DE602006021411D1 - Verfahren zur herstellung von optional 2-substituierten 1,6-dihydro-6-oxo-4-pyrimidincarboxylsäuren - Google Patents
Verfahren zur herstellung von optional 2-substituierten 1,6-dihydro-6-oxo-4-pyrimidincarboxylsäurenInfo
- Publication number
- DE602006021411D1 DE602006021411D1 DE602006021411T DE602006021411T DE602006021411D1 DE 602006021411 D1 DE602006021411 D1 DE 602006021411D1 DE 602006021411 T DE602006021411 T DE 602006021411T DE 602006021411 T DE602006021411 T DE 602006021411T DE 602006021411 D1 DE602006021411 D1 DE 602006021411D1
- Authority
- DE
- Germany
- Prior art keywords
- substituted
- dihydro
- oxo
- acids
- pyrimidincarboxylic
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Active
Links
- -1 2-SUBSTITUTED 1,6-DIHYDRO-6-OXO-4-PYRIMIDINCARBOXYLIC ACIDS Chemical class 0.000 title abstract 2
- 239000002253 acid Substances 0.000 title 1
- 238000004519 manufacturing process Methods 0.000 title 1
- OKTJSMMVPCPJKN-UHFFFAOYSA-N Carbon Chemical group [C] OKTJSMMVPCPJKN-UHFFFAOYSA-N 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 150000002148 esters Chemical class 0.000 abstract 1
- YPOXGDJGKBXRFP-UHFFFAOYSA-N pyrimidine-4-carboxylic acid Chemical class OC(=O)C1=CC=NC=N1 YPOXGDJGKBXRFP-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US67826405P | 2005-05-06 | 2005-05-06 | |
| PCT/US2006/016340 WO2006121648A2 (en) | 2005-05-06 | 2006-04-28 | Method for preparation of optionally 2-substituted 1,6-dihydro-6-oxo-4-pyrimidinecarboxylic acids |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DE602006021411D1 true DE602006021411D1 (de) | 2011-06-01 |
Family
ID=36952291
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE602006021411T Active DE602006021411D1 (de) | 2005-05-06 | 2006-04-28 | Verfahren zur herstellung von optional 2-substituierten 1,6-dihydro-6-oxo-4-pyrimidincarboxylsäuren |
Country Status (25)
| Country | Link |
|---|---|
| US (2) | US8198442B2 (enExample) |
| EP (1) | EP1877384B1 (enExample) |
| JP (1) | JP5161764B2 (enExample) |
| KR (1) | KR101379967B1 (enExample) |
| CN (2) | CN101171237B (enExample) |
| AT (1) | ATE506352T1 (enExample) |
| AU (1) | AU2006246374B2 (enExample) |
| BR (1) | BRPI0612475B8 (enExample) |
| CA (1) | CA2607934C (enExample) |
| DE (1) | DE602006021411D1 (enExample) |
| DK (1) | DK1877384T3 (enExample) |
| EG (1) | EG25480A (enExample) |
| ES (1) | ES2362005T3 (enExample) |
| GE (1) | GEP20105099B (enExample) |
| IL (2) | IL185885A (enExample) |
| MA (1) | MA29464B1 (enExample) |
| ME (1) | ME00498B (enExample) |
| MX (1) | MX2007013424A (enExample) |
| NZ (1) | NZ561399A (enExample) |
| PL (1) | PL1877384T3 (enExample) |
| RS (2) | RS51804B (enExample) |
| TN (1) | TNSN07403A1 (enExample) |
| UA (1) | UA92171C2 (enExample) |
| WO (1) | WO2006121648A2 (enExample) |
| ZA (1) | ZA200707975B (enExample) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2006124657A1 (en) * | 2005-05-16 | 2006-11-23 | E. I. Du Pont De Nemours And Company | Method for preparing substituted pyrimidines |
| BRPI0616647B1 (pt) * | 2005-09-29 | 2016-04-12 | Dsm Ip Assets Bv | sal de ácido metano-sulfônico, processo para esterificação de dihidro-fenil-glicina ou fenil-glicina no metil éster correspondente e uso de sal de ácido metano-sulfônico de metil éster de dihidro-fenil-glicina ou metil éster de fenil-glicina |
| BRPI0815349A2 (pt) * | 2007-08-13 | 2015-02-10 | Dow Agrosciences Llc | 6-amino-5-cloro-4-pirimidinacarboxilatos substituídos com 2-(2-fluorofeni-la) e seu uso como herbicidas |
| CN101883759B (zh) | 2007-10-02 | 2014-05-21 | 陶氏益农公司 | 2-取代的-6-氨基-5-烷基、烯基或炔基-嘧啶-4-羧酸和6-取代的-4-氨基-3-烷基、烯基或炔基吡啶-2-羧酸以及它们作为除草剂的用途 |
| JP5314126B2 (ja) * | 2008-04-18 | 2013-10-16 | ダウ アグロサイエンシィズ エルエルシー | ２−（置換フェニル）−６−ヒドロキシ又はアルコキシ−５−置換−４−ピリミジンカルボキシラート及び除草剤としてのそれらの使用 |
| TWI596088B (zh) * | 2011-01-25 | 2017-08-21 | 陶氏農業科學公司 | ４－胺基－６－（經取代的苯基）吡啶甲酸酯及６－胺基－２－（經取代的苯基）－４－嘧啶羧酸酯之芳烷酯以及其等作為除草劑之用途 |
| MX370455B (es) * | 2011-07-27 | 2019-12-13 | Bayer Ip Gmbh | Ácidos picolínicos y piridimin-4-carboxílicos sustituidos, procedimiento para su preparación y su uso como herbicidas y reguladores del crecimiento de plantas. |
| US9637505B2 (en) | 2013-03-15 | 2017-05-02 | Dow Agrosciences Llc | 4-amino-6-(heterocyclic)picolinates and 6-amino-2-(heterocyclic)pyrimidine-4-carboxylates and their use as herbicides |
| US9113629B2 (en) * | 2013-03-15 | 2015-08-25 | Dow Agrosciences Llc | 4-amino-6-(4-substituted-phenyl)-picolinates and 6-amino-2-(4-substituted-phenyl)-pyrimidine-4-carboxylates and their use as herbicides |
| RU2672584C2 (ru) * | 2013-03-15 | 2018-11-16 | ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи | 4-амино-6-(гетероциклил)пиколинаты и 6-амино-2-(гетероциклил)пиримидин-4-карбоксилаты и их применение в качестве гербицидов |
| TWI689252B (zh) | 2014-09-15 | 2020-04-01 | 美商陶氏農業科學公司 | 源自於施用吡啶羧酸除草劑與乙醯乳酸合成酶（ａｌｓ）抑制劑的協同性雜草控制 |
| TWI685302B (zh) | 2014-09-15 | 2020-02-21 | 美商陶氏農業科學公司 | 包含吡啶羧酸除草劑之安全的除草組成物 |
| TWI698178B (zh) | 2014-09-15 | 2020-07-11 | 美商陶氏農業科學公司 | 源自於施用吡啶羧酸除草劑與光系統ii抑制劑的協同性雜草控制 |
| TWI694770B (zh) | 2014-09-15 | 2020-06-01 | 美商陶氏農業科學公司 | 包含吡啶羧酸除草劑之安全的除草組成物（二） |
| TWI689251B (zh) | 2014-09-15 | 2020-04-01 | 美商陶氏農業科學公司 | 源自於施用吡啶羧酸除草劑與合成生長素除草劑及/或生長素轉運抑制劑的協同性雜草控制 |
Family Cites Families (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA207185A (en) | 1921-01-04 | C. Wagner Virgil | Warming plate | |
| JPS60100559A (ja) * | 1983-11-05 | 1985-06-04 | Morishita Seiyaku Kk | ２−アニリノ−１，６−ジヒドロ−６−オキソ−５−ピリミジンカルボン酸誘導体，その製法及び該化合物を含有する抗アレルギ−剤 |
| JPH0331267A (ja) | 1989-06-28 | 1991-02-12 | Morishita Pharmaceut Co Ltd | ２―アニリノ―１，６―ジヒドロ―６―オキソ―４―ピリミジンカルボン酸誘導体 |
| JPH0341071A (ja) | 1989-07-06 | 1991-02-21 | Morishita Pharmaceut Co Ltd | １，６―ジヒドロ―６―オキソ―２―フェノキシアルキルチオ―５―ピリミジンカルボン酸類 |
| DE3935277A1 (de) | 1989-10-24 | 1991-05-02 | Hoechst Ag | Sulfonierte heterocyclische carboxamide, verfahren zu ihrer herstellung, sie enthaltende mittel und ihre verwendung als herbizide oder wachstumsregulatoren |
| US5637618A (en) | 1990-06-01 | 1997-06-10 | Bioresearch, Inc. | Specific eatable taste modifiers |
| DE4029654A1 (de) | 1990-09-19 | 1992-04-02 | Hoechst Ag | 2-phenyl-pyrimidine, verfahren zu ihrer herstellung, sie enthaltende mittel und ihre verwendung als fungizide |
| DE4131924A1 (de) | 1991-09-25 | 1993-07-08 | Hoechst Ag | Substituierte 4-alkoxypyrimidine, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel |
| DE4408404A1 (de) | 1994-03-12 | 1995-09-14 | Huels Chemische Werke Ag | Verfahren zur Herstellung von Chlorpyrimidinen |
| WO1999041253A1 (en) | 1998-02-17 | 1999-08-19 | Tularik Inc. | Anti-viral pyrimidine derivatives |
| PL351088A1 (en) | 1999-04-15 | 2003-03-24 | Basf Ag | Process for the preparation of substituted pyrimidines |
| US6281358B1 (en) | 1999-04-15 | 2001-08-28 | American Cyanamid Company | Process for the preparation of substituted pyrimidines |
| AU2002258400A1 (en) | 2001-02-16 | 2002-08-28 | Tularik Inc. | Methods of using pyrimidine-based antiviral agents |
| ATE440825T1 (de) | 2003-06-06 | 2009-09-15 | Vertex Pharma | Pyrimidin-derivate zur verwendung als modulatoren von atp-bindende kassette transportern |
| TWI355894B (en) * | 2003-12-19 | 2012-01-11 | Du Pont | Herbicidal pyrimidines |
| EP1849765A4 (en) | 2005-02-02 | 2010-05-05 | Ajinomoto Kk | PROCESS FOR PREPARING A PYRIMIDINE COMPOUND |
| DE102005027150A1 (de) | 2005-03-12 | 2006-09-28 | Bayer Healthcare Ag | Pyrimidincarbonsäure-Derivate und ihre Verwendung |
| WO2006124657A1 (en) | 2005-05-16 | 2006-11-23 | E. I. Du Pont De Nemours And Company | Method for preparing substituted pyrimidines |
-
2006
- 2006-04-28 CN CN200680015454XA patent/CN101171237B/zh active Active
- 2006-04-28 DK DK06751830.8T patent/DK1877384T3/da active
- 2006-04-28 BR BRPI0612475A patent/BRPI0612475B8/pt active IP Right Grant
- 2006-04-28 PL PL06751830T patent/PL1877384T3/pl unknown
- 2006-04-28 AT AT06751830T patent/ATE506352T1/de active
- 2006-04-28 CA CA2607934A patent/CA2607934C/en active Active
- 2006-04-28 EP EP06751830A patent/EP1877384B1/en active Active
- 2006-04-28 ZA ZA200707975A patent/ZA200707975B/xx unknown
- 2006-04-28 AU AU2006246374A patent/AU2006246374B2/en active Active
- 2006-04-28 RS RS20110315A patent/RS51804B/sr unknown
- 2006-04-28 KR KR1020077025602A patent/KR101379967B1/ko active Active
- 2006-04-28 WO PCT/US2006/016340 patent/WO2006121648A2/en not_active Ceased
- 2006-04-28 NZ NZ561399A patent/NZ561399A/en unknown
- 2006-04-28 ME MEP-2008-798A patent/ME00498B/me unknown
- 2006-04-28 RS RSP-2007/0434A patent/RS20070434A/sr unknown
- 2006-04-28 GE GEAP200610412A patent/GEP20105099B/en unknown
- 2006-04-28 MX MX2007013424A patent/MX2007013424A/es active IP Right Grant
- 2006-04-28 CN CN2011100456237A patent/CN102153516B/zh active Active
- 2006-04-28 ES ES06751830T patent/ES2362005T3/es active Active
- 2006-04-28 JP JP2008510079A patent/JP5161764B2/ja active Active
- 2006-04-28 DE DE602006021411T patent/DE602006021411D1/de active Active
- 2006-04-28 US US11/886,605 patent/US8198442B2/en active Active
- 2006-04-28 UA UAA200712021A patent/UA92171C2/ru unknown
-
2007
- 2007-09-10 IL IL185885A patent/IL185885A/en active IP Right Grant
- 2007-10-31 TN TNP2007000403A patent/TNSN07403A1/en unknown
- 2007-11-04 EG EGNA2007001195 patent/EG25480A/xx active
- 2007-11-20 MA MA30392A patent/MA29464B1/fr unknown
-
2012
- 2012-05-22 US US13/477,683 patent/US20120232271A1/en not_active Abandoned
- 2012-09-20 IL IL222041A patent/IL222041A/en active IP Right Grant
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