JP2023530084A5 - - Google Patents

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Publication number
JP2023530084A5
JP2023530084A5 JP2022575997A JP2022575997A JP2023530084A5 JP 2023530084 A5 JP2023530084 A5 JP 2023530084A5 JP 2022575997 A JP2022575997 A JP 2022575997A JP 2022575997 A JP2022575997 A JP 2022575997A JP 2023530084 A5 JP2023530084 A5 JP 2023530084A5
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JP
Japan
Prior art keywords
compound
item
pharmaceutically acceptable
acceptable salt
composition
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JP2022575997A
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English (en)
Japanese (ja)
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JP2023530084A (ja
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Priority claimed from PCT/IB2020/000575 external-priority patent/WO2021111179A1/en
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Publication of JP2023530084A publication Critical patent/JP2023530084A/ja
Publication of JP2023530084A5 publication Critical patent/JP2023530084A5/ja
Priority to JP2025119617A priority Critical patent/JP2025157396A/ja
Withdrawn legal-status Critical Current

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JP2022575997A 2018-12-07 2021-06-09 ４－（２－クロロ－４－メトキシ－５－メチルフェニル）－ｎ－［（１ｓ）－２－シクロプロピル－１－（３－フルオロ－４－メチルフェニル）エチル］－５－メチル－ｎ－プロパ－２－イニル－１，３－チアゾール－２－アミンの調製のための合成法 Withdrawn JP2023530084A (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2025119617A JP2025157396A (ja) 2018-12-07 2025-07-16 ４－（２－クロロ－４－メトキシ－５－メチルフェニル）－ｎ－［（１ｓ）－２－シクロプロピル－１－（３－フルオロ－４－メチルフェニル）エチル］－５－メチル－ｎ－プロパ－２－イニル－１，３－チアゾール－２－アミンの調製のための合成法

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201862776763P 2018-12-07 2018-12-07
US201962816674P 2019-03-11 2019-03-11
IBPCT/IB2020/000575 2020-06-10
PCT/IB2020/000575 WO2021111179A1 (en) 2018-12-07 2020-06-10 Synthetic method for preparation of 4-(2-chloro-4-methoxy-5-methylphenyl)-n-[(1s)-2-cyclopropyl-1-(3-fluoro-4-methylphenyl)ethyl]-5-methyl-n-prop-2-ynyl-1,3-thiazol-2-amine
PCT/IB2021/000403 WO2021250468A2 (en) 2018-12-07 2021-06-09 Synthetic methods for preparation of 4-(2-chloro-4-methoxy-5- methylphenyl)-v-[(ls)-2-cyclopropyl-l-(3-fluoro-4-methylphenyl)ethyl]-5-methyl-v-prop-2-ynyl-l,3-thiazol-2-amine

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2025119617A Division JP2025157396A (ja) 2018-12-07 2025-07-16 ４－（２－クロロ－４－メトキシ－５－メチルフェニル）－ｎ－［（１ｓ）－２－シクロプロピル－１－（３－フルオロ－４－メチルフェニル）エチル］－５－メチル－ｎ－プロパ－２－イニル－１，３－チアゾール－２－アミンの調製のための合成法

Publications (2)

Publication Number Publication Date
JP2023530084A JP2023530084A (ja) 2023-07-13
JP2023530084A5 true JP2023530084A5 (https=) 2024-06-17

Family

ID=69500780

Family Applications (7)

Application Number Title Priority Date Filing Date
JP2021531723A Active JP7238130B2 (ja) 2018-12-07 2019-12-06 先天性副腎過形成を処置するためのｃｒｆ１受容体アンタゴニスト、その医薬製剤および固体形態
JP2022533467A Active JP7675717B6 (ja) 2018-12-07 2020-06-10 ４－（２－クロロ－４－メトキシ－５－メチルフェニル）－ｎ－［（１ｓ）－２－シクロプロピル－１－（３－フルオロ－４－メチルフェニル）エチル］－５－メチル－ｎ－プロパ－２－イニル－１，３－チアゾール－２－アミンの調製のための合成法
JP2022575997A Withdrawn JP2023530084A (ja) 2018-12-07 2021-06-09 ４－（２－クロロ－４－メトキシ－５－メチルフェニル）－ｎ－［（１ｓ）－２－シクロプロピル－１－（３－フルオロ－４－メチルフェニル）エチル］－５－メチル－ｎ－プロパ－２－イニル－１，３－チアゾール－２－アミンの調製のための合成法
JP2023095439A Pending JP2023105239A (ja) 2018-12-07 2023-06-09 ４－（２－クロロ－４－メトキシ－５－メチルフェニル）－ｎ－［（１ｓ）－２－シクロプロピル－１－（３－フルオロ－４－メチルフェニル）エチル］－５－メチル－ｎ－プロパ－２－イニル－１，３－チアゾール－２－アミンの調製のための合成法
JP2024229761A Pending JP2025036615A (ja) 2018-12-07 2024-12-26 ４－（２－クロロ－４－メトキシ－５－メチルフェニル）－ｎ－［（１ｓ）－２－シクロプロピル－１－（３－フルオロ－４－メチルフェニル）エチル］－５－メチル－ｎ－プロパ－２－イニル－１，３－チアゾール－２－アミンの調製のための合成法
JP2025119617A Pending JP2025157396A (ja) 2018-12-07 2025-07-16 ４－（２－クロロ－４－メトキシ－５－メチルフェニル）－ｎ－［（１ｓ）－２－シクロプロピル－１－（３－フルオロ－４－メチルフェニル）エチル］－５－メチル－ｎ－プロパ－２－イニル－１，３－チアゾール－２－アミンの調製のための合成法
JP2026000050A Pending JP2026042855A (ja) 2018-12-07 2026-01-04 ４－（２－クロロ－４－メトキシ－５－メチルフェニル）－ｎ－［（１ｓ）－２－シクロプロピル－１－（３－フルオロ－４－メチルフェニル）エチル］－５－メチル－ｎ－プロパ－２－イニル－１，３－チアゾール－２－アミンの調製のための合成法

Family Applications Before (2)

Application Number Title Priority Date Filing Date
JP2021531723A Active JP7238130B2 (ja) 2018-12-07 2019-12-06 先天性副腎過形成を処置するためのｃｒｆ１受容体アンタゴニスト、その医薬製剤および固体形態
JP2022533467A Active JP7675717B6 (ja) 2018-12-07 2020-06-10 ４－（２－クロロ－４－メトキシ－５－メチルフェニル）－ｎ－［（１ｓ）－２－シクロプロピル－１－（３－フルオロ－４－メチルフェニル）エチル］－５－メチル－ｎ－プロパ－２－イニル－１，３－チアゾール－２－アミンの調製のための合成法

Family Applications After (4)

Application Number Title Priority Date Filing Date
JP2023095439A Pending JP2023105239A (ja) 2018-12-07 2023-06-09 ４－（２－クロロ－４－メトキシ－５－メチルフェニル）－ｎ－［（１ｓ）－２－シクロプロピル－１－（３－フルオロ－４－メチルフェニル）エチル］－５－メチル－ｎ－プロパ－２－イニル－１，３－チアゾール－２－アミンの調製のための合成法
JP2024229761A Pending JP2025036615A (ja) 2018-12-07 2024-12-26 ４－（２－クロロ－４－メトキシ－５－メチルフェニル）－ｎ－［（１ｓ）－２－シクロプロピル－１－（３－フルオロ－４－メチルフェニル）エチル］－５－メチル－ｎ－プロパ－２－イニル－１，３－チアゾール－２－アミンの調製のための合成法
JP2025119617A Pending JP2025157396A (ja) 2018-12-07 2025-07-16 ４－（２－クロロ－４－メトキシ－５－メチルフェニル）－ｎ－［（１ｓ）－２－シクロプロピル－１－（３－フルオロ－４－メチルフェニル）エチル］－５－メチル－ｎ－プロパ－２－イニル－１，３－チアゾール－２－アミンの調製のための合成法
JP2026000050A Pending JP2026042855A (ja) 2018-12-07 2026-01-04 ４－（２－クロロ－４－メトキシ－５－メチルフェニル）－ｎ－［（１ｓ）－２－シクロプロピル－１－（３－フルオロ－４－メチルフェニル）エチル］－５－メチル－ｎ－プロパ－２－イニル－１，３－チアゾール－２－アミンの調製のための合成法

Country Status (27)

Country Link
US (4) US20220023266A1 (https=)
EP (4) EP3890706A2 (https=)
JP (7) JP7238130B2 (https=)
KR (2) KR20210100669A (https=)
CN (7) CN121129756A (https=)
AU (3) AU2019393256B2 (https=)
BR (1) BR112021010847A2 (https=)
CA (3) CA3121920A1 (https=)
DK (1) DK3984523T3 (https=)
ES (1) ES3052613T3 (https=)
FI (1) FI3984523T3 (https=)
HR (1) HRP20251224T1 (https=)
IL (2) IL283712A (https=)
LT (1) LT3984523T (https=)
MA (2) MA54395A (https=)
MD (1) MD3984523T2 (https=)
MX (3) MX2021006552A (https=)
PH (1) PH12021551290A1 (https=)
PL (1) PL3984523T3 (https=)
PT (1) PT3984523T (https=)
RS (1) RS67433B1 (https=)
SA (1) SA521421973B1 (https=)
SG (1) SG11202105930QA (https=)
SI (1) SI3984523T1 (https=)
SM (1) SMT202500435T1 (https=)
TW (3) TWI874339B (https=)
WO (3) WO2020115555A2 (https=)

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