KR101065979B1 - 피리딜 비방향족 질소 함유 헤테로환-1-카르복실산에스테르 유도체 - Google Patents

피리딜 비방향족 질소 함유 헤테로환-1-카르복실산에스테르 유도체 Download PDF

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KR101065979B1
KR101065979B1 KR1020097011569A KR20097011569A KR101065979B1 KR 101065979 B1 KR101065979 B1 KR 101065979B1 KR 1020097011569 A KR1020097011569 A KR 1020097011569A KR 20097011569 A KR20097011569 A KR 20097011569A KR 101065979 B1 KR101065979 B1 KR 101065979B1
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leu
gly
ser
ala
val
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KR20090077855A (ko
Inventor
다까히로 이시이
다까시 수가네
준 마에다
후미에 나라자끼
아끼오 가께후다
겐따로 사또
다쯔히사 다까하시
다까또시 가나야마
치까시 사이또
조따로 스즈끼
치사또 가나이
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아스텔라스세이야쿠 가부시키가이샤
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
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    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
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    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/472—Non-condensed isoquinolines, e.g. papaverine
    • A61K31/4725—Non-condensed isoquinolines, e.g. papaverine containing further heterocyclic rings
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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  • Child & Adolescent Psychology (AREA)
  • Diabetes (AREA)
  • Anesthesiology (AREA)
  • Vascular Medicine (AREA)
  • Otolaryngology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
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KR1020097011569A 2005-02-17 2006-02-16 피리딜 비방향족 질소 함유 헤테로환-1-카르복실산에스테르 유도체 Expired - Fee Related KR101065979B1 (ko)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JPJP-P-2005-040197 2005-02-17
JP2005040197 2005-02-17
JP2005303065 2005-10-18
JPJP-P-2005-303065 2005-10-18

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KR1020077020924A Division KR101063663B1 (ko) 2005-02-17 2006-02-16 피리딜 비방향족 질소 함유 헤테로환-1-카르복실산에스테르유도체

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KR20090077855A KR20090077855A (ko) 2009-07-15
KR101065979B1 true KR101065979B1 (ko) 2011-09-19

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KR1020077020924A Active KR101063663B1 (ko) 2005-02-17 2006-02-16 피리딜 비방향족 질소 함유 헤테로환-1-카르복실산에스테르유도체
KR1020097011570A Expired - Fee Related KR101063585B1 (ko) 2005-02-17 2006-02-16 피리딜 비방향족 질소 함유 헤테로환-1-카르복실산에스테르 유도체
KR1020097011569A Expired - Fee Related KR101065979B1 (ko) 2005-02-17 2006-02-16 피리딜 비방향족 질소 함유 헤테로환-1-카르복실산에스테르 유도체

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KR1020097011570A Expired - Fee Related KR101063585B1 (ko) 2005-02-17 2006-02-16 피리딜 비방향족 질소 함유 헤테로환-1-카르복실산에스테르 유도체

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EP (2) EP1849773B1 (enExample)
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KR (3) KR101063663B1 (enExample)
CN (1) CN101160287B (enExample)
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