TW201638102A - 製備氟酮內酯之方法 - Google Patents
製備氟酮內酯之方法 Download PDFInfo
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- TW201638102A TW201638102A TW105106986A TW105106986A TW201638102A TW 201638102 A TW201638102 A TW 201638102A TW 105106986 A TW105106986 A TW 105106986A TW 105106986 A TW105106986 A TW 105106986A TW 201638102 A TW201638102 A TW 201638102A
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- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H1/00—Processes for the preparation of sugar derivatives
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
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- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
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- Animal Behavior & Ethology (AREA)
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- Communicable Diseases (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Saccharide Compounds (AREA)
- Pyrane Compounds (AREA)
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| WO2010048600A1 (en) | 2008-10-24 | 2010-04-29 | Cempra Pharmaceuticals, Inc. | Methods for treating resistant diseases using triazole containing macrolides |
| US9937194B1 (en) | 2009-06-12 | 2018-04-10 | Cempra Pharmaceuticals, Inc. | Compounds and methods for treating inflammatory diseases |
| WO2013148891A1 (en) | 2012-03-27 | 2013-10-03 | Cempra Pharmaceuticals, Inc. | Parenteral formulations for administering macrolide antibiotics |
| EP2968801B1 (en) | 2013-03-14 | 2018-09-26 | Cempra Pharmaceuticals, Inc. | Methods for treating respiratory diseases and formulations therefor |
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| US3668282A (en) * | 1970-05-08 | 1972-06-06 | Stauffer Chemical Co | Stabilized mixture employing n-(beta-0,0-dialkyldithiophosphoryl) aryl sulfonamides |
| CA2529817C (en) * | 2003-03-10 | 2013-02-12 | Optimer Pharmaceuticals, Inc. | Novel antibacterial agents |
| US7595300B2 (en) * | 2005-12-13 | 2009-09-29 | Kosan Biosciences Incorporated | 7-quinolyl ketolide antibacterial agents |
| AU2008316830B2 (en) * | 2007-10-25 | 2016-03-17 | Cempra Pharmaceuticals, Inc. | Process for the preparation of macrolide antibacterial agents |
| US8376805B2 (en) * | 2008-07-24 | 2013-02-19 | Ideo Llc | Printable pre-sewn stuffed toy composite sheets |
| WO2012117357A2 (en) * | 2011-03-01 | 2012-09-07 | Wockhardt Limited | Process for preparation of ketolide intermediates |
| EP2968801B1 (en) * | 2013-03-14 | 2018-09-26 | Cempra Pharmaceuticals, Inc. | Methods for treating respiratory diseases and formulations therefor |
| MX356772B (es) * | 2013-03-15 | 2018-06-13 | Cempra Pharmaceuticals Inc | Procesos convergentes para la preparacion de agentes antibacterianos macrolidos. |
| CN105246334A (zh) * | 2013-04-04 | 2016-01-13 | 哈佛大学的校长及成员们 | 大环内酯及其制备和使用方法 |
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- 2016-03-05 AU AU2016230027A patent/AU2016230027A1/en not_active Abandoned
- 2016-03-05 PE PE2017001500A patent/PE20180219A1/es not_active Application Discontinuation
- 2016-03-05 HK HK18106628.7A patent/HK1247097A1/zh unknown
- 2016-03-05 SG SG10201908248P patent/SG10201908248PA/en unknown
- 2016-03-05 WO PCT/US2016/021085 patent/WO2016144833A1/en not_active Ceased
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- 2016-03-05 RU RU2017131253A patent/RU2017131253A/ru unknown
- 2016-03-05 MX MX2017011454A patent/MX2017011454A/es unknown
- 2016-03-05 JP JP2017546856A patent/JP6773672B2/ja active Active
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- 2016-03-05 EP EP16762268.7A patent/EP3265100A4/en not_active Withdrawn
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2017
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2020
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| EP3265100A4 (en) | 2019-01-09 |
| WO2016144833A1 (en) | 2016-09-15 |
| HK1247097A1 (zh) | 2018-09-21 |
| MX2017011454A (es) | 2018-01-23 |
| IL254306A0 (en) | 2017-11-30 |
| BR112017019176A2 (pt) | 2018-04-24 |
| US20180044365A1 (en) | 2018-02-15 |
| KR20170133377A (ko) | 2017-12-05 |
| CO2017010143A2 (es) | 2018-02-28 |
| RU2017131253A (ru) | 2019-04-08 |
| US20210070797A1 (en) | 2021-03-11 |
| SG10201908248PA (en) | 2019-10-30 |
| ZA201706505B (en) | 2021-04-28 |
| MX2020007742A (es) | 2020-09-25 |
| SG11201707215XA (en) | 2017-10-30 |
| JP6773672B2 (ja) | 2020-10-21 |
| CA2978731A1 (en) | 2016-09-15 |
| CN107405355A (zh) | 2017-11-28 |
| EP3265100A1 (en) | 2018-01-10 |
| PE20180219A1 (es) | 2018-01-31 |
| CL2017002255A1 (es) | 2018-05-11 |
| AU2016230027A1 (en) | 2017-09-28 |
| JP2018508537A (ja) | 2018-03-29 |
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