KR20110031349A - 티아졸릴 피페리딘 유도체 - Google Patents
티아졸릴 피페리딘 유도체 Download PDFInfo
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- KR20110031349A KR20110031349A KR1020117001604A KR20117001604A KR20110031349A KR 20110031349 A KR20110031349 A KR 20110031349A KR 1020117001604 A KR1020117001604 A KR 1020117001604A KR 20117001604 A KR20117001604 A KR 20117001604A KR 20110031349 A KR20110031349 A KR 20110031349A
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Classifications
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- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/22—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C07D277/28—Radicals substituted by nitrogen atoms
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
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- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102008029734.8 | 2008-06-23 | ||
| DE102008029734A DE102008029734A1 (de) | 2008-06-23 | 2008-06-23 | Thiazolyl-piperidinderivate |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| KR20110031349A true KR20110031349A (ko) | 2011-03-25 |
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| KR1020117001604A Withdrawn KR20110031349A (ko) | 2008-06-23 | 2009-05-28 | 티아졸릴 피페리딘 유도체 |
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| US (1) | US8436186B2 (enExample) |
| EP (1) | EP2313403B1 (enExample) |
| JP (1) | JP5607038B2 (enExample) |
| KR (1) | KR20110031349A (enExample) |
| CN (1) | CN102066367A (enExample) |
| AR (1) | AR072192A1 (enExample) |
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| MX (1) | MX2010013915A (enExample) |
| WO (1) | WO2009156041A2 (enExample) |
| ZA (1) | ZA201100566B (enExample) |
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| AU2008257693B2 (en) * | 2007-06-01 | 2011-01-27 | F. Hoffmann-La Roche Ag | Piperidine-amide derivatives |
| AU2010341229A1 (en) * | 2009-12-17 | 2012-08-02 | Merck Patent Gmbh | Sphingosine kinase inhibitors |
| WO2012018639A2 (en) | 2010-07-26 | 2012-02-09 | Biomatrica, Inc. | Compositions for stabilizing dna, rna and proteins in saliva and other biological samples during shipping and storage at ambient temperatures |
| GB201020161D0 (en) | 2010-11-26 | 2011-01-12 | Almac Discovery Ltd | Pharmaceutical compounds |
| GB2493142A (en) | 2011-07-20 | 2013-01-30 | Johann Wolfgang Goethe Uni T Frankfurt | Ceramide and ceramide synthase in the diagnosis and treatment of multiple sclerosis |
| JP6033791B2 (ja) * | 2011-12-23 | 2016-11-30 | Ｍｅｉｊｉ Ｓｅｉｋａファルマ株式会社 | 新規ｓ１ｐ受容体調整薬 |
| HK1217117A1 (zh) | 2012-12-20 | 2016-12-23 | 生物马特里卡公司 | 用於使pcr试剂稳定化的制剂和方法 |
| WO2014157382A1 (ja) * | 2013-03-29 | 2014-10-02 | 味の素株式会社 | スフィンゴシンキナーゼ阻害剤 |
| EP3942931A1 (en) | 2014-06-10 | 2022-01-26 | Biomatrica, INC. | Stabilization of thrombocytes at ambient temperatures |
| WO2016019312A2 (en) * | 2014-07-31 | 2016-02-04 | Oregon Health & Science University | Vmat inhibitory compounds |
| WO2016085933A1 (en) | 2014-11-24 | 2016-06-02 | The Board Of Trustees Of The University Of Illinois | Method of preventing or treating a pulmonary disease or condition |
| EP4242628B1 (en) | 2015-12-08 | 2025-07-02 | Biomatrica, Inc. | Reduction of erythrocyte sedimentation rate |
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| GB9624482D0 (en) | 1995-12-18 | 1997-01-15 | Zeneca Phaema S A | Chemical compounds |
| PL194689B1 (pl) | 1996-02-13 | 2007-06-29 | Astrazeneca Uk Ltd | Pochodne chinazoliny, ich kompozycje farmaceutyczne oraz ich zastosowania |
| EP0885198B1 (en) | 1996-03-05 | 2001-12-19 | AstraZeneca AB | 4-anilinoquinazoline derivatives |
| GB9718972D0 (en) | 1996-09-25 | 1997-11-12 | Zeneca Ltd | Chemical compounds |
| GB9714249D0 (en) | 1997-07-08 | 1997-09-10 | Angiogene Pharm Ltd | Vascular damaging agents |
| GB9900334D0 (en) | 1999-01-07 | 1999-02-24 | Angiogene Pharm Ltd | Tricylic vascular damaging agents |
| GB9900752D0 (en) | 1999-01-15 | 1999-03-03 | Angiogene Pharm Ltd | Benzimidazole vascular damaging agents |
| EP1289952A1 (en) | 2000-05-31 | 2003-03-12 | AstraZeneca AB | Indole derivatives with vascular damaging activity |
| CN1255391C (zh) | 2000-07-07 | 2006-05-10 | 安吉奥金尼药品有限公司 | 作为血管破坏剂的colchinol衍生物 |
| WO2002008213A1 (en) | 2000-07-07 | 2002-01-31 | Angiogene Pharmaceuticals Limited | Colchinol derivatives as angiogenesis inhibitors |
| ES2360232T3 (es) | 2005-06-29 | 2011-06-02 | Compumedics Limited | Conjunto sensor con puente conductor. |
| JP2009503107A (ja) | 2005-08-04 | 2009-01-29 | アポジー・バイオテクノロジー・コーポレイション | スフィンゴシンキナーゼ阻害剤およびそれらの使用方法 |
| KR100962827B1 (ko) | 2005-08-18 | 2010-06-10 | 에프. 호프만-라 로슈 아게 | Ｈ3 수용체 조절제로서 유용한 티아졸릴 피페리딘 유도체 |
| EP1957076A2 (en) | 2005-11-29 | 2008-08-20 | Merck & Co., Inc. | Thiazole derivatives as cxcr3 receptor modulators |
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2008
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2009
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- 2009-05-28 EA EA201100035A patent/EA201100035A1/ru unknown
- 2009-05-28 KR KR1020117001604A patent/KR20110031349A/ko not_active Withdrawn
- 2009-05-28 WO PCT/EP2009/003817 patent/WO2009156041A2/de not_active Ceased
- 2009-05-28 BR BRPI0913234A patent/BRPI0913234A2/pt not_active IP Right Cessation
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2010
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2011
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Also Published As
| Publication number | Publication date |
|---|---|
| CN102066367A (zh) | 2011-05-18 |
| DE102008029734A1 (de) | 2009-12-24 |
| US20110105505A1 (en) | 2011-05-05 |
| AU2009262631B2 (en) | 2013-08-22 |
| EP2313403A2 (de) | 2011-04-27 |
| ZA201100566B (en) | 2011-10-26 |
| AR072192A1 (es) | 2010-08-11 |
| US8436186B2 (en) | 2013-05-07 |
| AU2009262631A1 (en) | 2009-12-30 |
| JP5607038B2 (ja) | 2014-10-15 |
| BRPI0913234A2 (pt) | 2016-01-19 |
| WO2009156041A3 (de) | 2010-06-10 |
| CA2728851A1 (en) | 2009-12-30 |
| WO2009156041A2 (de) | 2009-12-30 |
| IL210164A0 (en) | 2011-03-31 |
| EP2313403B1 (de) | 2015-04-08 |
| EA201100035A1 (ru) | 2011-08-30 |
| JP2011525502A (ja) | 2011-09-22 |
| MX2010013915A (es) | 2011-02-21 |
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