PE20180219A1 - Procesos para preparar fluorocetolidos - Google Patents

Procesos para preparar fluorocetolidos

Info

Publication number
PE20180219A1
PE20180219A1 PE2017001500A PE2017001500A PE20180219A1 PE 20180219 A1 PE20180219 A1 PE 20180219A1 PE 2017001500 A PE2017001500 A PE 2017001500A PE 2017001500 A PE2017001500 A PE 2017001500A PE 20180219 A1 PE20180219 A1 PE 20180219A1
Authority
PE
Peru
Prior art keywords
processes
fluorocetolides
prepare
fluoroketolide
intermediates
Prior art date
Application number
PE2017001500A
Other languages
English (en)
Spanish (es)
Inventor
David Eugene Pereira
Stephen E Schneider
Keshav Deo
Original Assignee
Cempra Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cempra Pharmaceuticals Inc filed Critical Cempra Pharmaceuticals Inc
Publication of PE20180219A1 publication Critical patent/PE20180219A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00Processes for the preparation of sugar derivatives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Saccharide Compounds (AREA)
  • Pyrane Compounds (AREA)
PE2017001500A 2015-03-06 2016-03-05 Procesos para preparar fluorocetolidos PE20180219A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201562129305P 2015-03-06 2015-03-06

Publications (1)

Publication Number Publication Date
PE20180219A1 true PE20180219A1 (es) 2018-01-31

Family

ID=56880477

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2017001500A PE20180219A1 (es) 2015-03-06 2016-03-05 Procesos para preparar fluorocetolidos

Country Status (19)

Country Link
US (2) US20180044365A1 (enExample)
EP (1) EP3265100A4 (enExample)
JP (1) JP6773672B2 (enExample)
KR (1) KR20170133377A (enExample)
CN (1) CN107405355A (enExample)
AU (1) AU2016230027A1 (enExample)
BR (1) BR112017019176A2 (enExample)
CA (1) CA2978731A1 (enExample)
CL (1) CL2017002255A1 (enExample)
CO (1) CO2017010143A2 (enExample)
HK (1) HK1247097A1 (enExample)
IL (1) IL254306A0 (enExample)
MX (2) MX2017011454A (enExample)
PE (1) PE20180219A1 (enExample)
RU (1) RU2017131253A (enExample)
SG (2) SG10201908248PA (enExample)
TW (1) TW201638102A (enExample)
WO (1) WO2016144833A1 (enExample)
ZA (1) ZA201706505B (enExample)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2008316830B2 (en) 2007-10-25 2016-03-17 Cempra Pharmaceuticals, Inc. Process for the preparation of macrolide antibacterial agents
WO2010048600A1 (en) 2008-10-24 2010-04-29 Cempra Pharmaceuticals, Inc. Methods for treating resistant diseases using triazole containing macrolides
US9937194B1 (en) 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
WO2013148891A1 (en) 2012-03-27 2013-10-03 Cempra Pharmaceuticals, Inc. Parenteral formulations for administering macrolide antibiotics
EP2968801B1 (en) 2013-03-14 2018-09-26 Cempra Pharmaceuticals, Inc. Methods for treating respiratory diseases and formulations therefor

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3668282A (en) * 1970-05-08 1972-06-06 Stauffer Chemical Co Stabilized mixture employing n-(beta-0,0-dialkyldithiophosphoryl) aryl sulfonamides
CA2529817C (en) * 2003-03-10 2013-02-12 Optimer Pharmaceuticals, Inc. Novel antibacterial agents
US7595300B2 (en) * 2005-12-13 2009-09-29 Kosan Biosciences Incorporated 7-quinolyl ketolide antibacterial agents
AU2008316830B2 (en) * 2007-10-25 2016-03-17 Cempra Pharmaceuticals, Inc. Process for the preparation of macrolide antibacterial agents
US8376805B2 (en) * 2008-07-24 2013-02-19 Ideo Llc Printable pre-sewn stuffed toy composite sheets
WO2012117357A2 (en) * 2011-03-01 2012-09-07 Wockhardt Limited Process for preparation of ketolide intermediates
EP2968801B1 (en) * 2013-03-14 2018-09-26 Cempra Pharmaceuticals, Inc. Methods for treating respiratory diseases and formulations therefor
MX356772B (es) * 2013-03-15 2018-06-13 Cempra Pharmaceuticals Inc Procesos convergentes para la preparacion de agentes antibacterianos macrolidos.
CN105246334A (zh) * 2013-04-04 2016-01-13 哈佛大学的校长及成员们 大环内酯及其制备和使用方法

Also Published As

Publication number Publication date
EP3265100A4 (en) 2019-01-09
WO2016144833A1 (en) 2016-09-15
HK1247097A1 (zh) 2018-09-21
MX2017011454A (es) 2018-01-23
TW201638102A (zh) 2016-11-01
IL254306A0 (en) 2017-11-30
BR112017019176A2 (pt) 2018-04-24
US20180044365A1 (en) 2018-02-15
KR20170133377A (ko) 2017-12-05
CO2017010143A2 (es) 2018-02-28
RU2017131253A (ru) 2019-04-08
US20210070797A1 (en) 2021-03-11
SG10201908248PA (en) 2019-10-30
ZA201706505B (en) 2021-04-28
MX2020007742A (es) 2020-09-25
SG11201707215XA (en) 2017-10-30
JP6773672B2 (ja) 2020-10-21
CA2978731A1 (en) 2016-09-15
CN107405355A (zh) 2017-11-28
EP3265100A1 (en) 2018-01-10
CL2017002255A1 (es) 2018-05-11
AU2016230027A1 (en) 2017-09-28
JP2018508537A (ja) 2018-03-29

Similar Documents

Publication Publication Date Title
CL2016002455A1 (es) Anticuerpos multiespecíficos.
CL2016001871A1 (es) Anticuerpos humanos para pd-1
MX2017006283A (es) Peptidos macrociclicos utiles como inmunomoduladores.
LT3126499T (lt) Kompozicijos, skirtos sod-1 ekspresijos moduliavimui
IT201600117287A1 (it) Metodo di trasfezione transiente per produzione retrovirale.
BR112017002318A2 (pt) combinações de fármacos para tratar mieloma múltiplo.
BR112017022924A2 (pt) métodos para aperfeiçoamento hidráulico de culturas.
BR112017001391A2 (pt) componentes para o fusionamento de corpos vertebrais
IL268683A (en) Processes for preparing ag-10, its intermediates, and salts thereof
CO2017010143A2 (es) Procesos para preparar fluorocetólidos
CL2018003792A1 (es) Procedimiento para enfriamineto de elementos de madera acetilada.
MX389099B (es) Proceso para la preparación de 3-cloro-2-vinilfenilsulfonatos.
MX382631B (es) Proceso para la preparacion de derivados dihidroisoxazol.
MX2015011881A (es) Proceso para la preparacion de 3,7-dimetilnonan-1-ol.
MX380241B (es) Proceso para preparar 3-cloro-2-vinilfenol.
MX2016016398A (es) Preparacion de piperidin-4-carbotioamida.
MX2015009565A (es) Proceso para elaborar derivados de magnolol.
LT3493849T (lt) N,n-bis-2-merkaptoetilizoftalamido naujas panaudojimas
CL2016002925A1 (es) Procedimiento mejorado para preparar ácidos crotónicos sustituidos
UY36284A (es) Método para la preparación de imidazopiridazinas sustituidas
ES2722574R1 (es) Proceso para la preparación de 9beta,10alfa-progesterona (retroprogesterona)
CL2017000400A1 (es) Método de pegilación.
MX390312B (es) Proceso para la preparacion de derivados de fenilisoxazolina sustituida.
TN2014000384A1 (fr) نظام صوتي ذكي وآمن
ES2697706R1 (es) Proceso Para La Preparación De Galeterona.

Legal Events

Date Code Title Description
FD Application declared void or lapsed