JP2022534704A5 - - Google Patents

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Publication number
JP2022534704A5
JP2022534704A5 JP2021569903A JP2021569903A JP2022534704A5 JP 2022534704 A5 JP2022534704 A5 JP 2022534704A5 JP 2021569903 A JP2021569903 A JP 2021569903A JP 2021569903 A JP2021569903 A JP 2021569903A JP 2022534704 A5 JP2022534704 A5 JP 2022534704A5
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JP
Japan
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group
substituted
alkyl
optionally
aromatic
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
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JP2021569903A
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English (en)
Japanese (ja)
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JP2022534704A (ja
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Priority claimed from PCT/US2020/035848 external-priority patent/WO2020247445A1/en
Publication of JP2022534704A publication Critical patent/JP2022534704A/ja
Publication of JP2022534704A5 publication Critical patent/JP2022534704A5/ja
Pending legal-status Critical Current

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JP2021569903A 2019-06-04 2020-06-03 オレキシンアンタゴニストとしてのイミダゾロ誘導体、組成物、及び方法 Pending JP2022534704A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962856830P 2019-06-04 2019-06-04
US62/856,830 2019-06-04
PCT/US2020/035848 WO2020247445A1 (en) 2019-06-04 2020-06-03 Imidazolo derivatives, compositions and methods as orexin antagonists

Publications (2)

Publication Number Publication Date
JP2022534704A JP2022534704A (ja) 2022-08-03
JP2022534704A5 true JP2022534704A5 (https=) 2023-06-08

Family

ID=73652477

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021569903A Pending JP2022534704A (ja) 2019-06-04 2020-06-03 オレキシンアンタゴニストとしてのイミダゾロ誘導体、組成物、及び方法

Country Status (9)

Country Link
US (2) US12187737B2 (https=)
EP (1) EP3972588A4 (https=)
JP (1) JP2022534704A (https=)
KR (1) KR20220016918A (https=)
CN (1) CN114286675A (https=)
AU (1) AU2020286381C1 (https=)
CA (1) CA3140170A1 (https=)
SG (1) SG11202112827QA (https=)
WO (1) WO2020247445A1 (https=)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2020286381C1 (en) 2019-06-04 2025-07-10 Hager Biosciences, Llc Imidazolo derivatives, compositions and methods as orexin antagonists
AU2020288559C1 (en) * 2019-06-04 2025-07-24 Hager Biosciences, Llc Pyrazole and imidazole derivatives, compositions and methods as orexin antagonists
MX2022007376A (es) 2019-12-20 2022-09-02 Tenaya Therapeutics Inc Fluoroalqull-oxadiazoles y sus usos.
US20240252502A1 (en) 2021-05-04 2024-08-01 Tenaya Therapeutics, Inc. Hdac6 inhibitors for treatment of metabolic disease and hfpef
GB202311281D0 (en) 2023-07-21 2023-09-06 Bial Portela & Ca Sa Orexin receptor antagonists
GB202311280D0 (en) 2023-07-21 2023-09-06 Bial Portela & Ca Sa Orexin receptor antagonists
WO2025101004A1 (ko) * 2023-11-08 2025-05-15 한양대학교 에리카산학협력단 6-aryl imidazo[2,1-b]thi/oxazole-2-carboxilic acid 유도체 및 이를 유효성분으로 함유하는 알츠하이머병 치료용 약학 조성물
WO2025188753A1 (en) * 2024-03-05 2025-09-12 Hager Biosciences, Llc Pyrazole and imidazole derivatives as dual orexin and kappa-opioid receptors modulators, compositions, and methods for treating neurological and psychiatric disorders

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