JP2018501287A5 - - Google Patents

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Publication number
JP2018501287A5
JP2018501287A5 JP2017536301A JP2017536301A JP2018501287A5 JP 2018501287 A5 JP2018501287 A5 JP 2018501287A5 JP 2017536301 A JP2017536301 A JP 2017536301A JP 2017536301 A JP2017536301 A JP 2017536301A JP 2018501287 A5 JP2018501287 A5 JP 2018501287A5
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JP
Japan
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group
alkyl
independently selected
heterocyclyl
oxo
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JP2017536301A
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English (en)
Japanese (ja)
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JP2018501287A (ja
JP6659703B2 (ja
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Priority claimed from PCT/US2016/012659 external-priority patent/WO2016112298A1/en
Publication of JP2018501287A publication Critical patent/JP2018501287A/ja
Publication of JP2018501287A5 publication Critical patent/JP2018501287A5/ja
Application granted granted Critical
Publication of JP6659703B2 publication Critical patent/JP6659703B2/ja
Expired - Fee Related legal-status Critical Current
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JP2017536301A 2015-01-09 2016-01-08 ピリダジノン誘導体および癌の処置におけるそれらの使用 Expired - Fee Related JP6659703B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201562101953P 2015-01-09 2015-01-09
US62/101,953 2015-01-09
PCT/US2016/012659 WO2016112298A1 (en) 2015-01-09 2016-01-08 Pyridazinone derivatives and their use in the treatment of cancer

Publications (3)

Publication Number Publication Date
JP2018501287A JP2018501287A (ja) 2018-01-18
JP2018501287A5 true JP2018501287A5 (enExample) 2019-01-31
JP6659703B2 JP6659703B2 (ja) 2020-03-04

Family

ID=55299747

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2017536301A Expired - Fee Related JP6659703B2 (ja) 2015-01-09 2016-01-08 ピリダジノン誘導体および癌の処置におけるそれらの使用

Country Status (5)

Country Link
US (1) US10239861B2 (enExample)
EP (1) EP3242874B1 (enExample)
JP (1) JP6659703B2 (enExample)
CN (1) CN107406429B (enExample)
WO (1) WO2016112298A1 (enExample)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3189046B1 (en) 2014-09-05 2020-08-26 Genentech, Inc. Therapeutic compounds and uses thereof
CN107074824B (zh) 2014-09-05 2021-01-08 基因泰克公司 作为用于治疗癌症的pcaf和gcn5抑制剂的式(i)的酞嗪衍生物
KR102194536B1 (ko) * 2019-06-10 2020-12-23 연세대학교 산학협력단 타목시펜의 반응성 예측용 조성물
CN112824381B (zh) * 2019-11-21 2024-04-26 广东东阳光药业股份有限公司 一种哌啶胺的制备方法
JP2023529867A (ja) 2020-06-05 2023-07-12 キネート バイオファーマ インク． 線維芽細胞増殖因子受容体キナーゼの阻害剤
US20230391730A1 (en) * 2020-10-09 2023-12-07 Regents Of The University Of Minnesota Inhibitors of the bromodomain phd finger transcription factor (bptf) as anti-cancer agents
KR102766287B1 (ko) * 2021-10-15 2025-02-12 고려대학교 산학협력단 피리다벤을 포함하는 자궁내막 세포, 영양막 세포 또는 고환 세포의 비정상적 증식 관련 질환의 예방 또는 치료용 약학적 조성물
AU2023333181A1 (en) 2022-09-02 2025-03-13 Auron Therapeutics, Inc. Pyridazinon derivatives as kat2 degraders for the treatment of proliferative disorders

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CN107074824B (zh) 2014-09-05 2021-01-08 基因泰克公司 作为用于治疗癌症的pcaf和gcn5抑制剂的式(i)的酞嗪衍生物
EP3189046B1 (en) 2014-09-05 2020-08-26 Genentech, Inc. Therapeutic compounds and uses thereof

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