AU2003211629B8 - 5-substituted-alkylaminopyrazole derivatives as pesticides - Google Patents

5-substituted-alkylaminopyrazole derivatives as pesticides Download PDF

Info

Publication number
AU2003211629B8
AU2003211629B8 AU2003211629A AU2003211629A AU2003211629B8 AU 2003211629 B8 AU2003211629 B8 AU 2003211629B8 AU 2003211629 A AU2003211629 A AU 2003211629A AU 2003211629 A AU2003211629 A AU 2003211629A AU 2003211629 B8 AU2003211629 B8 AU 2003211629B8
Authority
AU
Australia
Prior art keywords
alkyl
halogen
group
substituted
haloalkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
AU2003211629A
Other languages
English (en)
Other versions
AU2003211629B2 (en
AU2003211629A1 (en
Inventor
Henricus Maria Martinus Bastiaans
David Teh-Wei Chou
Uwe Doller
Jamin Huang
Anke Kuhlmann
Adalberto A. Perez De Leon
Stefan Schnatterer
Andrew Scribner
Karl Seeger
Maria-Theresia Thonessen
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Boehringer Ingelheim Animal Health USA Inc
Original Assignee
Boehringer Ingelheim Animal Health USA Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Animal Health USA Inc filed Critical Boehringer Ingelheim Animal Health USA Inc
Publication of AU2003211629A1 publication Critical patent/AU2003211629A1/en
Assigned to MERIAL LTD reassignment MERIAL LTD Request for Assignment Assignors: BAYER CROPSCIENCE S.A.
Publication of AU2003211629B2 publication Critical patent/AU2003211629B2/en
Application granted granted Critical
Publication of AU2003211629B8 publication Critical patent/AU2003211629B8/en
Assigned to MERIAL, INC. reassignment MERIAL, INC. Request for Assignment Assignors: MERIAL LTD
Assigned to Boehringer Ingelheim Animal Health USA Inc. reassignment Boehringer Ingelheim Animal Health USA Inc. Request for Assignment Assignors: MERIAL, INC.
Anticipated expiration legal-status Critical
Expired legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/44—Oxygen and nitrogen or sulfur and nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Environmental Sciences (AREA)
  • Zoology (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
AU2003211629A 2002-03-05 2003-02-27 5-substituted-alkylaminopyrazole derivatives as pesticides Expired AU2003211629B8 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US36132802P 2002-03-05 2002-03-05
US60/361,328 2002-03-05
EP02027033.6 2002-12-03
EP02027033 2002-12-03
PCT/EP2003/002009 WO2003074492A2 (en) 2002-03-05 2003-02-27 5-substituted-alkylaminopyrazole derivatives as pesticides

Publications (3)

Publication Number Publication Date
AU2003211629A1 AU2003211629A1 (en) 2003-09-16
AU2003211629B2 AU2003211629B2 (en) 2009-01-08
AU2003211629B8 true AU2003211629B8 (en) 2009-01-22

Family

ID=44237171

Family Applications (2)

Application Number Title Priority Date Filing Date
AU2003211629A Expired AU2003211629B8 (en) 2002-03-05 2003-02-27 5-substituted-alkylaminopyrazole derivatives as pesticides
AU2003221298A Expired AU2003221298B2 (en) 2002-03-05 2003-02-27 5-substituted-alkylaminopyrazole derivatives as pesticides

Family Applications After (1)

Application Number Title Priority Date Filing Date
AU2003221298A Expired AU2003221298B2 (en) 2002-03-05 2003-02-27 5-substituted-alkylaminopyrazole derivatives as pesticides

Country Status (16)

Country Link
EP (2) EP1483246B1 (enExample)
JP (2) JP2005530701A (enExample)
KR (2) KR100969088B1 (enExample)
CN (2) CN100532364C (enExample)
AT (2) ATE335728T1 (enExample)
AU (2) AU2003211629B8 (enExample)
BR (2) BR0308135A (enExample)
DE (2) DE60302558T2 (enExample)
DK (2) DK1483245T3 (enExample)
ES (2) ES2274210T3 (enExample)
NZ (1) NZ535054A (enExample)
PL (2) PL373026A1 (enExample)
PT (1) PT1483245E (enExample)
RU (2) RU2336272C2 (enExample)
SI (2) SI1483245T1 (enExample)
WO (2) WO2003074492A2 (enExample)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7514464B2 (en) * 2003-12-18 2009-04-07 Pfizer Limited Substituted arylpyrazoles
PL1727805T3 (pl) * 2004-03-15 2009-01-30 Merial Ltd Pochodne 1-fenylo i 1-pirydylopirazolu oraz ich zastosowanie jako pestycydów
ES2345559T3 (es) 2004-03-24 2010-09-27 Merial Ltd. Derivados de 5-aminoalquilpirazol como agentes pesticidas.
JP4890451B2 (ja) 2004-06-26 2012-03-07 メリアル リミテッド 1−アリール−アミノピロールに基づく殺虫剤
JP4875614B2 (ja) 2004-06-26 2012-02-15 メリアル リミテッド 殺虫剤としてのn−フェニルピラゾール誘導体
MX2007000159A (es) * 2004-06-26 2007-10-10 Bayer Cropscience Sa Derivados de n-fenilpirazol pesticidas.
CA2587429C (en) 2004-12-07 2013-03-05 Merial Limited 5-aminopyrazole derivatives as pesticidal compounds
ES2377481T3 (es) * 2005-01-21 2012-03-28 Merial Ltd. Derivados de pirazole como pesticidas.
UA94278C2 (ru) * 2006-08-08 2011-04-26 БАЙЕР КРОПСАЙЕНС ЭлПи Способ обработки растений
CN100424139C (zh) * 2006-08-25 2008-10-08 蒋文兰 凹凸棒悬浮剂
DE102007003036A1 (de) 2006-12-20 2008-06-26 Bayer Cropscience Ag Pyrimidinylpyrazole
RU2384065C2 (ru) * 2007-12-10 2010-03-20 Общество с ограниченной ответственностью "ЯДЖУР-ВЕДА" Инсектоакарицидное средство
CN101998963B (zh) * 2008-02-12 2014-09-24 陶氏益农公司 杀虫组合物
US20110190365A1 (en) 2008-08-14 2011-08-04 Bayer Crop Science Ag Insecticidal 4-phenyl-1H-pyrazoles
KR20110116220A (ko) * 2009-02-11 2011-10-25 다우 아그로사이언시즈 엘엘씨 살충 조성물
EP2398771B1 (en) 2009-02-18 2015-07-29 Boehringer Ingelheim International GmbH Heterocyclic compounds which modulate the cb2 receptor
UA104057C2 (ru) * 2009-10-21 2013-12-25 Ніппон Сода Ко., Лтд. Композиция приманки для борьбы с клещами
EP2523936A1 (en) 2010-01-15 2012-11-21 Boehringer Ingelheim International GmbH Compounds which modulate the cb2 receptor
CN102206184B (zh) * 2010-03-29 2013-07-10 南开大学 3-氰基-1-(2,6-二氯-4-三氟甲基苯基)吡唑衍生物杀虫剂
WO2012012307A1 (en) * 2010-07-22 2012-01-26 Boehringer Ingelheim International Gmbh Sulfonyl compounds which modulate the cb2 rece
TW201321367A (zh) * 2011-10-25 2013-06-01 Du Pont 經1,3-二芳基取代之雜環殺蟲劑
RU2483539C1 (ru) * 2011-12-21 2013-06-10 Федеральное государственное бюджетное образовательное учреждение высшего профессионального образования "Башкирский государственный университет" Средство для борьбы с грибковыми заболеваниями сельскохозяйственных культур
EP2803668A1 (en) 2013-05-17 2014-11-19 Boehringer Ingelheim International Gmbh Novel (cyano-dimethyl-methyl)-isoxazoles and -[1,3,4]thiadiazoles
CN106187896B (zh) * 2016-07-19 2018-07-31 中南民族大学 超声波喷雾微波辐射一体化制备芳基吡唑单或多烷基化衍生物

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8531485D0 (en) * 1985-12-20 1986-02-05 May & Baker Ltd Compositions of matter
GB8713768D0 (en) * 1987-06-12 1987-07-15 May & Baker Ltd Compositions of matter
DE4343832A1 (de) * 1993-12-22 1995-06-29 Bayer Ag Substituierte 1-Arylpyrazole
GB9601128D0 (en) * 1995-08-11 1996-03-20 Pfizer Ltd Parasiticidal compounds
JPH0987111A (ja) * 1995-09-27 1997-03-31 Sumitomo Chem Co Ltd 害虫駆除用毒餌剤
FR2739255B1 (fr) * 1995-09-29 1998-09-04 Rhone Merieux Composition antiparasitaire pour le traitement et la protection des animaux de compagnie
GR1002899B (el) * 1996-03-29 1998-05-11 Rhone Merieux Περιλαιμιο κατα ψυλλων και κροτωνων για σκυλους και γατες, με βαση ν-φαινυλπυραζολη
US6069157A (en) * 1997-11-25 2000-05-30 Pfizer Inc. Parasiticidal compounds
DE19650197A1 (de) * 1996-12-04 1998-06-10 Bayer Ag 3-Thiocarbamoylpyrazol-Derivate
CZ294766B6 (cs) * 1996-12-24 2005-03-16 Rhone-Poulenc Agro 1-Arylpyrazolové sloučeniny, pesticidní prostředky obsahující tyto sloučeniny jako účinné látky a způsob hubení škůdců
US6350771B1 (en) * 1996-12-24 2002-02-26 Rhone-Poulenc, Inc. Pesticidal 1-arylpyrazoles
AR021608A1 (es) * 1998-12-11 2002-07-31 Merial Ltd Represion de artropodos en animales
CN101062920A (zh) * 2000-06-09 2007-10-31 阿方蒂农科股份有限公司 除虫化合物的制备方法及其新的中间体

Also Published As

Publication number Publication date
AU2003221298B2 (en) 2009-02-19
KR20040097155A (ko) 2004-11-17
ES2249709T3 (es) 2006-04-01
BR0308135A (pt) 2005-01-11
RU2004129578A (ru) 2005-04-10
AU2003211629B2 (en) 2009-01-08
JP2005526055A (ja) 2005-09-02
RU2336272C2 (ru) 2008-10-20
DE60302558D1 (de) 2006-01-05
CN100532364C (zh) 2009-08-26
DK1483245T3 (da) 2006-12-18
BRPI0308189B1 (pt) 2015-12-29
BR0308189A (pt) 2004-12-21
CN1642921A (zh) 2005-07-20
KR100966012B1 (ko) 2010-06-24
KR20040097151A (ko) 2004-11-17
RU2308452C2 (ru) 2007-10-20
SI1483245T1 (sl) 2007-02-28
WO2003074492A3 (en) 2003-12-24
DE60302558T2 (de) 2006-08-10
ATE311367T1 (de) 2005-12-15
KR100969088B1 (ko) 2010-07-09
AU2003221298A1 (en) 2003-09-16
JP4696311B2 (ja) 2011-06-08
RU2004129579A (ru) 2005-04-20
EP1483246B1 (en) 2005-11-30
WO2003074492A2 (en) 2003-09-12
ES2274210T3 (es) 2007-05-16
DK1483246T3 (da) 2006-04-10
EP1483246A1 (en) 2004-12-08
PL373026A1 (en) 2005-08-08
JP2005530701A (ja) 2005-10-13
SI1483246T1 (sl) 2006-04-30
WO2003074493A1 (en) 2003-09-12
DE60307438T2 (de) 2007-04-12
DE60307438D1 (de) 2006-09-21
AU2003211629A1 (en) 2003-09-16
EP1483245A2 (en) 2004-12-08
PT1483245E (pt) 2006-12-29
PL372918A1 (en) 2005-08-08
NZ535054A (en) 2006-09-29
CN1642920A (zh) 2005-07-20
CN1642920B (zh) 2010-05-26
ATE335728T1 (de) 2006-09-15
EP1483245B1 (en) 2006-08-09

Similar Documents

Publication Publication Date Title
AU2003211629B2 (en) 5-substituted-alkylaminopyrazole derivatives as pesticides
WO2004049803A1 (en) Pesticidal 5- (acylamino) pyrazole derivatives
EP1692939A1 (en) Pesticidal substituted piperidines
US7576107B2 (en) 5-substituted-alkylaminopyrazole derivatives as pesticides
EP1727805B1 (en) 1-phenyl and 1-pyridylpyrazole derivatives and their use as pesticides
WO2004049797A2 (en) Pesticidal sulphonylaminopyrazoles
EP1599451A1 (en) Pesticidal 1-ayl-3-amidoxime-pyrazole derivatives
EP1663985B1 (en) Pesticides
US7879897B2 (en) Pesticidal 5-substituted-oxyalkylamino-1-arylpyrazole derivatives
EP1730115A1 (en) 5-aminoalkylpyrazole derivatives as pesticidal agents
EP1671967A1 (en) 1-Arylpyrazoles and their use as pesticides
WO2005082916A1 (en) 5-phosphorylaminopyrazole derivatives and their use as pesticides
WO2005082917A1 (en) 4-phosphorylpyrazole derivatives for pesticidal use
MXPA06010447A (en) 1-phenyl and 1-pyridylpyrazole derivatives and their use as pesticides

Legal Events

Date Code Title Description
PC1 Assignment before grant (sect. 113)

Owner name: MERIAL LTD

Free format text: FORMER APPLICANT(S): BAYER CROPSCIENCE S.A.

TH Corrigenda

Free format text: IN VOL 23, NO 1, PAGE(S) 6161 UNDER THE HEADING APPLICATIONS ACCEPTED - NAME INDEX UNDER THE NAME MERIAL LTD, ALLPLICATION NO. 2003211629, UNDER INID(72), CORRECT THE CO-INVENTOR NAME TO BASTIAANS, HENRICUS MARIA MARTINUS

FGA Letters patent sealed or granted (standard patent)
PC Assignment registered

Owner name: MERIAL, INC.

Free format text: FORMER OWNER WAS: MERIAL LTD

PC Assignment registered

Owner name: BOEHRINGER INGELHEIM ANIMAL HEALTH USA INC.

Free format text: FORMER OWNER(S): MERIAL, INC.

MK14 Patent ceased section 143(a) (annual fees not paid) or expired