JP2023507569A5 - - Google Patents

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Publication number
JP2023507569A5
JP2023507569A5 JP2022537497A JP2022537497A JP2023507569A5 JP 2023507569 A5 JP2023507569 A5 JP 2023507569A5 JP 2022537497 A JP2022537497 A JP 2022537497A JP 2022537497 A JP2022537497 A JP 2022537497A JP 2023507569 A5 JP2023507569 A5 JP 2023507569A5
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JP
Japan
Prior art keywords
pharmaceutically acceptable
pharmaceutical composition
composition according
alkyl
polymorph
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2022537497A
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English (en)
Japanese (ja)
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JP2023507569A (ja
JP7737721B2 (ja
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Priority claimed from PCT/US2020/066182 external-priority patent/WO2021127543A1/en
Publication of JP2023507569A publication Critical patent/JP2023507569A/ja
Publication of JP2023507569A5 publication Critical patent/JP2023507569A5/ja
Priority to JP2025075567A priority Critical patent/JP2025107315A/ja
Application granted granted Critical
Publication of JP7737721B2 publication Critical patent/JP7737721B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2022537497A 2019-12-19 2020-12-18 認知障害を処置するためのベンゾジアゼピン誘導体、組成物および方法 Active JP7737721B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2025075567A JP2025107315A (ja) 2019-12-19 2025-04-30 認知障害を処置するためのベンゾジアゼピン誘導体、組成物および方法

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962950886P 2019-12-19 2019-12-19
US62/950,886 2019-12-19
PCT/US2020/066182 WO2021127543A1 (en) 2019-12-19 2020-12-18 Benzodiazepine derivatives, compositions, and methods for treating cognitive impairment

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2025075567A Division JP2025107315A (ja) 2019-12-19 2025-04-30 認知障害を処置するためのベンゾジアゼピン誘導体、組成物および方法

Publications (3)

Publication Number Publication Date
JP2023507569A JP2023507569A (ja) 2023-02-24
JP2023507569A5 true JP2023507569A5 (https=) 2023-12-21
JP7737721B2 JP7737721B2 (ja) 2025-09-11

Family

ID=76478828

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2022537497A Active JP7737721B2 (ja) 2019-12-19 2020-12-18 認知障害を処置するためのベンゾジアゼピン誘導体、組成物および方法
JP2025075567A Pending JP2025107315A (ja) 2019-12-19 2025-04-30 認知障害を処置するためのベンゾジアゼピン誘導体、組成物および方法

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2025075567A Pending JP2025107315A (ja) 2019-12-19 2025-04-30 認知障害を処置するためのベンゾジアゼピン誘導体、組成物および方法

Country Status (8)

Country Link
US (1) US20230098667A1 (https=)
EP (1) EP4077333A4 (https=)
JP (2) JP7737721B2 (https=)
CN (1) CN115175911A (https=)
AU (1) AU2020405233A1 (https=)
IL (1) IL294031A (https=)
MX (1) MX2022007725A (https=)
WO (1) WO2021127543A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20180170941A1 (en) * 2016-12-19 2018-06-21 Agenebio, Inc. Benzodiazepine derivatives, compositions, and methods for treating cognitive impairment
WO2020234880A1 (en) * 2019-05-23 2020-11-26 Life Guard Electrooptic Ltd. System and a method for surveilling swimmers
US20260033761A1 (en) 2022-07-29 2026-02-05 Hoffmann-La Roche Inc. Characterisation of neurological dysfunction
CN120584115A (zh) * 2022-08-19 2025-09-02 艾吉因生物股份有限公司 苯并氮杂䓬衍生物、组合物和用于治疗认知损害的方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ760341A (en) * 2013-12-20 2021-12-24 Agenebio Inc Benzodiazepine derivatives, compositions, and methods for treating cognitive impairment
MX392119B (es) * 2015-06-19 2025-03-11 Agenebio Inc Derivados de benzodiazepina, composiciones y metodos para tratar deterioro cognitivo
US20180170941A1 (en) * 2016-12-19 2018-06-21 Agenebio, Inc. Benzodiazepine derivatives, compositions, and methods for treating cognitive impairment
CN112601749B (zh) * 2018-06-19 2024-03-26 艾吉因生物股份有限公司 用于治疗认知损害的苯并二氮杂环庚三烯衍生物,组合物和方法
CN116075302A (zh) * 2020-07-10 2023-05-05 艾吉因生物股份有限公司 GABAAα5激动剂和SV2A抑制剂的组合以及在认知损害的治疗中的使用方法
WO2022011314A1 (en) * 2020-07-10 2022-01-13 Agenebio, Inc. POLYMORPHS OF A GABAA α5 AGONIST AND METHODS OF USING IN THE TREATMENT OF COGNITIVE IMPAIRMENT

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