JP4027092B2 - ２−アミノメチル−４−シアノ−チアゾールの製法 - Google Patents

２−アミノメチル−４−シアノ−チアゾールの製法 Download PDF

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Publication number
JP4027092B2
JP4027092B2 JP2001512510A JP2001512510A JP4027092B2 JP 4027092 B2 JP4027092 B2 JP 4027092B2 JP 2001512510 A JP2001512510 A JP 2001512510A JP 2001512510 A JP2001512510 A JP 2001512510A JP 4027092 B2 JP4027092 B2 JP 4027092B2
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JP
Japan
Prior art keywords
formula
thiazole
cyano
boc
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
JP2001512510A
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English (en)
Japanese (ja)
Other versions
JP2003505454A (ja
Inventor
プファイファー トーマス
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
BASF SE
Original Assignee
BASF SE
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by BASF SE filed Critical BASF SE
Publication of JP2003505454A publication Critical patent/JP2003505454A/ja
Application granted granted Critical
Publication of JP4027092B2 publication Critical patent/JP4027092B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06078—Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
JP2001512510A 1999-07-23 2000-07-11 ２−アミノメチル−４−シアノ−チアゾールの製法 Expired - Fee Related JP4027092B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE19933861.2 1999-07-23
DE19933861A DE19933861A1 (de) 1999-07-23 1999-07-23 Verfahren zur Herstellung von 2-Aminomethyl-4-cyano-thiazol
PCT/EP2000/006562 WO2001007425A1 (de) 1999-07-23 2000-07-11 Verfahren zur herstellung von 2-aminomethyl-4-cyano-thiazol

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2006129116A Division JP2006219498A (ja) 1999-07-23 2006-05-08 ２−アミノメチル−４−シアノ−チアゾールの製法

Publications (2)

Publication Number Publication Date
JP2003505454A JP2003505454A (ja) 2003-02-12
JP4027092B2 true JP4027092B2 (ja) 2007-12-26

Family

ID=7915334

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2001512510A Expired - Fee Related JP4027092B2 (ja) 1999-07-23 2000-07-11 ２−アミノメチル−４−シアノ−チアゾールの製法
JP2006129116A Withdrawn JP2006219498A (ja) 1999-07-23 2006-05-08 ２−アミノメチル−４−シアノ−チアゾールの製法

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2006129116A Withdrawn JP2006219498A (ja) 1999-07-23 2006-05-08 ２−アミノメチル−４−シアノ−チアゾールの製法

Country Status (19)

Country Link
US (1) US6642388B1 (pt)
EP (1) EP1196401A1 (pt)
JP (2) JP4027092B2 (pt)
KR (1) KR20020022781A (pt)
CN (1) CN1364163A (pt)
AU (1) AU6157900A (pt)
BG (1) BG106333A (pt)
BR (1) BR0012651A (pt)
CA (1) CA2380084C (pt)
DE (1) DE19933861A1 (pt)
HK (1) HK1048470A1 (pt)
HU (1) HUP0202109A2 (pt)
IL (1) IL147769A0 (pt)
MX (1) MXPA02000716A (pt)
NO (1) NO20020327L (pt)
PL (1) PL355110A1 (pt)
SK (1) SK1052002A3 (pt)
TR (1) TR200200183T2 (pt)
WO (1) WO2001007425A1 (pt)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19934066A1 (de) * 1999-07-23 2001-01-25 Basf Ag Verfahren zur Herstellung von 4-Cyano-2-aminomethylthiazol
JP7148792B2 (ja) 2018-09-27 2022-10-06 日亜化学工業株式会社 光半導体装置用金属材料、及びその製造方法、及びそれを用いた光半導体装置

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19632773A1 (de) * 1996-08-14 1998-02-19 Basf Ag Neue Thrombininhibitoren
EP0928790B1 (en) * 1998-01-02 2003-03-05 F. Hoffmann-La Roche Ag Thiazole derivatives
KR20000047461A (ko) 1998-12-29 2000-07-25 성재갑 트롬빈 억제제
DE19934066A1 (de) * 1999-07-23 2001-01-25 Basf Ag Verfahren zur Herstellung von 4-Cyano-2-aminomethylthiazol

Also Published As

Publication number Publication date
PL355110A1 (en) 2004-04-05
JP2003505454A (ja) 2003-02-12
BG106333A (bg) 2002-08-30
AU6157900A (en) 2001-02-13
EP1196401A1 (de) 2002-04-17
JP2006219498A (ja) 2006-08-24
TR200200183T2 (tr) 2002-08-21
HK1048470A1 (zh) 2003-04-04
WO2001007425A1 (de) 2001-02-01
KR20020022781A (ko) 2002-03-27
DE19933861A1 (de) 2001-01-25
CA2380084C (en) 2007-01-09
NO20020327L (no) 2002-03-21
SK1052002A3 (en) 2002-07-02
BR0012651A (pt) 2002-04-09
NO20020327D0 (no) 2002-01-22
HUP0202109A2 (en) 2002-09-28
CA2380084A1 (en) 2001-02-01
CN1364163A (zh) 2002-08-14
MXPA02000716A (es) 2002-07-22
US6642388B1 (en) 2003-11-04
IL147769A0 (en) 2002-08-14

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