JP5607038B2 - チアゾリルピペリジン誘導体 - Google Patents
チアゾリルピペリジン誘導体 Download PDFInfo
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- JP5607038B2 JP5607038B2 JP2011515144A JP2011515144A JP5607038B2 JP 5607038 B2 JP5607038 B2 JP 5607038B2 JP 2011515144 A JP2011515144 A JP 2011515144A JP 2011515144 A JP2011515144 A JP 2011515144A JP 5607038 B2 JP5607038 B2 JP 5607038B2
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- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/22—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
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- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102008029734A DE102008029734A1 (de) | 2008-06-23 | 2008-06-23 | Thiazolyl-piperidinderivate |
| DE102008029734.8 | 2008-06-23 | ||
| PCT/EP2009/003817 WO2009156041A2 (de) | 2008-06-23 | 2009-05-28 | Thiazolyl-piperidinderivate |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2011525502A JP2011525502A (ja) | 2011-09-22 |
| JP2011525502A5 JP2011525502A5 (enExample) | 2012-07-12 |
| JP5607038B2 true JP5607038B2 (ja) | 2014-10-15 |
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| Application Number | Title | Priority Date | Filing Date |
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| JP2011515144A Expired - Fee Related JP5607038B2 (ja) | 2008-06-23 | 2009-05-28 | チアゾリルピペリジン誘導体 |
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| US (1) | US8436186B2 (enExample) |
| EP (1) | EP2313403B1 (enExample) |
| JP (1) | JP5607038B2 (enExample) |
| KR (1) | KR20110031349A (enExample) |
| CN (1) | CN102066367A (enExample) |
| AR (1) | AR072192A1 (enExample) |
| AU (1) | AU2009262631B2 (enExample) |
| BR (1) | BRPI0913234A2 (enExample) |
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| WO (1) | WO2009156041A2 (enExample) |
| ZA (1) | ZA201100566B (enExample) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2013514287A (ja) * | 2009-12-17 | 2013-04-25 | メルク パテント ゲゼルシャフト ミット ベシュレンクテル ハフツング | スフィンゴシンキナーゼの阻害薬 |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2008257693B2 (en) * | 2007-06-01 | 2011-01-27 | F. Hoffmann-La Roche Ag | Piperidine-amide derivatives |
| EP2598661B1 (en) | 2010-07-26 | 2017-09-27 | Biomatrica, INC. | Compositions for stabilizing dna, rna and proteins in saliva and other biological samples during shipping and storage at ambient temperatures |
| GB201020161D0 (en) | 2010-11-26 | 2011-01-12 | Almac Discovery Ltd | Pharmaceutical compounds |
| GB2493142A (en) | 2011-07-20 | 2013-01-30 | Johann Wolfgang Goethe Uni T Frankfurt | Ceramide and ceramide synthase in the diagnosis and treatment of multiple sclerosis |
| AU2012354695B2 (en) * | 2011-12-23 | 2016-11-03 | Meiji Seika Pharma Co., Ltd. | Novel S1P receptor modulator |
| US9725703B2 (en) | 2012-12-20 | 2017-08-08 | Biomatrica, Inc. | Formulations and methods for stabilizing PCR reagents |
| WO2014157382A1 (ja) * | 2013-03-29 | 2014-10-02 | 味の素株式会社 | スフィンゴシンキナーゼ阻害剤 |
| WO2015191632A1 (en) | 2014-06-10 | 2015-12-17 | Biomatrica, Inc. | Stabilization of thrombocytes at ambient temperatures |
| EP3174864A4 (en) | 2014-07-31 | 2018-02-14 | Oregon Health & Science University | Vmat inhibitory compounds |
| EP3223807B1 (en) * | 2014-11-24 | 2021-09-15 | The Board of Trustees of the University of Illinois | Method of preventing or treating a pulmonary disease or condition |
| ES2946184T3 (es) | 2015-12-08 | 2023-07-13 | Biomatrica Inc | Reducción de la velocidad de eritrosedimentación |
Family Cites Families (14)
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| GB9624482D0 (en) | 1995-12-18 | 1997-01-15 | Zeneca Phaema S A | Chemical compounds |
| CA2242425C (en) | 1996-02-13 | 2006-07-18 | Zeneca Limited | Quinazoline derivatives as vegf inhibitors |
| NZ331191A (en) | 1996-03-05 | 2000-03-27 | Zeneca Ltd | 4-anilinoquinazoline derivatives and pharmaceutical compositions thereof |
| GB9718972D0 (en) | 1996-09-25 | 1997-11-12 | Zeneca Ltd | Chemical compounds |
| GB9714249D0 (en) | 1997-07-08 | 1997-09-10 | Angiogene Pharm Ltd | Vascular damaging agents |
| GB9900334D0 (en) | 1999-01-07 | 1999-02-24 | Angiogene Pharm Ltd | Tricylic vascular damaging agents |
| GB9900752D0 (en) | 1999-01-15 | 1999-03-03 | Angiogene Pharm Ltd | Benzimidazole vascular damaging agents |
| BR0111230A (pt) | 2000-05-31 | 2003-06-10 | Astrazeneca Ab | Composto, e, uso e processo para a preparação do mesmo |
| KR20030014425A (ko) | 2000-07-07 | 2003-02-17 | 앤지오젠 파마슈티칼스 리미티드 | 혈관 손상제인 콜치놀 유도체 |
| EE200300015A (et) | 2000-07-07 | 2004-10-15 | Angiogene Pharmaceuticals Limited | Kolhinooli derivaadid kui angiogeneesi inhibiitorid |
| ATE498358T1 (de) | 2005-06-29 | 2011-03-15 | Compumedics Ltd | Sensoranordnung mit leitfähiger brücke |
| CA2617788A1 (en) | 2005-08-04 | 2007-02-15 | Apogee Biotechnology Corporation | Sphingosine kinase inhibitors and methods of their use |
| DE602006006712D1 (de) | 2005-08-18 | 2009-06-18 | Hoffmann La Roche | Thiazolylpiperidin-derivate nützlich als h3 rezeptor modulatoren |
| US20090143413A1 (en) | 2005-11-29 | 2009-06-04 | Adams Alan D | Thiazole Derivatives as CXCR3 Receptor Modulators |
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2008
- 2008-06-23 DE DE102008029734A patent/DE102008029734A1/de not_active Withdrawn
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2009
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Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2013514287A (ja) * | 2009-12-17 | 2013-04-25 | メルク パテント ゲゼルシャフト ミット ベシュレンクテル ハフツング | スフィンゴシンキナーゼの阻害薬 |
Also Published As
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| ZA201100566B (en) | 2011-10-26 |
| CN102066367A (zh) | 2011-05-18 |
| AU2009262631A1 (en) | 2009-12-30 |
| MX2010013915A (es) | 2011-02-21 |
| IL210164A0 (en) | 2011-03-31 |
| EP2313403B1 (de) | 2015-04-08 |
| KR20110031349A (ko) | 2011-03-25 |
| WO2009156041A2 (de) | 2009-12-30 |
| CA2728851A1 (en) | 2009-12-30 |
| BRPI0913234A2 (pt) | 2016-01-19 |
| JP2011525502A (ja) | 2011-09-22 |
| DE102008029734A1 (de) | 2009-12-24 |
| US20110105505A1 (en) | 2011-05-05 |
| EP2313403A2 (de) | 2011-04-27 |
| AU2009262631B2 (en) | 2013-08-22 |
| EA201100035A1 (ru) | 2011-08-30 |
| AR072192A1 (es) | 2010-08-11 |
| WO2009156041A3 (de) | 2010-06-10 |
| US8436186B2 (en) | 2013-05-07 |
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