BR112017019176A2 - processos para a preparação de fluorocetolídeos - Google Patents

processos para a preparação de fluorocetolídeos

Info

Publication number
BR112017019176A2
BR112017019176A2 BR112017019176A BR112017019176A BR112017019176A2 BR 112017019176 A2 BR112017019176 A2 BR 112017019176A2 BR 112017019176 A BR112017019176 A BR 112017019176A BR 112017019176 A BR112017019176 A BR 112017019176A BR 112017019176 A2 BR112017019176 A2 BR 112017019176A2
Authority
BR
Brazil
Prior art keywords
preparation
fluorocetolides
processes
fluorocetolide
intermediates
Prior art date
Application number
BR112017019176A
Other languages
English (en)
Inventor
Eugene Pereira David
Deo Keshav
e schneider Stephen
Original Assignee
Cempra Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cempra Pharmaceuticals Inc filed Critical Cempra Pharmaceuticals Inc
Publication of BR112017019176A2 publication Critical patent/BR112017019176A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00—Processes for the preparation of sugar derivatives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biotechnology (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Saccharide Compounds (AREA)
  • Pyrane Compounds (AREA)

Abstract

processos e intermediários para a preparação de compostos de fluorocetolídeos são descritos neste documento.
BR112017019176A 2015-03-06 2016-03-05 processos para a preparação de fluorocetolídeos BR112017019176A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201562129305P 2015-03-06 2015-03-06
PCT/US2016/021085 WO2016144833A1 (en) 2015-03-06 2016-03-05 Processes for preparing fluoroketolides

Publications (1)

Publication Number Publication Date
BR112017019176A2 true BR112017019176A2 (pt) 2018-04-24

Family

ID=56880477

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112017019176A BR112017019176A2 (pt) 2015-03-06 2016-03-05 processos para a preparação de fluorocetolídeos

Country Status (19)

Country Link
US (2) US20180044365A1 (pt)
EP (1) EP3265100A4 (pt)
JP (1) JP6773672B2 (pt)
KR (1) KR20170133377A (pt)
CN (1) CN107405355A (pt)
AU (1) AU2016230027A1 (pt)
BR (1) BR112017019176A2 (pt)
CA (1) CA2978731A1 (pt)
CL (1) CL2017002255A1 (pt)
CO (1) CO2017010143A2 (pt)
HK (1) HK1247097A1 (pt)
IL (1) IL254306A0 (pt)
MX (2) MX2017011454A (pt)
PE (1) PE20180219A1 (pt)
RU (1) RU2017131253A (pt)
SG (2) SG11201707215XA (pt)
TW (1) TW201638102A (pt)
WO (1) WO2016144833A1 (pt)
ZA (1) ZA201706505B (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101917850B (zh) 2007-10-25 2016-01-13 森普拉制药公司 大环内酯类抗菌剂的制备方法
ES2565083T3 (es) 2008-10-24 2016-03-31 Cempra Pharmaceuticals, Inc. Biodefensas usando macrólidos que contienen triazol
US9937194B1 (en) 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
KR20140139083A (ko) 2012-03-27 2014-12-04 셈프라 파마슈티컬스, 인크. 마크롤라이드계 항생제를 투여하기 위한 비경구 제제
JP6426696B2 (ja) 2013-03-14 2018-11-21 センプラ ファーマシューティカルズ，インコーポレイテッド 呼吸器疾患の治療のための方法および製剤

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3668282A (en) * 1970-05-08 1972-06-06 Stauffer Chemical Co Stabilized mixture employing n-(beta-0,0-dialkyldithiophosphoryl) aryl sulfonamides
US7601695B2 (en) * 2003-03-10 2009-10-13 Optimer Pharmaceuticals, Inc. Antibacterial agents
US7595300B2 (en) * 2005-12-13 2009-09-29 Kosan Biosciences Incorporated 7-quinolyl ketolide antibacterial agents
CN101917850B (zh) * 2007-10-25 2016-01-13 森普拉制药公司 大环内酯类抗菌剂的制备方法
US8283012B2 (en) * 2008-07-24 2012-10-09 Ideo Llc Printable pre-sewn stuffed toy composite sheets
US9206214B2 (en) * 2011-03-01 2015-12-08 Wockhardt Ltd. Process for preparation of ketolide intermediates
JP6426696B2 (ja) * 2013-03-14 2018-11-21 センプラ ファーマシューティカルズ，インコーポレイテッド 呼吸器疾患の治療のための方法および製剤
AU2014233240B2 (en) * 2013-03-15 2018-08-09 Cempra Pharmaceuticals, Inc. Convergent processes for preparing macrolide antibacterial agents
JP6437523B2 (ja) * 2013-04-04 2018-12-12 プレジデント アンド フェローズ オブ ハーバード カレッジ マクロライドならびにそれらの調製および使用の方法

Also Published As

Publication number Publication date
RU2017131253A (ru) 2019-04-08
PE20180219A1 (es) 2018-01-31
CA2978731A1 (en) 2016-09-15
SG10201908248PA (en) 2019-10-30
EP3265100A4 (en) 2019-01-09
WO2016144833A1 (en) 2016-09-15
SG11201707215XA (en) 2017-10-30
CL2017002255A1 (es) 2018-05-11
AU2016230027A1 (en) 2017-09-28
US20210070797A1 (en) 2021-03-11
IL254306A0 (en) 2017-11-30
ZA201706505B (en) 2021-04-28
MX2020007742A (es) 2020-09-25
HK1247097A1 (zh) 2018-09-21
US20180044365A1 (en) 2018-02-15
CN107405355A (zh) 2017-11-28
EP3265100A1 (en) 2018-01-10
JP2018508537A (ja) 2018-03-29
TW201638102A (zh) 2016-11-01
CO2017010143A2 (es) 2018-02-28
MX2017011454A (es) 2018-01-23
KR20170133377A (ko) 2017-12-05
JP6773672B2 (ja) 2020-10-21

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Legal Events

Date Code Title Description
B11A Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing
B04C Request for examination: application reinstated [chapter 4.3 patent gazette]
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]

Free format text: DE ACORDO COM O ARTIGO 229-C DA LEI NO 10196/2001, QUE MODIFICOU A LEI NO 9279/96, A CONCESSAO DA PATENTE ESTA CONDICIONADA A ANUENCIA PREVIA DA ANVISA. CONSIDERANDO A APROVACAO DOS TERMOS DO PARECER NO 337/PGF/EA/2010, BEM COMO A PORTARIA INTERMINISTERIAL NO 1065 DE 24/05/2012, ENCAMINHA-SE O PRESENTE PEDIDO PARA AS PROVIDENCIAS CABIVEIS.

B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]
B06U Preliminary requirement: requests with searches performed by other patent offices: procedure suspended [chapter 6.21 patent gazette]
B11B Dismissal acc. art. 36, par 1 of ipl - no reply within 90 days to fullfil the necessary requirements
B350 Update of information on the portal [chapter 15.35 patent gazette]