JP2018508537A5 - - Google Patents

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Publication number
JP2018508537A5
JP2018508537A5 JP2017546856A JP2017546856A JP2018508537A5 JP 2018508537 A5 JP2018508537 A5 JP 2018508537A5 JP 2017546856 A JP2017546856 A JP 2017546856A JP 2017546856 A JP2017546856 A JP 2017546856A JP 2018508537 A5 JP2018508537 A5 JP 2018508537A5
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JP
Japan
Prior art keywords
compound
salt
formula
base
derivative
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JP2017546856A
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English (en)
Japanese (ja)
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JP6773672B2 (ja
JP2018508537A (ja
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Priority claimed from PCT/US2016/021085 external-priority patent/WO2016144833A1/en
Publication of JP2018508537A publication Critical patent/JP2018508537A/ja
Publication of JP2018508537A5 publication Critical patent/JP2018508537A5/ja
Application granted granted Critical
Publication of JP6773672B2 publication Critical patent/JP6773672B2/ja
Active legal-status Critical Current
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JP2017546856A 2015-03-06 2016-03-05 フルオロケトライドを調製するための方法 Active JP6773672B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201562129305P 2015-03-06 2015-03-06
US62/129,305 2015-03-06
PCT/US2016/021085 WO2016144833A1 (en) 2015-03-06 2016-03-05 Processes for preparing fluoroketolides

Publications (3)

Publication Number Publication Date
JP2018508537A JP2018508537A (ja) 2018-03-29
JP2018508537A5 true JP2018508537A5 (enExample) 2019-04-18
JP6773672B2 JP6773672B2 (ja) 2020-10-21

Family

ID=56880477

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2017546856A Active JP6773672B2 (ja) 2015-03-06 2016-03-05 フルオロケトライドを調製するための方法

Country Status (19)

Country Link
US (2) US20180044365A1 (enExample)
EP (1) EP3265100A4 (enExample)
JP (1) JP6773672B2 (enExample)
KR (1) KR20170133377A (enExample)
CN (1) CN107405355A (enExample)
AU (1) AU2016230027A1 (enExample)
BR (1) BR112017019176A2 (enExample)
CA (1) CA2978731A1 (enExample)
CL (1) CL2017002255A1 (enExample)
CO (1) CO2017010143A2 (enExample)
HK (1) HK1247097A1 (enExample)
IL (1) IL254306A0 (enExample)
MX (2) MX2017011454A (enExample)
PE (1) PE20180219A1 (enExample)
RU (1) RU2017131253A (enExample)
SG (2) SG11201707215XA (enExample)
TW (1) TW201638102A (enExample)
WO (1) WO2016144833A1 (enExample)
ZA (1) ZA201706505B (enExample)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2214484A4 (en) 2007-10-25 2013-01-02 Cempra Pharmaceuticals Inc PROCESS FOR PREPARING ANTIBACTERIAL MAKROLIDE AGENTS
JP5711135B2 (ja) 2008-10-24 2015-04-30 センプラ ファーマシューティカルズ,インコーポレイテッド 胃腸疾患を治療するための方法
US9937194B1 (en) 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
NZ700182A (en) 2012-03-27 2017-02-24 Cempra Pharmaceuticals Inc Parenteral formulations for administering macrolide antibiotics
AU2014239959A1 (en) 2013-03-14 2015-10-01 Cempra Pharmaceuticals, Inc. Methods for treating respiratory diseases and formulations therefor

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3668282A (en) * 1970-05-08 1972-06-06 Stauffer Chemical Co Stabilized mixture employing n-(beta-0,0-dialkyldithiophosphoryl) aryl sulfonamides
EP1638549A4 (en) * 2003-03-10 2011-06-15 Optimer Pharmaceuticals Inc NEW ANTIBACTERIAL AGENTS
US7595300B2 (en) * 2005-12-13 2009-09-29 Kosan Biosciences Incorporated 7-quinolyl ketolide antibacterial agents
EP2214484A4 (en) * 2007-10-25 2013-01-02 Cempra Pharmaceuticals Inc PROCESS FOR PREPARING ANTIBACTERIAL MAKROLIDE AGENTS
US8283012B2 (en) * 2008-07-24 2012-10-09 Ideo Llc Printable pre-sewn stuffed toy composite sheets
JP5718488B2 (ja) * 2011-03-01 2015-05-13 ウォックハート リミテッド ケトライド中間体の調製方法
AU2014239959A1 (en) * 2013-03-14 2015-10-01 Cempra Pharmaceuticals, Inc. Methods for treating respiratory diseases and formulations therefor
CN105188712A (zh) * 2013-03-15 2015-12-23 森普拉制药公司 用于制备大环内酯抗菌剂的收敛方法
JP6437523B2 (ja) * 2013-04-04 2018-12-12 プレジデント アンド フェローズ オブ ハーバード カレッジ マクロライドならびにそれらの調製および使用の方法

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