) 2008-11-20
WO2006121648A2 (en) 2006-11-16
RS51804B (sr) 2011-12-31
DE602006021411D1 (de) 2011-06-01
AU2006246374A1 (en) 2006-11-16
WO2006121648A3 (en) 2006-12-28
NZ561399A (en) 2009-11-27
MX2007013424A (es) 2008-01-16
DK1877384T3 (da) 2011-08-15
KR20080006576A (ko) 2008-01-16
UA92171C2 (ru) 2010-10-11
KR101379967B1 (ko) 2014-04-01

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Free format text: FORMER OWNER(S): E. I. DU PONT DE NEMOURS AND COMPANY