KR100969088B1 - 살충제로서의 5-치환된-알킬아미노피라졸 유도체 - Google Patents

살충제로서의 5-치환된-알킬아미노피라졸 유도체 Download PDF

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Publication number
KR100969088B1
KR100969088B1 KR1020047013930A KR20047013930A KR100969088B1 KR 100969088 B1 KR100969088 B1 KR 100969088B1 KR 1020047013930 A KR1020047013930 A KR 1020047013930A KR 20047013930 A KR20047013930 A KR 20047013930A KR 100969088 B1 KR100969088 B1 KR 100969088B1
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KR
South Korea
Prior art keywords
alkyl
haloalkyl
group
cycloalkyl
halogen
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Expired - Fee Related
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KR1020047013930A
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English (en)
Korean (ko)
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KR20040097151A (ko
Inventor
초우데이비드테-웨이
바스티안스헨리쿠스마리아마티너스
쿨만안케
토네쎈마리아-테레시아
슈나테러스테판
돌러우베
후앙자민
시거칼
스크리브너앤드류
페레즈드레온아달베르토에이
Original Assignee
메리얼 리미티드
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Publication of KR20040097151A publication Critical patent/KR20040097151A/ko
Application granted granted Critical
Publication of KR100969088B1 publication Critical patent/KR100969088B1/ko
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Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/44—Oxygen and nitrogen or sulfur and nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Environmental Sciences (AREA)
  • Zoology (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
KR1020047013930A 2002-03-05 2003-02-27 살충제로서의 5-치환된-알킬아미노피라졸 유도체 Expired - Fee Related KR100969088B1 (ko)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US36132802P 2002-03-05 2002-03-05
US60/361,328 2002-03-05
EP02027033.6 2002-12-03
EP02027033 2002-12-03
PCT/EP2003/002010 WO2003074493A1 (en) 2002-03-05 2003-02-27 5-substituted-alkylaminopyrazole derivatives as pesticides

Publications (2)

Publication Number Publication Date
KR20040097151A KR20040097151A (ko) 2004-11-17
KR100969088B1 true KR100969088B1 (ko) 2010-07-09

Family

ID=44237171

Family Applications (2)

Application Number Title Priority Date Filing Date
KR1020047013930A Expired - Fee Related KR100969088B1 (ko) 2002-03-05 2003-02-27 살충제로서의 5-치환된-알킬아미노피라졸 유도체
KR1020047013964A Expired - Fee Related KR100966012B1 (ko) 2002-03-05 2003-02-27 살충제로서의 5-치환된-알킬아미노피라졸 유도체

Family Applications After (1)

Application Number Title Priority Date Filing Date
KR1020047013964A Expired - Fee Related KR100966012B1 (ko) 2002-03-05 2003-02-27 살충제로서의 5-치환된-알킬아미노피라졸 유도체

Country Status (16)

Country Link
EP (2) EP1483246B1 (enExample)
JP (2) JP2005530701A (enExample)
KR (2) KR100969088B1 (enExample)
CN (2) CN100532364C (enExample)
AT (2) ATE335728T1 (enExample)
AU (2) AU2003211629B8 (enExample)
BR (2) BR0308135A (enExample)
DE (2) DE60302558T2 (enExample)
DK (2) DK1483245T3 (enExample)
ES (2) ES2274210T3 (enExample)
NZ (1) NZ535054A (enExample)
PL (2) PL373026A1 (enExample)
PT (1) PT1483245E (enExample)
RU (2) RU2336272C2 (enExample)
SI (2) SI1483245T1 (enExample)
WO (2) WO2003074492A2 (enExample)

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US7514464B2 (en) * 2003-12-18 2009-04-07 Pfizer Limited Substituted arylpyrazoles
PL1727805T3 (pl) * 2004-03-15 2009-01-30 Merial Ltd Pochodne 1-fenylo i 1-pirydylopirazolu oraz ich zastosowanie jako pestycydów
ES2345559T3 (es) 2004-03-24 2010-09-27 Merial Ltd. Derivados de 5-aminoalquilpirazol como agentes pesticidas.
JP4890451B2 (ja) 2004-06-26 2012-03-07 メリアル リミテッド 1−アリール−アミノピロールに基づく殺虫剤
JP4875614B2 (ja) 2004-06-26 2012-02-15 メリアル リミテッド 殺虫剤としてのn−フェニルピラゾール誘導体
MX2007000159A (es) * 2004-06-26 2007-10-10 Bayer Cropscience Sa Derivados de n-fenilpirazol pesticidas.
CA2587429C (en) 2004-12-07 2013-03-05 Merial Limited 5-aminopyrazole derivatives as pesticidal compounds
ES2377481T3 (es) * 2005-01-21 2012-03-28 Merial Ltd. Derivados de pirazole como pesticidas.
UA94278C2 (ru) * 2006-08-08 2011-04-26 БАЙЕР КРОПСАЙЕНС ЭлПи Способ обработки растений
CN100424139C (zh) * 2006-08-25 2008-10-08 蒋文兰 凹凸棒悬浮剂
DE102007003036A1 (de) 2006-12-20 2008-06-26 Bayer Cropscience Ag Pyrimidinylpyrazole
RU2384065C2 (ru) * 2007-12-10 2010-03-20 Общество с ограниченной ответственностью "ЯДЖУР-ВЕДА" Инсектоакарицидное средство
CN101998963B (zh) * 2008-02-12 2014-09-24 陶氏益农公司 杀虫组合物
US20110190365A1 (en) 2008-08-14 2011-08-04 Bayer Crop Science Ag Insecticidal 4-phenyl-1H-pyrazoles
KR20110116220A (ko) * 2009-02-11 2011-10-25 다우 아그로사이언시즈 엘엘씨 살충 조성물
EP2398771B1 (en) 2009-02-18 2015-07-29 Boehringer Ingelheim International GmbH Heterocyclic compounds which modulate the cb2 receptor
UA104057C2 (ru) * 2009-10-21 2013-12-25 Ніппон Сода Ко., Лтд. Композиция приманки для борьбы с клещами
EP2523936A1 (en) 2010-01-15 2012-11-21 Boehringer Ingelheim International GmbH Compounds which modulate the cb2 receptor
CN102206184B (zh) * 2010-03-29 2013-07-10 南开大学 3-氰基-1-(2,6-二氯-4-三氟甲基苯基)吡唑衍生物杀虫剂
WO2012012307A1 (en) * 2010-07-22 2012-01-26 Boehringer Ingelheim International Gmbh Sulfonyl compounds which modulate the cb2 rece
TW201321367A (zh) * 2011-10-25 2013-06-01 Du Pont 經1,3-二芳基取代之雜環殺蟲劑
RU2483539C1 (ru) * 2011-12-21 2013-06-10 Федеральное государственное бюджетное образовательное учреждение высшего профессионального образования "Башкирский государственный университет" Средство для борьбы с грибковыми заболеваниями сельскохозяйственных культур
EP2803668A1 (en) 2013-05-17 2014-11-19 Boehringer Ingelheim International Gmbh Novel (cyano-dimethyl-methyl)-isoxazoles and -[1,3,4]thiadiazoles
CN106187896B (zh) * 2016-07-19 2018-07-31 中南民族大学 超声波喷雾微波辐射一体化制备芳基吡唑单或多烷基化衍生物

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2000035884A1 (en) * 1998-12-11 2000-06-22 Aventis Cropscience S.A. Control of arthropods in animals
JP2001506664A (ja) * 1996-12-24 2001-05-22 ローヌ−プーラン・アグロ 農薬の1−アリールピラゾール類

Family Cites Families (11)

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Publication number Priority date Publication date Assignee Title
GB8531485D0 (en) * 1985-12-20 1986-02-05 May & Baker Ltd Compositions of matter
GB8713768D0 (en) * 1987-06-12 1987-07-15 May & Baker Ltd Compositions of matter
DE4343832A1 (de) * 1993-12-22 1995-06-29 Bayer Ag Substituierte 1-Arylpyrazole
GB9601128D0 (en) * 1995-08-11 1996-03-20 Pfizer Ltd Parasiticidal compounds
JPH0987111A (ja) * 1995-09-27 1997-03-31 Sumitomo Chem Co Ltd 害虫駆除用毒餌剤
FR2739255B1 (fr) * 1995-09-29 1998-09-04 Rhone Merieux Composition antiparasitaire pour le traitement et la protection des animaux de compagnie
GR1002899B (el) * 1996-03-29 1998-05-11 Rhone Merieux Περιλαιμιο κατα ψυλλων και κροτωνων για σκυλους και γατες, με βαση ν-φαινυλπυραζολη
US6069157A (en) * 1997-11-25 2000-05-30 Pfizer Inc. Parasiticidal compounds
DE19650197A1 (de) * 1996-12-04 1998-06-10 Bayer Ag 3-Thiocarbamoylpyrazol-Derivate
US6350771B1 (en) * 1996-12-24 2002-02-26 Rhone-Poulenc, Inc. Pesticidal 1-arylpyrazoles
CN101062920A (zh) * 2000-06-09 2007-10-31 阿方蒂农科股份有限公司 除虫化合物的制备方法及其新的中间体

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2001506664A (ja) * 1996-12-24 2001-05-22 ローヌ−プーラン・アグロ 農薬の1−アリールピラゾール類
WO2000035884A1 (en) * 1998-12-11 2000-06-22 Aventis Cropscience S.A. Control of arthropods in animals

Also Published As

Publication number Publication date
AU2003221298B2 (en) 2009-02-19
KR20040097155A (ko) 2004-11-17
ES2249709T3 (es) 2006-04-01
BR0308135A (pt) 2005-01-11
RU2004129578A (ru) 2005-04-10
AU2003211629B2 (en) 2009-01-08
JP2005526055A (ja) 2005-09-02
RU2336272C2 (ru) 2008-10-20
DE60302558D1 (de) 2006-01-05
CN100532364C (zh) 2009-08-26
AU2003211629B8 (en) 2009-01-22
DK1483245T3 (da) 2006-12-18
BRPI0308189B1 (pt) 2015-12-29
BR0308189A (pt) 2004-12-21
CN1642921A (zh) 2005-07-20
KR100966012B1 (ko) 2010-06-24
KR20040097151A (ko) 2004-11-17
RU2308452C2 (ru) 2007-10-20
SI1483245T1 (sl) 2007-02-28
WO2003074492A3 (en) 2003-12-24
DE60302558T2 (de) 2006-08-10
ATE311367T1 (de) 2005-12-15
AU2003221298A1 (en) 2003-09-16
JP4696311B2 (ja) 2011-06-08
RU2004129579A (ru) 2005-04-20
EP1483246B1 (en) 2005-11-30
WO2003074492A2 (en) 2003-09-12
ES2274210T3 (es) 2007-05-16
DK1483246T3 (da) 2006-04-10
EP1483246A1 (en) 2004-12-08
PL373026A1 (en) 2005-08-08
JP2005530701A (ja) 2005-10-13
SI1483246T1 (sl) 2006-04-30
WO2003074493A1 (en) 2003-09-12
DE60307438T2 (de) 2007-04-12
DE60307438D1 (de) 2006-09-21
AU2003211629A1 (en) 2003-09-16
EP1483245A2 (en) 2004-12-08
PT1483245E (pt) 2006-12-29
PL372918A1 (en) 2005-08-08
NZ535054A (en) 2006-09-29
CN1642920A (zh) 2005-07-20
CN1642920B (zh) 2010-05-26
ATE335728T1 (de) 2006-09-15
EP1483245B1 (en) 2006-08-09

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