JP5782377B2 - 細胞内カルシウムを調節する化合物 - Google Patents

細胞内カルシウムを調節する化合物 Download PDF

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JP5782377B2
JP5782377B2 JP2011525178A JP2011525178A JP5782377B2 JP 5782377 B2 JP5782377 B2 JP 5782377B2 JP 2011525178 A JP2011525178 A JP 2011525178A JP 2011525178 A JP2011525178 A JP 2011525178A JP 5782377 B2 JP5782377 B2 JP 5782377B2
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calcium
compound
thiophene
carboxylic acid
formula
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JP2012501337A (ja
JP2012501337A5 (enExample
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ヴェリセレビ，ゴヌル
スタウダーマン，ケネス，エー．
ホイッテン，ジェフリー，ピー．
ペイ，ヤズホング
カオ，ジャングオ
ワァング，ズィジュン
ロジャーズ，エバン
ディック，ブライアン
グレイ，ジョナサン
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カルシメディカ，インク．
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  • Diabetes (AREA)
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  • Urology & Nephrology (AREA)
  • Dermatology (AREA)
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  • Gastroenterology & Hepatology (AREA)
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
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JP2011525178A 2008-08-27 2009-08-26 細胞内カルシウムを調節する化合物 Expired - Fee Related JP5782377B2 (ja)

Applications Claiming Priority (13)

Application Number Priority Date Filing Date Title
US9236408P 2008-08-27 2008-08-27
US61/092,364 2008-08-27
US14284609P 2009-01-06 2009-01-06
US61/142,846 2009-01-06
US14373909P 2009-01-09 2009-01-09
US61/143,739 2009-01-09
US15727409P 2009-03-04 2009-03-04
US61/157,274 2009-03-04
US15870209P 2009-03-09 2009-03-09
US15871009P 2009-03-09 2009-03-09
US61/158,710 2009-03-09
US61/158,702 2009-03-09
PCT/US2009/055090 WO2010027875A2 (en) 2008-08-27 2009-08-26 Compounds that modulate intracellular calcium

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JP2012501337A JP2012501337A (ja) 2012-01-19
JP2012501337A5 JP2012501337A5 (enExample) 2012-10-04
JP5782377B2 true JP5782377B2 (ja) 2015-09-24

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US (7) US7981925B2 (enExample)
EP (1) EP2321303B1 (enExample)
JP (1) JP5782377B2 (enExample)
KR (1) KR101724161B1 (enExample)
CN (1) CN102256969A (enExample)
AU (1) AU2009288245B2 (enExample)
BR (1) BRPI0917719A2 (enExample)
CA (1) CA2734500A1 (enExample)
IL (1) IL211391B (enExample)
MX (1) MX2011002149A (enExample)
MY (1) MY157445A (enExample)
RU (1) RU2472791C2 (enExample)
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KR101724161B1 (ko) * 2008-08-27 2017-04-06 칼시메디카, 인크 세포내 칼슘을 조절하는 화합물
US8524763B2 (en) * 2008-09-22 2013-09-03 Calcimedica, Inc. Inhibitors of store operated calcium release
US8618307B2 (en) * 2009-09-16 2013-12-31 Calcimedica, Inc. Compounds that modulate intracellular calcium
US8377970B2 (en) 2009-10-08 2013-02-19 Rhizen Pharmaceuticals Sa Modulators of calcium release-activated calcium channel
US8993612B2 (en) 2009-10-08 2015-03-31 Rhizen Pharmaceuticals Sa Modulators of calcium release-activated calcium channel and methods for treatment of non-small cell lung cancer
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US10703722B2 (en) 2010-04-27 2020-07-07 Calcimedica, Inc. Compounds that modulate intracellular calcium
TWI504404B (zh) * 2010-07-22 2015-10-21 Univ Kaohsiung Medical 用於抑制結腸直腸癌細胞及子宮上皮癌細胞生長轉移之醫藥組合物
WO2012027710A2 (en) 2010-08-27 2012-03-01 Calcimedica Inc. Compounds that modulate intracellular calcium
US20120071516A1 (en) * 2010-09-22 2012-03-22 Calcimedica, Inc. Compounds that modulate intracellular calcium
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US9409898B2 (en) 2012-05-02 2016-08-09 Lupin Limited Substituted pyrazole compounds as CRAC modulators
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WO2014203217A1 (en) 2013-06-21 2014-12-24 Lupin Limited Substituted heterocyclic compounds as crac modulators
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