JP6664385B2 - Ｂｕｂ１阻害薬としてのベンジル置換インダゾール類 - Google Patents
Ｂｕｂ１阻害薬としてのベンジル置換インダゾール類 Download PDFInfo
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- JP6664385B2 JP6664385B2 JP2017514825A JP2017514825A JP6664385B2 JP 6664385 B2 JP6664385 B2 JP 6664385B2 JP 2017514825 A JP2017514825 A JP 2017514825A JP 2017514825 A JP2017514825 A JP 2017514825A JP 6664385 B2 JP6664385 B2 JP 6664385B2
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- Prior art keywords
- methyl
- amino
- indazol
- difluoro
- alkyl
- Prior art date
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- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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| SG10201708520YA (en) | 2013-04-19 | 2017-12-28 | Incyte Corp | Bicyclic heterocycles as fgfr inhibitors |
| CN105408324A (zh) | 2013-06-21 | 2016-03-16 | 拜耳制药股份公司 | 取代的苄基吡唑 |
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| US9682974B2 (en) | 2013-10-30 | 2017-06-20 | Bayer Pharma Aktiengesellschaft | Heteroaryl substituted pyrazoles |
| RU2685230C2 (ru) | 2014-02-06 | 2019-04-17 | Хептарес Терапьютикс Лимитед | Бициклические азотсодержащие соединения как агонисты М1 мускариновых рецепторов |
| JP6545199B2 (ja) | 2014-06-17 | 2019-07-17 | バイエル ファーマ アクチエンゲゼルシャフト | ３−アミノ−１，５，６，７−テトラヒドロ−４ｈ−インドール−４−オン類 |
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| TWI794171B (zh) | 2016-05-11 | 2023-03-01 | 美商滬亞生物國際有限公司 | Ｈｄａｃ抑制劑與ｐｄ-ｌ１抑制劑之組合治療 |
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| MX2017003664A (es) | 2017-07-13 |
| DOP2017000078A (es) | 2017-06-30 |
| IL251071A0 (en) | 2017-04-30 |
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| AU2015316796A1 (en) | 2017-03-30 |
| CO2017002532A2 (es) | 2017-07-11 |
| WO2016042084A1 (en) | 2016-03-24 |
| KR20170049604A (ko) | 2017-05-10 |
| JP2017530962A (ja) | 2017-10-19 |
| US20170273980A1 (en) | 2017-09-28 |
| UY36311A (es) | 2016-04-29 |
| EA032401B1 (ru) | 2019-05-31 |
| NI201700034A (es) | 2017-06-16 |
| PE20170697A1 (es) | 2017-06-24 |
| TN2017000092A1 (en) | 2018-07-04 |
| ECSP17016797A (es) | 2017-05-31 |
| EP3194379A1 (en) | 2017-07-26 |
| CL2017000654A1 (es) | 2017-12-11 |
| SG11201702082VA (en) | 2017-04-27 |
| CN107001331A (zh) | 2017-08-01 |
| US10350206B2 (en) | 2019-07-16 |
| CR20170100A (es) | 2017-04-24 |
| BR112017005444A2 (pt) | 2018-04-24 |
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