RS20070434A - Method for preparation of optionally 2-substituted 1,6- dihydro-6-oxo-4-pyrimidinecarboxylic acids - Google Patents

Method for preparation of optionally 2-substituted 1,6- dihydro-6-oxo-4-pyrimidinecarboxylic acids

Info

Publication number
RS20070434A
RS20070434A RSP-2007/0434A RSP20070434A RS20070434A RS 20070434 A RS20070434 A RS 20070434A RS P20070434 A RSP20070434 A RS P20070434A RS 20070434 A RS20070434 A RS 20070434A
Authority
RS
Serbia
Prior art keywords
optionally
substituted
dihydro
oxo
preparation
Prior art date
Application number
RSP-2007/0434A
Other languages
English (en)
Inventor
Rafael Shapiro
Original Assignee
E.I. Du Pont De Nemours And Company,
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by E.I. Du Pont De Nemours And Company, filed Critical E.I. Du Pont De Nemours And Company,
Publication of RS20070434A publication Critical patent/RS20070434A/sr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Izložen je novi postupak za izradu opciono 2-supstituisanih jedinjenja 1,6-dihidro-6-okso-4-pirimidinkarboksilne kiseline, formule (I), u kojoj R1 je H ili opciono supstituisani ugljenični deo. Takođe, izložen je i postupak, koji sadrži dodatne korake za izradu opciono supstituisanih 4 pirimidin-karboksilnih kiselina i estara korišćenjem jedinjenja formule (1) kao intermedijera.
RSP-2007/0434A 2005-05-06 2006-04-28 Method for preparation of optionally 2-substituted 1,6- dihydro-6-oxo-4-pyrimidinecarboxylic acids RS20070434A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US67826405P 2005-05-06 2005-05-06
PCT/US2006/016340 WO2006121648A2 (en) 2005-05-06 2006-04-28 Method for preparation of optionally 2-substituted 1,6-dihydro-6-oxo-4-pyrimidinecarboxylic acids

Publications (1)

Publication Number Publication Date
RS20070434A true RS20070434A (en) 2009-01-22

Family

ID=36952291

Family Applications (2)

Application Number Title Priority Date Filing Date
RSP-2007/0434A RS20070434A (en) 2005-05-06 2006-04-28 Method for preparation of optionally 2-substituted 1,6- dihydro-6-oxo-4-pyrimidinecarboxylic acids
RS20110315A RS51804B (sr) 2005-05-06 2006-04-28 Postupak za dobijanje eventualno 2-supstituisanih 1,6-dihidro-6-okso-4-pirimidinkarboksilnih kiselina

Family Applications After (1)

Application Number Title Priority Date Filing Date
RS20110315A RS51804B (sr) 2005-05-06 2006-04-28 Postupak za dobijanje eventualno 2-supstituisanih 1,6-dihidro-6-okso-4-pirimidinkarboksilnih kiselina

Country Status (25)

Country Link
US (2) US8198442B2 (sr)
EP (1) EP1877384B1 (sr)
JP (1) JP5161764B2 (sr)
KR (1) KR101379967B1 (sr)
CN (2) CN102153516B (sr)
AT (1) ATE506352T1 (sr)
AU (1) AU2006246374B2 (sr)
BR (1) BRPI0612475B8 (sr)
CA (1) CA2607934C (sr)
DE (1) DE602006021411D1 (sr)
DK (1) DK1877384T3 (sr)
EG (1) EG25480A (sr)
ES (1) ES2362005T3 (sr)
GE (1) GEP20105099B (sr)
IL (2) IL185885A (sr)
MA (1) MA29464B1 (sr)
ME (1) ME00498B (sr)
MX (1) MX2007013424A (sr)
NZ (1) NZ561399A (sr)
PL (1) PL1877384T3 (sr)
RS (2) RS20070434A (sr)
TN (1) TNSN07403A1 (sr)
UA (1) UA92171C2 (sr)
WO (1) WO2006121648A2 (sr)
ZA (1) ZA200707975B (sr)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8013155B2 (en) * 2005-05-16 2011-09-06 E. I. Du Pont De Nemours And Company Method for preparing substituted pyrimidines
WO2007039522A2 (en) * 2005-09-29 2007-04-12 Dsm Ip Assets B.V. Process for esterification of an organic acid
EP2311815B1 (en) * 2007-08-13 2012-12-19 Dow AgroSciences LLC 2-(2-Fluoro-substituted phenyl)-6-amino-5-chloro-4-pyrimidinecarboxylates and their use as herbicides
AU2008308815B2 (en) 2007-10-02 2012-02-02 Corteva Agriscience Llc 2-substituted-6-amino-5-alkyl, alkenyl or alkynyl-4-pyrimidinecarboxylic acids and 6-substituted-4-amino-3- alkyl, alkenyl or alkynyl picolinic acids and their use as herbicides
BRPI0911207B8 (pt) * 2008-04-18 2022-10-11 Dow Agrosciences Llc 2-(fenil substituído)-6-hidróxi ou alcóxi-5-substituído-4-pirimidinacarboxilatos, composição herbicida, e método para controle de vegetação indesejável".
TWI596088B (zh) * 2011-01-25 2017-08-21 陶氏農業科學公司 ４－胺基－６－（經取代的苯基）吡啶甲酸酯及６－胺基－２－（經取代的苯基）－４－嘧啶羧酸酯之芳烷酯以及其等作為除草劑之用途
US9179676B2 (en) * 2011-07-27 2015-11-10 Bayer Intellectual Property Gmbh Substituted picolinic acids and pyrimidine-4-carboxylic acids, method for the production thereof and use thereof as herbicides and plant growth regulators
US9113629B2 (en) * 2013-03-15 2015-08-25 Dow Agrosciences Llc 4-amino-6-(4-substituted-phenyl)-picolinates and 6-amino-2-(4-substituted-phenyl)-pyrimidine-4-carboxylates and their use as herbicides
US9637505B2 (en) 2013-03-15 2017-05-02 Dow Agrosciences Llc 4-amino-6-(heterocyclic)picolinates and 6-amino-2-(heterocyclic)pyrimidine-4-carboxylates and their use as herbicides
AU2014235455B2 (en) * 2013-03-15 2018-08-09 Corteva Agriscience Llc 4-amino-6-(heterocyclic)picolinates and 6-amino-2-(heterocyclic)pyrimidine-4-carboxylates and their use as herbicides
TWI689251B (zh) 2014-09-15 2020-04-01 美商陶氏農業科學公司 源自於施用吡啶羧酸除草劑與合成生長素除草劑及/或生長素轉運抑制劑的協同性雜草控制
TWI694770B (zh) 2014-09-15 2020-06-01 美商陶氏農業科學公司 包含吡啶羧酸除草劑之安全的除草組成物（二）
WO2016044276A1 (en) 2014-09-15 2016-03-24 Dow Agrosciences Llc Synergistic weed control from applications of pyridine carboxylic acid herbicides and photosystem ii inhibitors
TWI685302B (zh) 2014-09-15 2020-02-21 美商陶氏農業科學公司 包含吡啶羧酸除草劑之安全的除草組成物
TWI689252B (zh) 2014-09-15 2020-04-01 美商陶氏農業科學公司 源自於施用吡啶羧酸除草劑與乙醯乳酸合成酶（ａｌｓ）抑制劑的協同性雜草控制

Family Cites Families (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA207185A (en) 1921-01-04 C. Wagner Virgil Warming plate
JPS60100559A (ja) * 1983-11-05 1985-06-04 Morishita Seiyaku Kk ２−アニリノ−１，６−ジヒドロ−６−オキソ−５−ピリミジンカルボン酸誘導体，その製法及び該化合物を含有する抗アレルギ−剤
JPH0331267A (ja) 1989-06-28 1991-02-12 Morishita Pharmaceut Co Ltd ２―アニリノ―１，６―ジヒドロ―６―オキソ―４―ピリミジンカルボン酸誘導体
JPH0341071A (ja) 1989-07-06 1991-02-21 Morishita Pharmaceut Co Ltd １，６―ジヒドロ―６―オキソ―２―フェノキシアルキルチオ―５―ピリミジンカルボン酸類
DE3935277A1 (de) 1989-10-24 1991-05-02 Hoechst Ag Sulfonierte heterocyclische carboxamide, verfahren zu ihrer herstellung, sie enthaltende mittel und ihre verwendung als herbizide oder wachstumsregulatoren
US5637618A (en) 1990-06-01 1997-06-10 Bioresearch, Inc. Specific eatable taste modifiers
DE4029654A1 (de) 1990-09-19 1992-04-02 Hoechst Ag 2-phenyl-pyrimidine, verfahren zu ihrer herstellung, sie enthaltende mittel und ihre verwendung als fungizide
DE4131924A1 (de) 1991-09-25 1993-07-08 Hoechst Ag Substituierte 4-alkoxypyrimidine, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
DE4408404A1 (de) 1994-03-12 1995-09-14 Huels Chemische Werke Ag Verfahren zur Herstellung von Chlorpyrimidinen
CN1297447A (zh) 1998-02-17 2001-05-30 图拉列克股份有限公司 抗病毒嘧啶衍生物
IL145888A0 (en) 1999-04-15 2002-07-25 Basf Ag Process for the preparation of substituted pyrimidines
US6281358B1 (en) 1999-04-15 2001-08-28 American Cyanamid Company Process for the preparation of substituted pyrimidines
AU2002258400A1 (en) 2001-02-16 2002-08-28 Tularik Inc. Methods of using pyrimidine-based antiviral agents
EP1646615B1 (en) 2003-06-06 2009-08-26 Vertex Pharmaceuticals Incorporated Pyrimidine derivatives as modulators of atp-binding cassette transporters
TWI355894B (en) 2003-12-19 2012-01-11 Du Pont Herbicidal pyrimidines
JPWO2006083012A1 (ja) 2005-02-02 2008-06-26 味の素株式会社 ピリミジン化合物の製造方法
DE102005027150A1 (de) 2005-03-12 2006-09-28 Bayer Healthcare Ag Pyrimidincarbonsäure-Derivate und ihre Verwendung
US8013155B2 (en) 2005-05-16 2011-09-06 E. I. Du Pont De Nemours And Company Method for preparing substituted pyrimidines

Also Published As

Publication number Publication date
BRPI0612475A2 (pt) 2010-11-23
WO2006121648A3 (en) 2006-12-28
GEP20105099B (en) 2010-10-25
NZ561399A (en) 2009-11-27
CN102153516A (zh) 2011-08-17
CN101171237A (zh) 2008-04-30
IL222041A (en) 2016-10-31
KR101379967B1 (ko) 2014-04-01
DE602006021411D1 (de) 2011-06-01
KR20080006576A (ko) 2008-01-16
PL1877384T3 (pl) 2011-09-30
IL185885A (en) 2012-10-31
MA29464B1 (fr) 2008-05-02
AU2006246374A1 (en) 2006-11-16
BRPI0612475B8 (pt) 2022-12-06
JP5161764B2 (ja) 2013-03-13
US20090043098A1 (en) 2009-02-12
ATE506352T1 (de) 2011-05-15
TNSN07403A1 (en) 2009-03-17
CA2607934C (en) 2013-10-01
EP1877384B1 (en) 2011-04-20
EG25480A (en) 2012-01-15
BRPI0612475B1 (pt) 2020-03-10
WO2006121648A2 (en) 2006-11-16
ES2362005T3 (es) 2011-06-27
ZA200707975B (en) 2008-11-26
ME00498B (me) 2011-10-10
MX2007013424A (es) 2008-01-16
CN102153516B (zh) 2013-02-06
IL185885A0 (en) 2008-01-06
JP2008540414A (ja) 2008-11-20
US20120232271A1 (en) 2012-09-13
DK1877384T3 (da) 2011-08-15
UA92171C2 (ru) 2010-10-11
AU2006246374B2 (en) 2012-03-29
US8198442B2 (en) 2012-06-12
EP1877384A2 (en) 2008-01-16
CN101171237B (zh) 2011-04-20
RS51804B (sr) 2011-12-31
CA2607934A1 (en) 2006-11-16

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