PE20180219A1 - Procesos para preparar fluorocetolidos - Google Patents

Procesos para preparar fluorocetolidos

Info

Publication number
PE20180219A1
PE20180219A1 PE2017001500A PE2017001500A PE20180219A1 PE 20180219 A1 PE20180219 A1 PE 20180219A1 PE 2017001500 A PE2017001500 A PE 2017001500A PE 2017001500 A PE2017001500 A PE 2017001500A PE 20180219 A1 PE20180219 A1 PE 20180219A1
Authority
PE
Peru
Prior art keywords
processes
fluorocetolides
prepare
fluoroketolide
intermediates
Prior art date
Application number
PE2017001500A
Other languages
English (en)
Spanish (es)
Inventor
David Eugene Pereira
Stephen E Schneider
Keshav Deo
Original Assignee
Cempra Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cempra Pharmaceuticals Inc filed Critical Cempra Pharmaceuticals Inc
Publication of PE20180219A1 publication Critical patent/PE20180219A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00Processes for the preparation of sugar derivatives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Saccharide Compounds (AREA)
  • Pyrane Compounds (AREA)
PE2017001500A 2015-03-06 2016-03-05 Procesos para preparar fluorocetolidos PE20180219A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201562129305P 2015-03-06 2015-03-06

Publications (1)

Publication Number Publication Date
PE20180219A1 true PE20180219A1 (es) 2018-01-31

Family

ID=56880477

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2017001500A PE20180219A1 (es) 2015-03-06 2016-03-05 Procesos para preparar fluorocetolidos

Country Status (19)

Country Link
US (2) US20180044365A1 (enExample)
EP (1) EP3265100A4 (enExample)
JP (1) JP6773672B2 (enExample)
KR (1) KR20170133377A (enExample)
CN (1) CN107405355A (enExample)
AU (1) AU2016230027A1 (enExample)
BR (1) BR112017019176A2 (enExample)
CA (1) CA2978731A1 (enExample)
CL (1) CL2017002255A1 (enExample)
CO (1) CO2017010143A2 (enExample)
HK (1) HK1247097A1 (enExample)
IL (1) IL254306A0 (enExample)
MX (2) MX2017011454A (enExample)
PE (1) PE20180219A1 (enExample)
RU (1) RU2017131253A (enExample)
SG (2) SG11201707215XA (enExample)
TW (1) TW201638102A (enExample)
WO (1) WO2016144833A1 (enExample)
ZA (1) ZA201706505B (enExample)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2214484A4 (en) 2007-10-25 2013-01-02 Cempra Pharmaceuticals Inc PROCESS FOR PREPARING ANTIBACTERIAL MAKROLIDE AGENTS
JP5711135B2 (ja) 2008-10-24 2015-04-30 センプラ ファーマシューティカルズ,インコーポレイテッド 胃腸疾患を治療するための方法
US9937194B1 (en) 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
NZ700182A (en) 2012-03-27 2017-02-24 Cempra Pharmaceuticals Inc Parenteral formulations for administering macrolide antibiotics
AU2014239959A1 (en) 2013-03-14 2015-10-01 Cempra Pharmaceuticals, Inc. Methods for treating respiratory diseases and formulations therefor

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3668282A (en) * 1970-05-08 1972-06-06 Stauffer Chemical Co Stabilized mixture employing n-(beta-0,0-dialkyldithiophosphoryl) aryl sulfonamides
EP1638549A4 (en) * 2003-03-10 2011-06-15 Optimer Pharmaceuticals Inc NEW ANTIBACTERIAL AGENTS
US7595300B2 (en) * 2005-12-13 2009-09-29 Kosan Biosciences Incorporated 7-quinolyl ketolide antibacterial agents
EP2214484A4 (en) * 2007-10-25 2013-01-02 Cempra Pharmaceuticals Inc PROCESS FOR PREPARING ANTIBACTERIAL MAKROLIDE AGENTS
US8283012B2 (en) * 2008-07-24 2012-10-09 Ideo Llc Printable pre-sewn stuffed toy composite sheets
JP5718488B2 (ja) * 2011-03-01 2015-05-13 ウォックハート リミテッド ケトライド中間体の調製方法
AU2014239959A1 (en) * 2013-03-14 2015-10-01 Cempra Pharmaceuticals, Inc. Methods for treating respiratory diseases and formulations therefor
CN105188712A (zh) * 2013-03-15 2015-12-23 森普拉制药公司 用于制备大环内酯抗菌剂的收敛方法
JP6437523B2 (ja) * 2013-04-04 2018-12-12 プレジデント アンド フェローズ オブ ハーバード カレッジ マクロライドならびにそれらの調製および使用の方法

Also Published As

Publication number Publication date
EP3265100A4 (en) 2019-01-09
MX2020007742A (es) 2020-09-25
SG11201707215XA (en) 2017-10-30
US20180044365A1 (en) 2018-02-15
JP6773672B2 (ja) 2020-10-21
RU2017131253A (ru) 2019-04-08
CA2978731A1 (en) 2016-09-15
JP2018508537A (ja) 2018-03-29
HK1247097A1 (zh) 2018-09-21
TW201638102A (zh) 2016-11-01
US20210070797A1 (en) 2021-03-11
EP3265100A1 (en) 2018-01-10
WO2016144833A1 (en) 2016-09-15
AU2016230027A1 (en) 2017-09-28
IL254306A0 (en) 2017-11-30
CN107405355A (zh) 2017-11-28
ZA201706505B (en) 2021-04-28
SG10201908248PA (en) 2019-10-30
KR20170133377A (ko) 2017-12-05
CO2017010143A2 (es) 2018-02-28
MX2017011454A (es) 2018-01-23
CL2017002255A1 (es) 2018-05-11
BR112017019176A2 (pt) 2018-04-24

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