JP5688877B2 - 癌疾患の治療用キナゾリン誘導体 - Google Patents

癌疾患の治療用キナゾリン誘導体 Download PDF

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JP5688877B2
JP5688877B2 JP2008539440A JP2008539440A JP5688877B2 JP 5688877 B2 JP5688877 B2 JP 5688877B2 JP 2008539440 A JP2008539440 A JP 2008539440A JP 2008539440 A JP2008539440 A JP 2008539440A JP 5688877 B2 JP5688877 B2 JP 5688877B2
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amino
cancer
patient
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exon
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JP2009515851A5 (enExample
JP2009515851A (ja
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フラヴィオ ゾルカ
フラヴィオ ゾルカ
アンドレー アメルスベルク
アンドレー アメルスベルク
ゲルト シュテーレ
ゲルト シュテーレ
メール ヤコブス セー アー ファン
メール ヤコブス セー アー ファン
アンケ バウム
アンケ バウム
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ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング
ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング
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Application filed by ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング, ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング filed Critical ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/553—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one oxygen as ring hetero atoms, e.g. loxapine, staurosporine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Inorganic Chemistry (AREA)
JP2008539440A 2005-11-11 2006-11-09 癌疾患の治療用キナゾリン誘導体 Active JP5688877B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP05110656.5 2005-11-11
EP05110656 2005-11-11
PCT/EP2006/068313 WO2007054550A1 (en) 2005-11-11 2006-11-09 Quinazoline derivatives for the treatment of cancer diseases

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2013006405A Division JP5695680B2 (ja) 2005-11-11 2013-01-17 癌疾患の治療用キナゾリン誘導体

Publications (3)

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JP2009515851A JP2009515851A (ja) 2009-04-16
JP2009515851A5 JP2009515851A5 (enExample) 2010-01-07
JP5688877B2 true JP5688877B2 (ja) 2015-03-25

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ID=37700909

Family Applications (2)

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JP2008539440A Active JP5688877B2 (ja) 2005-11-11 2006-11-09 癌疾患の治療用キナゾリン誘導体
JP2013006405A Active JP5695680B2 (ja) 2005-11-11 2013-01-17 癌疾患の治療用キナゾリン誘導体

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US (5) US8404697B2 (enExample)
EP (2) EP1948179A1 (enExample)
JP (2) JP5688877B2 (enExample)
CA (3) CA2833852C (enExample)
WO (1) WO2007054550A1 (enExample)

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JP6783224B2 (ja) * 2014-04-04 2020-11-11 デル マー ファーマシューティカルズ 肺の非小細胞癌腫及び卵巣癌を処置するためのジアンヒドロガラクチトール及びその類縁体又は誘導体の使用
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