DE602006013970D1 - Verfahren zur herstellung substituierter pyrimidine - Google Patents

Verfahren zur herstellung substituierter pyrimidine

Info

Publication number
DE602006013970D1
DE602006013970D1 DE602006013970T DE602006013970T DE602006013970D1 DE 602006013970 D1 DE602006013970 D1 DE 602006013970D1 DE 602006013970 T DE602006013970 T DE 602006013970T DE 602006013970 T DE602006013970 T DE 602006013970T DE 602006013970 D1 DE602006013970 D1 DE 602006013970D1
Authority
DE
Germany
Prior art keywords
formula
compound
preparing
substituted pyrimidines
preparing substituted
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
DE602006013970T
Other languages
English (en)
Inventor
Gary David Annis
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
EIDP Inc
Original Assignee
EI Du Pont de Nemours and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by EI Du Pont de Nemours and Co filed Critical EI Du Pont de Nemours and Co
Publication of DE602006013970D1 publication Critical patent/DE602006013970D1/de
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/42—One nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/30—Halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/34—One oxygen atom
    • C07D239/36—One oxygen atom as doubly bound oxygen atom or as unsubstituted hydroxy radical

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
DE602006013970T 2005-05-16 2006-05-12 Verfahren zur herstellung substituierter pyrimidine Active DE602006013970D1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US68129805P 2005-05-16 2005-05-16
PCT/US2006/018522 WO2006124657A1 (en) 2005-05-16 2006-05-12 Method for preparing substituted pyrimidines

Publications (1)

Publication Number Publication Date
DE602006013970D1 true DE602006013970D1 (de) 2010-06-10

Family

ID=36867439

Family Applications (1)

Application Number Title Priority Date Filing Date
DE602006013970T Active DE602006013970D1 (de) 2005-05-16 2006-05-12 Verfahren zur herstellung substituierter pyrimidine

Country Status (13)

Country Link
US (1) US8013155B2 (de)
EP (1) EP1888536B1 (de)
JP (1) JP5069677B2 (de)
KR (1) KR101348458B1 (de)
CN (1) CN101175730B (de)
AT (1) ATE465999T1 (de)
AU (1) AU2006247581B2 (de)
BR (1) BRPI0612414A2 (de)
DE (1) DE602006013970D1 (de)
IL (1) IL185884A (de)
PL (1) PL1888536T3 (de)
WO (1) WO2006124657A1 (de)
ZA (1) ZA200707974B (de)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA200707975B (en) * 2005-05-06 2008-11-26 Du Pont Method for preparation of optionally 2-substituted 1,6-dihydro-6-oxo-4-pyrimidinecarboxylic acids
WO2007120706A2 (en) * 2006-04-10 2007-10-25 E. I. Du Pont De Nemours And Company Herbicidal mixtures
WO2013124246A1 (de) 2012-02-22 2013-08-29 Bayer Intellectual Property Gmbh Herbizid wirksame 4-dialkoxymethyl-2-phenylpyrimidine
CN102977050B (zh) * 2012-11-20 2015-04-22 浙江工业大学 一种2-苯并噻唑二甲缩醛和2-苯并噻唑甲醛的合成方法
CN116063179A (zh) * 2023-02-20 2023-05-05 南京杰运医药科技有限公司 一种4-甲氧基乙酰乙酸甲酯的合成方法

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA207185A (en) 1921-01-04 C. Wagner Virgil Warming plate
GB2095240A (en) 1981-03-05 1982-09-29 Fujisawa Pharmaceutical Co Dihydropyrimidine derivatives, processes for preparation thereof and pharmaceutical composition comprising the same
JPS57158779A (en) * 1981-03-05 1982-09-30 Fujisawa Pharmaceut Co Ltd Dihydropyrimidine derivative and its salt, their preparation and antiallergic containing the same
DE3935277A1 (de) 1989-10-24 1991-05-02 Hoechst Ag Sulfonierte heterocyclische carboxamide, verfahren zu ihrer herstellung, sie enthaltende mittel und ihre verwendung als herbizide oder wachstumsregulatoren
CN1071049A (zh) * 1991-10-09 1993-04-21 纳幕尔杜邦公司 用于稻中杂草防治的除草剂
JP2002503662A (ja) * 1998-02-17 2002-02-05 テュラリク インコーポレイテッド 抗ウイルス性ピリミジン誘導体
WO2000063183A1 (en) 1999-04-15 2000-10-26 American Cyanamid Company Process for the preparation of substituted pyrimidines
WO2002064096A2 (en) 2001-02-16 2002-08-22 Tularik Inc. Methods of using pyrimidine-based antiviral agents
WO2004111014A1 (en) * 2003-06-06 2004-12-23 Vertex Pharmaceuticals Incorporated Pyrimidine derivatives as modulators of atp-binding cassette transporters
TWI355894B (en) * 2003-12-19 2012-01-11 Du Pont Herbicidal pyrimidines
ZA200707975B (en) * 2005-05-06 2008-11-26 Du Pont Method for preparation of optionally 2-substituted 1,6-dihydro-6-oxo-4-pyrimidinecarboxylic acids

Also Published As

Publication number Publication date
JP2008540655A (ja) 2008-11-20
WO2006124657A1 (en) 2006-11-23
JP5069677B2 (ja) 2012-11-07
ZA200707974B (en) 2008-11-26
BRPI0612414A2 (pt) 2010-11-09
KR20080016640A (ko) 2008-02-21
AU2006247581A1 (en) 2006-11-23
EP1888536B1 (de) 2010-04-28
US20090054647A1 (en) 2009-02-26
KR101348458B1 (ko) 2014-01-07
PL1888536T3 (pl) 2010-09-30
ATE465999T1 (de) 2010-05-15
EP1888536A1 (de) 2008-02-20
US8013155B2 (en) 2011-09-06
IL185884A (en) 2012-03-29
IL185884A0 (en) 2008-01-06
AU2006247581B2 (en) 2011-10-20
CN101175730B (zh) 2011-05-25
CN101175730A (zh) 2008-05-07

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Legal Events

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