JP2017523215A5 - - Google Patents

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JP2017523215A5
JP2017523215A5 JP2017506392A JP2017506392A JP2017523215A5 JP 2017523215 A5 JP2017523215 A5 JP 2017523215A5 JP 2017506392 A JP2017506392 A JP 2017506392A JP 2017506392 A JP2017506392 A JP 2017506392A JP 2017523215 A5 JP2017523215 A5 JP 2017523215A5
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Japan
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amino
pyridin
carboxamide
pyrazine
trifluoromethyl
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JP2017506392A
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Japanese (ja)
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JP2017523215A (ja
JP6644765B2 (ja
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Priority claimed from PCT/IB2015/055951 external-priority patent/WO2016020864A1/en
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Publication of JP2017523215A5 publication Critical patent/JP2017523215A5/ja
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JP2017506392A 2014-08-06 2015-08-05 プロテインキナーゼｃ阻害剤およびその使用方法 Active JP6644765B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201462033679P 2014-08-06 2014-08-06
US62/033,679 2014-08-06
PCT/IB2015/055951 WO2016020864A1 (en) 2014-08-06 2015-08-05 Protein kinase c inhibitors and methods of their use

Publications (3)

Publication Number Publication Date
JP2017523215A JP2017523215A (ja) 2017-08-17
JP2017523215A5 true JP2017523215A5 (enExample) 2018-09-13
JP6644765B2 JP6644765B2 (ja) 2020-02-12

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JP2017506392A Active JP6644765B2 (ja) 2014-08-06 2015-08-05 プロテインキナーゼｃ阻害剤およびその使用方法

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US (7) US9452998B2 (enExample)
EP (3) EP4552697A3 (enExample)
JP (1) JP6644765B2 (enExample)
KR (2) KR102605181B1 (enExample)
CN (2) CN113214246A (enExample)
AP (1) AP2017009729A0 (enExample)
AR (1) AR101456A1 (enExample)
AU (1) AU2015298364B2 (enExample)
BR (1) BR112017002263B1 (enExample)
CA (1) CA2956996C (enExample)
CL (1) CL2017000290A1 (enExample)
CO (1) CO2017001049A2 (enExample)
CR (1) CR20170036A (enExample)
CU (1) CU24465B1 (enExample)
CY (1) CY1122407T1 (enExample)
DK (2) DK3177608T3 (enExample)
DO (1) DOP2017000035A (enExample)
EA (1) EA033361B1 (enExample)
EC (1) ECSP17013903A (enExample)
ES (2) ES2754248T3 (enExample)
FI (1) FI3514151T3 (enExample)
GT (1) GT201700025A (enExample)
HR (2) HRP20192224T1 (enExample)
HU (2) HUE071920T2 (enExample)
IL (1) IL250318B (enExample)
JO (1) JO3589B1 (enExample)
LT (2) LT3514151T (enExample)
MX (1) MX2017001640A (enExample)
MY (1) MY195488A (enExample)
NI (1) NI201700012A (enExample)
PE (1) PE20170241A1 (enExample)
PH (1) PH12017500215B1 (enExample)
PL (2) PL3514151T3 (enExample)
PT (2) PT3514151T (enExample)
RS (2) RS67005B1 (enExample)
SG (1) SG11201700664UA (enExample)
SI (2) SI3177608T1 (enExample)
SM (1) SMT201900703T1 (enExample)
SV (1) SV2017005373A (enExample)
TN (1) TN2017000032A1 (enExample)
TW (1) TWI680968B (enExample)
UY (1) UY36258A (enExample)
WO (1) WO2016020864A1 (enExample)
ZA (1) ZA201700786B (enExample)

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CA3191363A1 (en) * 2020-09-08 2022-03-17 Ideaya Biosciences, Inc. Pharmaceutical combination and tumor treatment
WO2024125543A1 (zh) * 2022-12-16 2024-06-20 苏州科睿思制药有限公司 达洛色替的晶型及其制备方法和用途
WO2025042981A2 (en) * 2023-08-21 2025-02-27 Ideaya Biosciences, Inc. Pharmaceutical compositions comprising a pkc inhibitor
CN117327053A (zh) * 2023-09-20 2024-01-02 云南万宏医药科技有限公司 一种PKC抑制剂darovasertib的制备方法

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