UY33539A - Compuestos químicos alk - Google Patents
Compuestos químicos alkInfo
- Publication number
- UY33539A UY33539A UY0001033539A UY33539A UY33539A UY 33539 A UY33539 A UY 33539A UY 0001033539 A UY0001033539 A UY 0001033539A UY 33539 A UY33539 A UY 33539A UY 33539 A UY33539 A UY 33539A
- Authority
- UY
- Uruguay
- Prior art keywords
- alk
- chemical compounds
- formula
- methods
- compounds
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 3
- 101710168331 ALK tyrosine kinase receptor Proteins 0.000 abstract 1
- 102100033793 ALK tyrosine kinase receptor Human genes 0.000 abstract 1
- 206010028980 Neoplasm Diseases 0.000 abstract 1
- 201000011510 cancer Diseases 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6564—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms
- C07F9/6568—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms having phosphorus atoms as the only ring hetero atoms
- C07F9/65685—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms having phosphorus atoms as the only ring hetero atoms the ring phosphorus atom being part of a phosphine oxide or thioxide
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
La presente invención se refiere a compuestos de Fórmula (I) y/o Fórmula (Ia) y a sus sales, composiciones farmacéuticas, métodos de empleo y métodos para su preparación. Estos compuestos inhiben la actividad cinasa de ALK y, por lo tanto, se pueden utilizar para tratar el cáncer.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US36991710P | 2010-08-02 | 2010-08-02 | |
US37205510P | 2010-08-09 | 2010-08-09 | |
US39094410P | 2010-10-07 | 2010-10-07 |
Publications (1)
Publication Number | Publication Date |
---|---|
UY33539A true UY33539A (es) | 2012-02-29 |
Family
ID=45527326
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UY0001033539A UY33539A (es) | 2010-08-02 | 2011-08-01 | Compuestos químicos alk |
Country Status (14)
Country | Link |
---|---|
US (1) | US8461170B2 (es) |
EP (1) | EP2601186A2 (es) |
JP (1) | JP2013534221A (es) |
KR (1) | KR20130096241A (es) |
CN (1) | CN103153982A (es) |
AR (1) | AR089550A1 (es) |
AU (1) | AU2011287386A1 (es) |
BR (1) | BR112013002587A2 (es) |
CA (1) | CA2805827A1 (es) |
MX (1) | MX2013001361A (es) |
RU (1) | RU2013109132A (es) |
TW (1) | TW201219383A (es) |
UY (1) | UY33539A (es) |
WO (1) | WO2012017239A2 (es) |
Families Citing this family (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP5427321B2 (ja) | 2011-07-27 | 2014-02-26 | アストラゼネカ アクチボラグ | 2−(2,4,5−置換−アニリノ)ピリミジン化合物 |
CN102899882B (zh) * | 2012-11-07 | 2014-08-06 | 西南大学 | 超亲水涤纶织物的磷酸制备方法 |
CN104876914B (zh) * | 2014-02-28 | 2017-04-19 | 山东轩竹医药科技有限公司 | 嘧啶衍生物类间变性淋巴瘤激酶抑制剂 |
CN105085550B (zh) * | 2014-05-21 | 2017-05-24 | 海门慧聚药业有限公司 | 一类alk激酶抑制剂及其制备方法 |
ES2715500T3 (es) * | 2014-06-19 | 2019-06-04 | Ariad Pharma Inc | Compuestos de heteroarilo para la inhibición de la quinasa |
EP3345906B1 (en) * | 2015-08-31 | 2022-05-25 | Wuxi Shuangliang Biotechnology Co., Ltd. | 2-arylamino pyridine, pyridine or triazine derivative, preparation method and use thereof |
CN106810553B (zh) * | 2015-11-30 | 2020-03-17 | 江苏正大丰海制药有限公司 | 3-(4,5-取代氨基嘧啶)苯基衍生物及其应用 |
KR102444835B1 (ko) | 2016-05-26 | 2022-09-19 | 리커리엄 아이피 홀딩스, 엘엘씨 | Egfr 억제제 화합물 |
PT3514153T (pt) * | 2017-01-26 | 2021-09-22 | Hanmi Pharm Ind Co Ltd | Composto de pirimidina e utilização farmacêutica do mesmo |
CN107995869B (zh) * | 2017-07-26 | 2021-04-16 | 鼎科医疗技术(苏州)有限公司 | 一种表面液化药物涂层球囊 |
KR102548191B1 (ko) * | 2018-04-09 | 2023-06-28 | 상하이테크 유니버시티 | 표적 단백질 분해 화합물, 이의 항종양 응용, 이의 중간체 및 중간체의 응용 |
KR101954370B1 (ko) * | 2018-07-25 | 2019-03-05 | 한미약품 주식회사 | 피리미딘 화합물 및 이를 포함하는 암의 예방 또는 치료용 약학 조성물 |
EP3942045A1 (en) | 2019-03-21 | 2022-01-26 | Onxeo | A dbait molecule in combination with kinase inhibitor for the treatment of cancer |
EP4054579A1 (en) | 2019-11-08 | 2022-09-14 | Institut National de la Santé et de la Recherche Médicale (INSERM) | Methods for the treatment of cancers that have acquired resistance to kinase inhibitors |
WO2021148581A1 (en) | 2020-01-22 | 2021-07-29 | Onxeo | Novel dbait molecule and its use |
CN113387935B (zh) * | 2021-07-23 | 2022-06-10 | 苏州雅深智慧科技有限公司 | 抑制三突变表皮生长因子受体酪氨酸激酶的化合物及用途 |
CN116763792B (zh) * | 2023-06-19 | 2024-03-12 | 西安国际医学中心医院 | Hg-14-10-04在制备治疗食管鳞癌的药物中的应用 |
Family Cites Families (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB9624482D0 (en) | 1995-12-18 | 1997-01-15 | Zeneca Phaema S A | Chemical compounds |
BR9707495A (pt) | 1996-02-13 | 1999-07-27 | Zeneca Ltd | Derivado de quinazolina processo para a preparação do mesmo composição farmacêutica e processo para a produç o de um efeito antiangiogênico e/ou de redução de permeabilidade vascular em um animal de sangue quente |
KR100489174B1 (ko) | 1996-03-05 | 2005-09-30 | 제네카-파마 소시에떼아노님 | 4-아닐리노퀴나졸린유도체 |
GB9718972D0 (en) | 1996-09-25 | 1997-11-12 | Zeneca Ltd | Chemical compounds |
GB9714249D0 (en) | 1997-07-08 | 1997-09-10 | Angiogene Pharm Ltd | Vascular damaging agents |
GB9900334D0 (en) | 1999-01-07 | 1999-02-24 | Angiogene Pharm Ltd | Tricylic vascular damaging agents |
GB9900752D0 (en) | 1999-01-15 | 1999-03-03 | Angiogene Pharm Ltd | Benzimidazole vascular damaging agents |
IL152682A0 (en) | 2000-05-31 | 2003-06-24 | Astrazeneca Ab | Indole derivatives with vascular damaging activity |
KR20030022264A (ko) | 2000-07-07 | 2003-03-15 | 앤지오젠 파마슈티칼스 리미티드 | 신생 혈관 형성 억제제인 콜치놀 유도체 |
US20050277627A1 (en) | 2000-07-07 | 2005-12-15 | Arnould Jean C | Colchinol derivatives as vascular damaging agents |
CA2633563A1 (en) | 2005-12-23 | 2007-06-28 | Astrazeneca Ab | Antibacterial pyrrolopyridines, pyrrolopyrimidines, and pyrroloazepines |
JP2009541318A (ja) | 2006-06-22 | 2009-11-26 | メルク エンド カムパニー インコーポレーテッド | チロシンキナーゼ阻害剤 |
US20100216779A1 (en) * | 2007-06-01 | 2010-08-26 | Glaxosmithkline Llc | Imidazopyridine Kinase Inhibitors |
CA2696200A1 (en) * | 2007-08-23 | 2009-02-26 | Astrazeneca Ab | 2-anilinopurin-8-ones as inhibitors of ttk/mps1 for the treatment of proliferative disorders |
UY32203A (es) | 2008-10-29 | 2010-05-31 | Astrazeneca Ab | Amino pirimidinas y su uso en terapia |
-
2011
- 2011-08-01 TW TW100127241A patent/TW201219383A/zh unknown
- 2011-08-01 UY UY0001033539A patent/UY33539A/es not_active Application Discontinuation
- 2011-08-02 MX MX2013001361A patent/MX2013001361A/es not_active Application Discontinuation
- 2011-08-02 AU AU2011287386A patent/AU2011287386A1/en not_active Abandoned
- 2011-08-02 AR ARP110102793A patent/AR089550A1/es not_active Application Discontinuation
- 2011-08-02 BR BR112013002587A patent/BR112013002587A2/pt not_active IP Right Cessation
- 2011-08-02 US US13/196,189 patent/US8461170B2/en not_active Expired - Fee Related
- 2011-08-02 RU RU2013109132/04A patent/RU2013109132A/ru not_active Application Discontinuation
- 2011-08-02 JP JP2013522307A patent/JP2013534221A/ja not_active Withdrawn
- 2011-08-02 EP EP11746007.1A patent/EP2601186A2/en not_active Withdrawn
- 2011-08-02 KR KR1020137003860A patent/KR20130096241A/ko not_active Application Discontinuation
- 2011-08-02 CN CN201180047702XA patent/CN103153982A/zh active Pending
- 2011-08-02 WO PCT/GB2011/051465 patent/WO2012017239A2/en active Application Filing
- 2011-08-02 CA CA2805827A patent/CA2805827A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
US8461170B2 (en) | 2013-06-11 |
JP2013534221A (ja) | 2013-09-02 |
WO2012017239A3 (en) | 2012-04-05 |
EP2601186A2 (en) | 2013-06-12 |
CN103153982A (zh) | 2013-06-12 |
MX2013001361A (es) | 2013-05-17 |
KR20130096241A (ko) | 2013-08-29 |
CA2805827A1 (en) | 2012-02-09 |
BR112013002587A2 (pt) | 2019-09-24 |
AR089550A1 (es) | 2014-09-03 |
TW201219383A (en) | 2012-05-16 |
RU2013109132A (ru) | 2014-09-10 |
AU2011287386A1 (en) | 2013-03-07 |
WO2012017239A2 (en) | 2012-02-09 |
US20120028924A1 (en) | 2012-02-02 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
109 | Application deemed to be withdrawn |
Effective date: 20200813 |