JP4669611B2 - 化合物 - Google Patents

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Publication number
JP4669611B2
JP4669611B2 JP2000571053A JP2000571053A JP4669611B2 JP 4669611 B2 JP4669611 B2 JP 4669611B2 JP 2000571053 A JP2000571053 A JP 2000571053A JP 2000571053 A JP2000571053 A JP 2000571053A JP 4669611 B2 JP4669611 B2 JP 4669611B2
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compound
formula
mmol
substituents
group
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JP2000571053A
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Japanese (ja)
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JP2002525284A (ja
JP2002525284A5 (https=
Inventor
サーストン，デイビツド・エドウイン
ハワード，フイリツプ・ウイルソン
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スパイロジエン・リミテツド
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pyrrole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
JP2000571053A 1998-08-27 1999-08-27 化合物 Expired - Lifetime JP4669611B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB9818731.3 1998-08-27
GBGB9818731.3A GB9818731D0 (en) 1998-08-27 1998-08-27 Compounds
PCT/GB1999/002837 WO2000012507A2 (en) 1998-08-27 1999-08-27 Pyrrolobenzodiazepines

Publications (3)

Publication Number Publication Date
JP2002525284A JP2002525284A (ja) 2002-08-13
JP2002525284A5 JP2002525284A5 (https=) 2011-01-13
JP4669611B2 true JP4669611B2 (ja) 2011-04-13

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ID=10837953

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2000571053A Expired - Lifetime JP4669611B2 (ja) 1998-08-27 1999-08-27 化合物

Country Status (12)

Country Link
US (2) US6562806B1 (https=)
EP (1) EP1109811B1 (https=)
JP (1) JP4669611B2 (https=)
AT (1) ATE246687T1 (https=)
CA (1) CA2341968C (https=)
DE (1) DE69910227T2 (https=)
DK (1) DK1109811T3 (https=)
ES (1) ES2205872T3 (https=)
GB (1) GB9818731D0 (https=)
NZ (1) NZ510492A (https=)
PT (1) PT1109811E (https=)
WO (1) WO2000012507A2 (https=)

Families Citing this family (145)

* Cited by examiner, † Cited by third party
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GB9818732D0 (en) * 1998-08-27 1998-10-21 Univ Portsmouth Collection of compounds
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FR2835186B1 (fr) 2002-01-28 2006-10-20 Aventis Pharma Sa Nouveaux composes heterocycliques, actifs comme inhibiteurs de beta-lactamases
FR2844273B1 (fr) 2002-09-05 2008-04-04 Aventis Pharma Sa Nouveaux composes heterocycliques, procede et intermediaires de preparation et utilisation comme medicament, notamment comme inhibiteurs de beta-lactamases et anti-bacteriens.
GB0226593D0 (en) * 2002-11-14 2002-12-24 Consultants Ltd Compounds
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