JP5438250B2 - オピオイド及びオピオイド様の化合物並びにそれらの使用 - Google Patents

オピオイド及びオピオイド様の化合物並びにそれらの使用 Download PDF

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JP5438250B2
JP5438250B2 JP2004505341A JP2004505341A JP5438250B2 JP 5438250 B2 JP5438250 B2 JP 5438250B2 JP 2004505341 A JP2004505341 A JP 2004505341A JP 2004505341 A JP2004505341 A JP 2004505341A JP 5438250 B2 JP5438250 B2 JP 5438250B2
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pharmaceutical composition
compound
compounds
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mmol
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JP2005530798A (ja
JP2005530798A5 (https=
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イェン，マオ−シュン
ファン，チン−ツァイ
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ジェンケン バイオサイエンスィズ，インコーポレイテッド
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/485—Morphinan derivatives, e.g. morphine, codeine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

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  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Urology & Nephrology (AREA)
  • Rheumatology (AREA)
  • Epidemiology (AREA)
  • Vascular Medicine (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Emergency Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Pulmonology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
JP2004505341A 2002-05-17 2003-05-16 オピオイド及びオピオイド様の化合物並びにそれらの使用 Expired - Fee Related JP5438250B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US38084102P 2002-05-17 2002-05-17
US60/380,841 2002-05-17
PCT/US2003/015461 WO2003097608A2 (en) 2002-05-17 2003-05-16 Opioid and opioid-like compounds and uses thereof

Related Child Applications (1)

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JP2013228118A Division JP6165592B2 (ja) 2002-05-17 2013-11-01 薬学的な組成物

Publications (3)

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JP2005530798A JP2005530798A (ja) 2005-10-13
JP2005530798A5 JP2005530798A5 (https=) 2006-06-29
JP5438250B2 true JP5438250B2 (ja) 2014-03-12

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JP2004505341A Expired - Fee Related JP5438250B2 (ja) 2002-05-17 2003-05-16 オピオイド及びオピオイド様の化合物並びにそれらの使用
JP2013228118A Expired - Fee Related JP6165592B2 (ja) 2002-05-17 2013-11-01 薬学的な組成物
JP2015089558A Expired - Lifetime JP6193298B2 (ja) 2002-05-17 2015-04-24 薬学的な組成物

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JP2013228118A Expired - Fee Related JP6165592B2 (ja) 2002-05-17 2013-11-01 薬学的な組成物
JP2015089558A Expired - Lifetime JP6193298B2 (ja) 2002-05-17 2015-04-24 薬学的な組成物

Country Status (9)

Country Link
EP (2) EP1506174B1 (https=)
JP (3) JP5438250B2 (https=)
CN (2) CN103405431B (https=)
AU (2) AU2003234621A1 (https=)
CA (1) CA2486157C (https=)
HK (1) HK1220452A1 (https=)
MX (1) MXPA04011327A (https=)
TW (1) TWI275591B (https=)
WO (1) WO2003097608A2 (https=)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2521914Y2 (ja) 1988-12-23 1997-01-08 エヌティエヌ株式会社 大型転がり軸受

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JP4805256B2 (ja) * 2004-05-14 2011-11-02 グリーン・クロス・コーポレイション 右旋性モルヒナンの神経保護特性
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Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2521914Y2 (ja) 1988-12-23 1997-01-08 エヌティエヌ株式会社 大型転がり軸受

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AU2010212517A1 (en) 2010-09-16
CN103405431A (zh) 2013-11-27
AU2003234621A1 (en) 2003-12-02
CA2486157A1 (en) 2003-11-27
CN103405431B (zh) 2016-04-13
JP6165592B2 (ja) 2017-07-19
TW200427690A (en) 2004-12-16
WO2003097608A2 (en) 2003-11-27
CN1653050A (zh) 2005-08-10
WO2003097608A3 (en) 2004-03-18
MXPA04011327A (es) 2005-08-15
HK1220452A1 (en) 2017-06-09
HK1192711A1 (zh) 2014-08-29
JP2005530798A (ja) 2005-10-13
JP2014043452A (ja) 2014-03-13
JP2015155449A (ja) 2015-08-27
TWI275591B (en) 2007-03-11
EP1506174B1 (en) 2015-09-30
EP1506174A2 (en) 2005-02-16
EP2987788A1 (en) 2016-02-24
JP6193298B2 (ja) 2017-09-06
CN1653050B (zh) 2013-04-24

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