JP2017533249A5 - - Google Patents

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JP2017533249A5
JP2017533249A5 JP2017525078A JP2017525078A JP2017533249A5 JP 2017533249 A5 JP2017533249 A5 JP 2017533249A5 JP 2017525078 A JP2017525078 A JP 2017525078A JP 2017525078 A JP2017525078 A JP 2017525078A JP 2017533249 A5 JP2017533249 A5 JP 2017533249A5
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methyl
oxo
alkyl
phenyl
heterocyclyl
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JP2017525078A
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JP2017533249A (ja
JP6669745B2 (ja
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Priority claimed from PCT/US2015/060007 external-priority patent/WO2016077380A1/en
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Publication of JP2017533249A5 publication Critical patent/JP2017533249A5/ja
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JP2017525078A 2014-11-10 2015-11-10 ブロモドメインのインヒビターとしての置換ピロロピリジン Expired - Fee Related JP6669745B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201462077707P 2014-11-10 2014-11-10
US62/077,707 2014-11-10
PCT/US2015/060007 WO2016077380A1 (en) 2014-11-10 2015-11-10 Substituted pyrrolopyridines as inhibitors of bromodomain

Publications (3)

Publication Number Publication Date
JP2017533249A JP2017533249A (ja) 2017-11-09
JP2017533249A5 true JP2017533249A5 (enExample) 2018-12-20
JP6669745B2 JP6669745B2 (ja) 2020-03-18

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JP2017525078A Expired - Fee Related JP6669745B2 (ja) 2014-11-10 2015-11-10 ブロモドメインのインヒビターとしての置換ピロロピリジン

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US (1) US10150767B2 (enExample)
EP (1) EP3218374B1 (enExample)
JP (1) JP6669745B2 (enExample)
CN (1) CN107108614B (enExample)
MA (1) MA40940A (enExample)
WO (1) WO2016077380A1 (enExample)

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CN115667237A (zh) * 2020-07-17 2023-01-31 成都苑东生物制药股份有限公司 作为bet抑制剂的新型杂环化合物
TW202237095A (zh) 2020-12-03 2022-10-01 德商艾斯巴赫生物有限公司 Ａｌｃ１抑制劑及與ｐａｒｐｉ之協同性
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TW202330519A (zh) * 2021-09-29 2023-08-01 香港商德琪研發有限公司 作為ｔａｍ抑制劑的吡唑并吡啶化合物
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