BR0012651A - Processos para preparar 2-aminometil-4-cianotiazol e seus sais, para preparar o composto, e, composto - Google Patents
Processos para preparar 2-aminometil-4-cianotiazol e seus sais, para preparar o composto, e, compostoInfo
- Publication number
- BR0012651A BR0012651A BR0012651-9A BR0012651A BR0012651A BR 0012651 A BR0012651 A BR 0012651A BR 0012651 A BR0012651 A BR 0012651A BR 0012651 A BR0012651 A BR 0012651A
- Authority
- BR
- Brazil
- Prior art keywords
- compound
- preparing
- aminomethyl
- salts
- cyanothiazole
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06008—Dipeptides with the first amino acid being neutral
- C07K5/06078—Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Medicinal Chemistry (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
"PROCESSOS PARA PREPARAR 2-AMINOMETIL-4-CIANOTIAZOL E SEUS SAIS, PARA PREPARAR O COMPOSTO, E, COMPOSTO". A presente invenção refere-se a um processo para produzir 2-aminometil-4-cianotiazol e seus sais de fórmulas gerais (Ia) e (Ib) (Ia) (Ib) nas quais n é 1 ou 2; quando n for 1, então X será cloreto, brometo, triflato e hidrogeno sulfato; e quando n for 2, então X será sulfato. O processo envolve a agitação de tioamida de fórmula (IV) com um éster de ácido bromo-pirúvico de fórmula (V) na qual R^ 1^ é uma C~ 1-4~-aquila linear ou ramificada, em um álcool R^ 2^OH, no qual R^ 2^ é C~ 1-8~-alquila linear ou ramificada, HO-CH~ 2~-CH~ 2~-, HO-CH~ 2~-CH~ 2~-CH~ 2~- ou C~ 1-4~-alquil-O-CH~ 2~-CH~ 2~-. O citado processo de agitação é realizado em uma temperatura de -5<198>C a 40<198>C até que a reação da tioamida de fórmula (IV) esteja praticamente completa. Esta invenção também se refere aos compostos de fórmulas (Ia) e (Ib).
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19933861A DE19933861A1 (de) | 1999-07-23 | 1999-07-23 | Verfahren zur Herstellung von 2-Aminomethyl-4-cyano-thiazol |
| PCT/EP2000/006562 WO2001007425A1 (de) | 1999-07-23 | 2000-07-11 | Verfahren zur herstellung von 2-aminomethyl-4-cyano-thiazol |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR0012651A true BR0012651A (pt) | 2002-04-09 |
Family
ID=7915334
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR0012651-9A BR0012651A (pt) | 1999-07-23 | 2000-07-11 | Processos para preparar 2-aminometil-4-cianotiazol e seus sais, para preparar o composto, e, composto |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US6642388B1 (pt) |
| EP (1) | EP1196401A1 (pt) |
| JP (2) | JP4027092B2 (pt) |
| KR (1) | KR20020022781A (pt) |
| CN (1) | CN1364163A (pt) |
| AU (1) | AU6157900A (pt) |
| BG (1) | BG106333A (pt) |
| BR (1) | BR0012651A (pt) |
| CA (1) | CA2380084C (pt) |
| DE (1) | DE19933861A1 (pt) |
| HK (1) | HK1048470A1 (pt) |
| HU (1) | HUP0202109A2 (pt) |
| IL (1) | IL147769A0 (pt) |
| MX (1) | MXPA02000716A (pt) |
| NO (1) | NO20020327L (pt) |
| PL (1) | PL355110A1 (pt) |
| SK (1) | SK1052002A3 (pt) |
| TR (1) | TR200200183T2 (pt) |
| WO (1) | WO2001007425A1 (pt) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19934066A1 (de) * | 1999-07-23 | 2001-01-25 | Basf Ag | Verfahren zur Herstellung von 4-Cyano-2-aminomethylthiazol |
| JP7148792B2 (ja) | 2018-09-27 | 2022-10-06 | 日亜化学工業株式会社 | 光半導体装置用金属材料、及びその製造方法、及びそれを用いた光半導体装置 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19632773A1 (de) * | 1996-08-14 | 1998-02-19 | Basf Ag | Neue Thrombininhibitoren |
| SI0928790T1 (en) | 1998-01-02 | 2003-06-30 | F. Hoffmann-La Roche Ag | Thiazole derivatives |
| KR20000047461A (ko) | 1998-12-29 | 2000-07-25 | 성재갑 | 트롬빈 억제제 |
| DE19934066A1 (de) * | 1999-07-23 | 2001-01-25 | Basf Ag | Verfahren zur Herstellung von 4-Cyano-2-aminomethylthiazol |
-
1999
- 1999-07-23 DE DE19933861A patent/DE19933861A1/de not_active Withdrawn
-
2000
- 2000-07-11 JP JP2001512510A patent/JP4027092B2/ja not_active Expired - Fee Related
- 2000-07-11 TR TR2002/00183T patent/TR200200183T2/xx unknown
- 2000-07-11 EP EP00947968A patent/EP1196401A1/de not_active Withdrawn
- 2000-07-11 US US10/031,700 patent/US6642388B1/en not_active Expired - Lifetime
- 2000-07-11 CA CA002380084A patent/CA2380084C/en not_active Expired - Fee Related
- 2000-07-11 KR KR1020027000959A patent/KR20020022781A/ko not_active Application Discontinuation
- 2000-07-11 IL IL14776900A patent/IL147769A0/xx unknown
- 2000-07-11 AU AU61579/00A patent/AU6157900A/en not_active Abandoned
- 2000-07-11 CN CN00810618A patent/CN1364163A/zh active Pending
- 2000-07-11 PL PL00355110A patent/PL355110A1/xx not_active Application Discontinuation
- 2000-07-11 WO PCT/EP2000/006562 patent/WO2001007425A1/de not_active Application Discontinuation
- 2000-07-11 HU HU0202109A patent/HUP0202109A2/hu unknown
- 2000-07-11 SK SK105-2002A patent/SK1052002A3/sk not_active Application Discontinuation
- 2000-07-11 MX MXPA02000716A patent/MXPA02000716A/es active IP Right Grant
- 2000-07-11 BR BR0012651-9A patent/BR0012651A/pt not_active IP Right Cessation
-
2002
- 2002-01-21 BG BG106333A patent/BG106333A/bg unknown
- 2002-01-22 NO NO20020327A patent/NO20020327L/no not_active Application Discontinuation
-
2003
- 2003-01-02 HK HK03100004.1A patent/HK1048470A1/zh unknown
-
2006
- 2006-05-08 JP JP2006129116A patent/JP2006219498A/ja not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| HUP0202109A2 (en) | 2002-09-28 |
| CA2380084C (en) | 2007-01-09 |
| BG106333A (bg) | 2002-08-30 |
| SK1052002A3 (en) | 2002-07-02 |
| NO20020327L (no) | 2002-03-21 |
| PL355110A1 (en) | 2004-04-05 |
| WO2001007425A1 (de) | 2001-02-01 |
| CN1364163A (zh) | 2002-08-14 |
| NO20020327D0 (no) | 2002-01-22 |
| JP4027092B2 (ja) | 2007-12-26 |
| AU6157900A (en) | 2001-02-13 |
| IL147769A0 (en) | 2002-08-14 |
| JP2006219498A (ja) | 2006-08-24 |
| DE19933861A1 (de) | 2001-01-25 |
| KR20020022781A (ko) | 2002-03-27 |
| EP1196401A1 (de) | 2002-04-17 |
| TR200200183T2 (tr) | 2002-08-21 |
| CA2380084A1 (en) | 2001-02-01 |
| MXPA02000716A (es) | 2002-07-22 |
| US6642388B1 (en) | 2003-11-04 |
| HK1048470A1 (zh) | 2003-04-04 |
| JP2003505454A (ja) | 2003-02-12 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 3A, 4A, 5A, 6A E 7A ANUIDADES. |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 1927 DE 11/12/2007. |