JPWO2020140098A5 - - Google Patents

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JPWO2020140098A5
JPWO2020140098A5 JP2021538099A JP2021538099A JPWO2020140098A5 JP WO2020140098 A5 JPWO2020140098 A5 JP WO2020140098A5 JP 2021538099 A JP2021538099 A JP 2021538099A JP 2021538099 A JP2021538099 A JP 2021538099A JP WO2020140098 A5 JPWO2020140098 A5 JP WO2020140098A5
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JP7660063B2 (ja
JP2022517740A (ja
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JP2021538099A 2018-12-28 2019-12-27 サイクリン依存性キナーゼ7のインヒビターおよびそれらの使用 Active JP7660063B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862786328P 2018-12-28 2018-12-28
US62/786,328 2018-12-28
PCT/US2019/068835 WO2020140098A1 (en) 2018-12-28 2019-12-27 Inhibitors of cyclin-dependent kinase 7 and uses thereof

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JP2022517740A JP2022517740A (ja) 2022-03-10
JPWO2020140098A5 true JPWO2020140098A5 (enExample) 2023-01-06
JP7660063B2 JP7660063B2 (ja) 2025-04-10

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US (1) US12281126B2 (enExample)
EP (1) EP3902542A4 (enExample)
JP (1) JP7660063B2 (enExample)
CN (1) CN113557017B (enExample)
AU (1) AU2019413694B2 (enExample)
CA (1) CA3124422A1 (enExample)
WO (1) WO2020140098A1 (enExample)

Families Citing this family (10)

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CA3041563C (en) 2016-11-22 2023-10-31 Dana-Farber Cancer Institute, Inc. Pyrimidin-2-amine derivatives and pharmaceutical compositions thereof useful as inhibitors of cyclin-dependent kinase 12 (cdk12)
JP7590185B2 (ja) 2018-06-25 2024-11-26 ダナ-ファーバー キャンサー インスティテュート, インコーポレイテッド Taireファミリーキナーゼインヒビターおよびそれらの使用
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AU2020414418A1 (en) * 2019-12-24 2022-07-21 Dana-Farber Cancer Institute, Inc. The combination of cyclin dependent kinase 7 inhibitor and immunotherapy for treatment of cancer
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CN114452391B (zh) * 2022-01-28 2023-08-25 深圳市泰尔康生物医药科技有限公司 Cdk16作为靶标在制备用于治疗三阴性乳腺癌的药物中的应用
WO2023246371A1 (zh) * 2022-06-24 2023-12-28 中国科学院基础医学与肿瘤研究所(筹) 具有嘧啶并噻吩结构的小分子化合物及其应用

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