JP2019530725A5 - - Google Patents

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Publication number
JP2019530725A5
JP2019530725A5 JP2019520420A JP2019520420A JP2019530725A5 JP 2019530725 A5 JP2019530725 A5 JP 2019530725A5 JP 2019520420 A JP2019520420 A JP 2019520420A JP 2019520420 A JP2019520420 A JP 2019520420A JP 2019530725 A5 JP2019530725 A5 JP 2019530725A5
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JP
Japan
Prior art keywords
ethyl
cyclohexane
cyano
diazepan
dihydrospiro
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JP2019520420A
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English (en)
Japanese (ja)
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JP2019530725A (ja
JP7100634B2 (ja
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Priority claimed from GBGB1617454.2A external-priority patent/GB201617454D0/en
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Publication of JP2019530725A5 publication Critical patent/JP2019530725A5/ja
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Publication of JP7100634B2 publication Critical patent/JP7100634B2/ja
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JP2019520420A 2016-10-14 2017-10-16 Cns疾患及び疼痛の治療におけるムスカリンm1及び/又はm4受容体の調節因子として活性を有する複素環式化合物。 Active JP7100634B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201662408468P 2016-10-14 2016-10-14
GB1617454.2 2016-10-14
GBGB1617454.2A GB201617454D0 (en) 2016-10-14 2016-10-14 Pharmaceutical compounds
US62/408,468 2016-10-14
PCT/GB2017/053115 WO2018069732A1 (en) 2016-10-14 2017-10-16 Heterocyclic compounds having activity as modulators of muscarinic m1 and/or m4 receptors in the treatment of cns diseases and pains.

Publications (3)

Publication Number Publication Date
JP2019530725A JP2019530725A (ja) 2019-10-24
JP2019530725A5 true JP2019530725A5 (https=) 2020-11-26
JP7100634B2 JP7100634B2 (ja) 2022-07-13

Family

ID=57680777

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2019520420A Active JP7100634B2 (ja) 2016-10-14 2017-10-16 Cns疾患及び疼痛の治療におけるムスカリンm1及び/又はm4受容体の調節因子として活性を有する複素環式化合物。

Country Status (8)

Country Link
US (1) US11834407B2 (https=)
EP (1) EP3526207B1 (https=)
JP (1) JP7100634B2 (https=)
CN (1) CN109996792B (https=)
DK (1) DK3526207T3 (https=)
ES (1) ES2898206T3 (https=)
GB (1) GB201617454D0 (https=)
WO (1) WO2018069732A1 (https=)

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GB201819961D0 (en) 2018-12-07 2019-01-23 Heptares Therapeutics Ltd Pharmaceutical compounds
GB202020191D0 (en) 2020-12-18 2021-02-03 Heptares Therapeutics Ltd Pharmaceutical compounds
GB202103211D0 (en) 2021-03-08 2021-04-21 Heptares Therapeutics Ltd Pharmaceutical compounds for use in therapy

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