JP2018520187A5 - - Google Patents

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Publication number
JP2018520187A5
JP2018520187A5 JP2018501972A JP2018501972A JP2018520187A5 JP 2018520187 A5 JP2018520187 A5 JP 2018520187A5 JP 2018501972 A JP2018501972 A JP 2018501972A JP 2018501972 A JP2018501972 A JP 2018501972A JP 2018520187 A5 JP2018520187 A5 JP 2018520187A5
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JP
Japan
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pharmaceutical composition
dementia
disease
composition according
parkinson
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Pending
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JP2018501972A
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Japanese (ja)
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JP2018520187A (ja
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Priority claimed from PCT/US2016/042556 external-priority patent/WO2017011767A2/en
Publication of JP2018520187A publication Critical patent/JP2018520187A/ja
Publication of JP2018520187A5 publication Critical patent/JP2018520187A5/ja
Priority to JP2021125769A priority Critical patent/JP2021185144A/ja
Pending legal-status Critical Current

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JP2018501972A 2015-07-15 2016-07-15 神経変性疾患と関連する幻覚の予防および処置のために有用な5−ht2aセロトニン受容体のモジュレーターとしてのジアリールおよびアリールヘテロアリール尿素誘導体 Pending JP2018520187A (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2021125769A JP2021185144A (ja) 2015-07-15 2021-07-30 神経変性疾患と関連する幻覚の予防および処置のために有用な5−ht2aセロトニン受容体のモジュレーターとしてのジアリールおよびアリールヘテロアリール尿素誘導体

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US201562192939P 2015-07-15 2015-07-15
US62/192,939 2015-07-15
US201562236618P 2015-10-02 2015-10-02
US62/236,618 2015-10-02
US201562261381P 2015-12-01 2015-12-01
US62/261,381 2015-12-01
PCT/US2016/042556 WO2017011767A2 (en) 2015-07-15 2016-07-15 Diaryl and arylheteroaryl urea derivatives as modulators of the 5-ht2a serotonin receptor useful for the prophylaxis and treatment of hallucinations associated with a neurodegenerative disease

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2021125769A Division JP2021185144A (ja) 2015-07-15 2021-07-30 神経変性疾患と関連する幻覚の予防および処置のために有用な5−ht2aセロトニン受容体のモジュレーターとしてのジアリールおよびアリールヘテロアリール尿素誘導体

Publications (2)

Publication Number Publication Date
JP2018520187A JP2018520187A (ja) 2018-07-26
JP2018520187A5 true JP2018520187A5 (OSRAM) 2019-08-22

Family

ID=57757714

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2018501972A Pending JP2018520187A (ja) 2015-07-15 2016-07-15 神経変性疾患と関連する幻覚の予防および処置のために有用な5−ht2aセロトニン受容体のモジュレーターとしてのジアリールおよびアリールヘテロアリール尿素誘導体
JP2021125769A Pending JP2021185144A (ja) 2015-07-15 2021-07-30 神経変性疾患と関連する幻覚の予防および処置のために有用な5−ht2aセロトニン受容体のモジュレーターとしてのジアリールおよびアリールヘテロアリール尿素誘導体

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2021125769A Pending JP2021185144A (ja) 2015-07-15 2021-07-30 神経変性疾患と関連する幻覚の予防および処置のために有用な5−ht2aセロトニン受容体のモジュレーターとしてのジアリールおよびアリールヘテロアリール尿素誘導体

Country Status (14)

Country Link
US (3) US10034859B2 (OSRAM)
EP (1) EP3322415A4 (OSRAM)
JP (2) JP2018520187A (OSRAM)
KR (1) KR20180064373A (OSRAM)
CN (1) CN108472285A (OSRAM)
AU (1) AU2016291673A1 (OSRAM)
BR (1) BR112018000728A2 (OSRAM)
CA (1) CA2992518A1 (OSRAM)
HK (1) HK1247555A1 (OSRAM)
IL (1) IL256831A (OSRAM)
MX (1) MX391031B (OSRAM)
RU (1) RU2018103338A (OSRAM)
TW (1) TW201720439A (OSRAM)
WO (1) WO2017011767A2 (OSRAM)

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WO2017165635A1 (en) 2016-03-25 2017-09-28 Acadia Pharmaceuticals Inc. Combination of pimavanserin and cytochrome p450 modulators
WO2017172757A1 (en) * 2016-03-29 2017-10-05 Acadia Pharmaceuticals Inc. 5-ht2a serotonin receptor inverse agonists or antagonists for use in reducing amyloid-beta peptides and accumulation of amyloid plaques
EP3558311A1 (en) 2016-12-20 2019-10-30 Acadia Pharmaceuticals Inc. Pimavanserin alone or in combination for use in the treatment of alzheimer's disease psychosis
WO2018148737A1 (en) * 2017-02-13 2018-08-16 Axovant Sciences Gmbh 5-ht2a serotonin receptor serotonin receptor inverse agonists useful for the prophylaxis and treatment of parkinsonian symptoms associated with a neurodegenerative disease
US11135211B2 (en) 2017-04-28 2021-10-05 Acadia Pharmaceuticals Inc. Pimavanserin for treating impulse control disorder
WO2019033068A1 (en) * 2017-08-10 2019-02-14 Axovant Sciences Gmbh USE OF INVERSE AGONISTS OF 5 HT2A FOR THE TREATMENT OF PSYCHOSES
EP3675827A1 (en) 2017-08-30 2020-07-08 Acadia Pharmaceuticals Inc. Formulations of pimavanserin
US11622970B2 (en) 2020-04-28 2023-04-11 Prelude Therapeutics Incorporation BCL-2 inhibitors and their use as pharmaceuticals
US20230346811A1 (en) * 2020-09-18 2023-11-02 Mydecine Innovations Group Inc. Novel Formulations of Psilocybin And Psilocin Compounds as Serotonin Agonists in Combination With 3,4 Methylenedioxymethamphetamine (MDMA)
USD980157S1 (en) * 2021-02-26 2023-03-07 The Goodyear Tire & Rubber Company Tire
CN116354925B (zh) * 2021-12-27 2025-09-09 江苏恩华药业股份有限公司 吡唑衍生物及其应用

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