CO2017010143A2 - Procesos para preparar fluorocetólidos - Google Patents

Procesos para preparar fluorocetólidos

Info

Publication number
CO2017010143A2
CO2017010143A2 CONC2017/0010143A CO2017010143A CO2017010143A2 CO 2017010143 A2 CO2017010143 A2 CO 2017010143A2 CO 2017010143 A CO2017010143 A CO 2017010143A CO 2017010143 A2 CO2017010143 A2 CO 2017010143A2
Authority
CO
Colombia
Prior art keywords
processes
fluorocetolides
prepare
fluorocetolide
intermediates
Prior art date
Application number
CONC2017/0010143A
Other languages
English (en)
Inventor
David Eugene Pereira
Stephen E Schneider
Keshav Deo
Original Assignee
Cempra Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cempra Pharmaceuticals Inc filed Critical Cempra Pharmaceuticals Inc
Publication of CO2017010143A2 publication Critical patent/CO2017010143A2/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00Processes for the preparation of sugar derivatives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biotechnology (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Saccharide Compounds (AREA)
  • Pyrane Compounds (AREA)

Abstract

En la presente, se describen procesos e intermediarios para preparar compuestos de fluorocetólido.
CONC2017/0010143A 2015-03-06 2017-10-05 Procesos para preparar fluorocetólidos CO2017010143A2 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201562129305P 2015-03-06 2015-03-06
PCT/US2016/021085 WO2016144833A1 (en) 2015-03-06 2016-03-05 Processes for preparing fluoroketolides

Publications (1)

Publication Number Publication Date
CO2017010143A2 true CO2017010143A2 (es) 2018-02-28

Family

ID=56880477

Family Applications (1)

Application Number Title Priority Date Filing Date
CONC2017/0010143A CO2017010143A2 (es) 2015-03-06 2017-10-05 Procesos para preparar fluorocetólidos

Country Status (19)

Country Link
US (2) US20180044365A1 (es)
EP (1) EP3265100A4 (es)
JP (1) JP6773672B2 (es)
KR (1) KR20170133377A (es)
CN (1) CN107405355A (es)
AU (1) AU2016230027A1 (es)
BR (1) BR112017019176A2 (es)
CA (1) CA2978731A1 (es)
CL (1) CL2017002255A1 (es)
CO (1) CO2017010143A2 (es)
HK (1) HK1247097A1 (es)
IL (1) IL254306A0 (es)
MX (2) MX2017011454A (es)
PE (1) PE20180219A1 (es)
RU (1) RU2017131253A (es)
SG (2) SG11201707215XA (es)
TW (1) TW201638102A (es)
WO (1) WO2016144833A1 (es)
ZA (1) ZA201706505B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101917850B (zh) 2007-10-25 2016-01-13 森普拉制药公司 大环内酯类抗菌剂的制备方法
ES2565083T3 (es) 2008-10-24 2016-03-31 Cempra Pharmaceuticals, Inc. Biodefensas usando macrólidos que contienen triazol
US9937194B1 (en) 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
KR20140139083A (ko) 2012-03-27 2014-12-04 셈프라 파마슈티컬스, 인크. 마크롤라이드계 항생제를 투여하기 위한 비경구 제제
JP6426696B2 (ja) 2013-03-14 2018-11-21 センプラ ファーマシューティカルズ,インコーポレイテッド 呼吸器疾患の治療のための方法および製剤

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3668282A (en) * 1970-05-08 1972-06-06 Stauffer Chemical Co Stabilized mixture employing n-(beta-0,0-dialkyldithiophosphoryl) aryl sulfonamides
US7601695B2 (en) * 2003-03-10 2009-10-13 Optimer Pharmaceuticals, Inc. Antibacterial agents
US7595300B2 (en) * 2005-12-13 2009-09-29 Kosan Biosciences Incorporated 7-quinolyl ketolide antibacterial agents
CN101917850B (zh) * 2007-10-25 2016-01-13 森普拉制药公司 大环内酯类抗菌剂的制备方法
US8283012B2 (en) * 2008-07-24 2012-10-09 Ideo Llc Printable pre-sewn stuffed toy composite sheets
US9206214B2 (en) * 2011-03-01 2015-12-08 Wockhardt Ltd. Process for preparation of ketolide intermediates
JP6426696B2 (ja) * 2013-03-14 2018-11-21 センプラ ファーマシューティカルズ,インコーポレイテッド 呼吸器疾患の治療のための方法および製剤
AU2014233240B2 (en) * 2013-03-15 2018-08-09 Cempra Pharmaceuticals, Inc. Convergent processes for preparing macrolide antibacterial agents
JP6437523B2 (ja) * 2013-04-04 2018-12-12 プレジデント アンド フェローズ オブ ハーバード カレッジ マクロライドならびにそれらの調製および使用の方法

Also Published As

Publication number Publication date
RU2017131253A (ru) 2019-04-08
PE20180219A1 (es) 2018-01-31
CA2978731A1 (en) 2016-09-15
SG10201908248PA (en) 2019-10-30
EP3265100A4 (en) 2019-01-09
WO2016144833A1 (en) 2016-09-15
SG11201707215XA (en) 2017-10-30
CL2017002255A1 (es) 2018-05-11
AU2016230027A1 (en) 2017-09-28
US20210070797A1 (en) 2021-03-11
IL254306A0 (en) 2017-11-30
ZA201706505B (en) 2021-04-28
BR112017019176A2 (pt) 2018-04-24
MX2020007742A (es) 2020-09-25
HK1247097A1 (zh) 2018-09-21
US20180044365A1 (en) 2018-02-15
CN107405355A (zh) 2017-11-28
EP3265100A1 (en) 2018-01-10
JP2018508537A (ja) 2018-03-29
TW201638102A (zh) 2016-11-01
MX2017011454A (es) 2018-01-23
KR20170133377A (ko) 2017-12-05
JP6773672B2 (ja) 2020-10-21

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