JP6664385B2 - Ｂｕｂ１阻害薬としてのベンジル置換インダゾール類 - Google Patents
Ｂｕｂ１阻害薬としてのベンジル置換インダゾール類 Download PDFInfo
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- JP6664385B2 JP6664385B2 JP2017514825A JP2017514825A JP6664385B2 JP 6664385 B2 JP6664385 B2 JP 6664385B2 JP 2017514825 A JP2017514825 A JP 2017514825A JP 2017514825 A JP2017514825 A JP 2017514825A JP 6664385 B2 JP6664385 B2 JP 6664385B2
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- Prior art keywords
- methyl
- amino
- indazol
- difluoro
- alkyl
- Prior art date
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- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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| MA41551A (fr) | 2015-02-20 | 2017-12-26 | Incyte Corp | Hétérocycles bicycliques utilisés en tant qu'inhibiteurs de fgfr4 |
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| TWI794171B (zh) | 2016-05-11 | 2023-03-01 | 美商滬亞生物國際有限公司 | Ｈｄａｃ抑制劑與ｐｄ-ｌ１抑制劑之組合治療 |
| TWI808055B (zh) | 2016-05-11 | 2023-07-11 | 美商滬亞生物國際有限公司 | Hdac 抑制劑與 pd-1 抑制劑之組合治療 |
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| US20170273980A1 (en) | 2017-09-28 |
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| PH12017500509A1 (en) | 2017-08-30 |
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| DOP2017000078A (es) | 2017-06-30 |
| TW201615636A (zh) | 2016-05-01 |
| EA032401B1 (ru) | 2019-05-31 |
| WO2016042084A1 (en) | 2016-03-24 |
| CL2017000654A1 (es) | 2017-12-11 |
| AP2017009803A0 (en) | 2017-03-31 |
| CN107001331A (zh) | 2017-08-01 |
| MX2017003664A (es) | 2017-07-13 |
| PE20170697A1 (es) | 2017-06-24 |
| UY36311A (es) | 2016-04-29 |
| BR112017005444A2 (pt) | 2018-04-24 |
| EP3194379A1 (en) | 2017-07-26 |
| US10350206B2 (en) | 2019-07-16 |
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