AU2009288245B2 - Compounds that modulate intracellular calcium - Google Patents

Compounds that modulate intracellular calcium Download PDF

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Publication number
AU2009288245B2
AU2009288245B2 AU2009288245A AU2009288245A AU2009288245B2 AU 2009288245 B2 AU2009288245 B2 AU 2009288245B2 AU 2009288245 A AU2009288245 A AU 2009288245A AU 2009288245 A AU2009288245 A AU 2009288245A AU 2009288245 B2 AU2009288245 B2 AU 2009288245B2
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Australia
Prior art keywords
compound
calcium
thiophene
carboxylic acid
phenyl
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Ceased
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AU2009288245A
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AU2009288245A1 (en
Inventor
Jianguo Cao
Brian Dyck
Jonathan Grey
Yazhong Pei
Evan Rogers
Kenneth A. Stauderman
Gonul Velicelebi
Zhijun Wang
Jeffrey P. Whitten
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Calcimedica Inc
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Calcimedica Inc
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    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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  • Health & Medical Sciences (AREA)
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  • Pharmacology & Pharmacy (AREA)
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  • General Health & Medical Sciences (AREA)
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  • Diabetes (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Neurology (AREA)
  • Pulmonology (AREA)
  • Rheumatology (AREA)
  • Neurosurgery (AREA)
  • Endocrinology (AREA)
  • Biomedical Technology (AREA)
  • Urology & Nephrology (AREA)
  • Hematology (AREA)
  • Dermatology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Emergency Medicine (AREA)
  • Transplantation (AREA)
  • Reproductive Health (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Hospice & Palliative Care (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AU2009288245A 2008-08-27 2009-08-26 Compounds that modulate intracellular calcium Ceased AU2009288245B2 (en)

Applications Claiming Priority (13)

Application Number Priority Date Filing Date Title
US9236408P 2008-08-27 2008-08-27
US61/092,364 2008-08-27
US14284609P 2009-01-06 2009-01-06
US61/142,846 2009-01-06
US14373909P 2009-01-09 2009-01-09
US61/143,739 2009-01-09
US15727409P 2009-03-04 2009-03-04
US61/157,274 2009-03-04
US15870209P 2009-03-09 2009-03-09
US15871009P 2009-03-09 2009-03-09
US61/158,702 2009-03-09
US61/158,710 2009-03-09
PCT/US2009/055090 WO2010027875A2 (en) 2008-08-27 2009-08-26 Compounds that modulate intracellular calcium

Publications (2)

Publication Number Publication Date
AU2009288245A1 AU2009288245A1 (en) 2010-03-11
AU2009288245B2 true AU2009288245B2 (en) 2012-12-20

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AU2009288245A Ceased AU2009288245B2 (en) 2008-08-27 2009-08-26 Compounds that modulate intracellular calcium

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US (7) US7906553B2 (enExample)
EP (1) EP2321303B1 (enExample)
JP (1) JP5782377B2 (enExample)
KR (1) KR101724161B1 (enExample)
CN (1) CN102256969A (enExample)
AU (1) AU2009288245B2 (enExample)
BR (1) BRPI0917719A2 (enExample)
CA (1) CA2734500A1 (enExample)
IL (1) IL211391B (enExample)
MX (1) MX2011002149A (enExample)
MY (1) MY157445A (enExample)
RU (1) RU2472791C2 (enExample)
TW (1) TWI392673B (enExample)
WO (2) WO2010027875A2 (enExample)
ZA (1) ZA201101335B (enExample)

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CA2734500A1 (en) * 2008-08-27 2010-03-11 Calcimedica Inc. Compounds that modulate intracellular calcium
US8524763B2 (en) * 2008-09-22 2013-09-03 Calcimedica, Inc. Inhibitors of store operated calcium release
US8618307B2 (en) * 2009-09-16 2013-12-31 Calcimedica, Inc. Compounds that modulate intracellular calcium
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US8993612B2 (en) 2009-10-08 2015-03-31 Rhizen Pharmaceuticals Sa Modulators of calcium release-activated calcium channel and methods for treatment of non-small cell lung cancer
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CN103180316A (zh) 2010-08-27 2013-06-26 钙医学公司 调节细胞内钙的化合物
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RU2472791C2 (ru) 2013-01-20
US8372991B2 (en) 2013-02-12
AU2009288245A1 (en) 2010-03-11
WO2010025295A3 (en) 2010-06-17
TWI392673B (zh) 2013-04-11
MX2011002149A (es) 2011-04-05
EP2321303B1 (en) 2019-11-27
US8394848B2 (en) 2013-03-12
IL211391B (en) 2018-10-31
WO2010025295A2 (en) 2010-03-04
TW201022256A (en) 2010-06-16
KR101724161B1 (ko) 2017-04-06
US20100056532A1 (en) 2010-03-04
KR20110059723A (ko) 2011-06-03
EP2321303A2 (en) 2011-05-18
US20130231344A1 (en) 2013-09-05
JP5782377B2 (ja) 2015-09-24
US20130245025A1 (en) 2013-09-19
US7981925B2 (en) 2011-07-19

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