|
US9493484B2
(en)
|
2012-02-08 |
2016-11-15 |
Takeda Pharmaceutical Company Limited |
Heterocyclic compound and use thereof
|
|
JO3225B1
(ar)
*
|
2012-11-27 |
2018-03-08 |
Lilly Co Eli |
6-((s)-1-{1-[5-(2-هيدروكسي-إيثوكسي)-بيريدين-2-يل]-1h-بيرازول-3-يل}إيثيل)-3h-1 ، 3-بنزو ثيازول-2- أون باعتباره مضاد مستقبل ampa يعتمد على tarp- جاما 8
|
|
JP6431088B2
(ja)
|
2014-03-24 |
2018-11-28 |
バイエル・クロップサイエンス・アクチェンゲゼルシャフト |
α,α−ジハロアミン類およびケチミン類からの3,5−ビス(ハロアルキル)ピラゾール誘導体の製造方法
|
|
EP3015458A1
(en)
*
|
2014-11-03 |
2016-05-04 |
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Process for preparing 3,5-bis(haloalkyl)pyrazole derivatives from a,a-dihaloamines and ketimines
|
|
EP4438041A3
(en)
*
|
2016-02-04 |
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|
|
US20190112300A1
(en)
|
2016-03-29 |
2019-04-18 |
Arnold Stan Lippa |
Compositions And Methods For Treating Attention Deficit Disorders
|
|
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(es)
|
2016-06-21 |
2018-10-03 |
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Ácidos de carbamoiloximetil triazol ciclohexilo como antagonistas de lpa
|
|
JP7012703B2
(ja)
|
2017-03-08 |
2022-02-14 |
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|
|
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(en)
|
2017-03-08 |
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|
|
JP6574918B1
(ja)
|
2017-08-03 |
2019-09-11 |
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|
|
JP7189140B2
(ja)
*
|
2017-08-03 |
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|
|
EP3693360B1
(en)
|
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|
|
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(ja)
|
2017-10-06 |
2023-04-03 |
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|
|
WO2019126099A1
(en)
|
2017-12-19 |
2019-06-27 |
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|
|
KR20200100713A
(ko)
|
2017-12-19 |
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|
|
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(en)
|
2017-12-19 |
2019-06-27 |
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Cyclohexyl acid isoxazole azoles as lpa antagonists
|
|
WO2019126093A1
(en)
|
2017-12-19 |
2019-06-27 |
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Cyclohexyl acid triazole azines as lpa antagonists
|
|
AR113964A1
(es)
|
2017-12-19 |
2020-07-01 |
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|
|
US11319309B2
(en)
|
2017-12-19 |
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|
|
ES2925626T3
(es)
|
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|
|
EA039459B1
(ru)
*
|
2017-12-25 |
2022-01-28 |
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|
|
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(zh)
|
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|
|
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(ja)
|
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|
|
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(en)
|
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|
|
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(ko)
|
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|
|
US20220041572A1
(en)
|
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Cycloheptyl acids as lpa antagonists
|
|
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(ja)
|
2018-12-12 |
2023-11-14 |
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|
|
US12091410B2
(en)
|
2018-12-12 |
2024-09-17 |
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Heterocyclic compound
|
|
CN118271298A
(zh)
*
|
2019-01-31 |
2024-07-02 |
武田药品工业株式会社 |
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|
|
TW202045476A
(zh)
|
2019-02-13 |
2020-12-16 |
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5-烷基吡咯啶食慾素受體促效劑
|
|
EP3923933A4
(en)
|
2019-02-13 |
2022-08-17 |
Merck Sharp & Dohme Corp. |
PYRROLIDINOREXINE RECEPTOR AGONISTS
|
|
ES3054967T3
(en)
|
2019-06-18 |
2026-02-09 |
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Triazole carboxylic acids as lpa antagonists
|
|
EP3986552B1
(en)
|
2019-06-18 |
2024-09-18 |
Bristol-Myers Squibb Company |
Isoxazole carboxylic acids as lpa antagonists
|
|
KR102791678B1
(ko)
|
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2025-04-04 |
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Lpa 길항제로서의 시클로부틸 카르복실산
|
|
WO2021026047A1
(en)
|
2019-08-08 |
2021-02-11 |
Merck Sharp & Dohme Corp. |
Heteroaryl pyrrolidine and piperidine orexin receptor agonists
|
|
AU2020394444B2
(en)
|
2019-11-25 |
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Alkermes, Inc. |
Substituted macrocyclic compounds and related methods of treatment
|
|
WO2021106975A1
(ja)
|
2019-11-27 |
2021-06-03 |
武田薬品工業株式会社 |
複素環化合物
|
|
MX2023001840A
(es)
|
2020-08-18 |
2023-03-13 |
Merck Sharp & Dohme Llc |
Agonistas de bicicloheptano pirrolidina de los receptores de orexina.
|
|
US11760747B2
(en)
*
|
2020-12-21 |
2023-09-19 |
Alkermes, Inc. |
Substituted piperidino compounds and related methods of treatment
|
|
US12006330B2
(en)
|
2020-12-21 |
2024-06-11 |
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|
|
WO2023186692A1
(de)
|
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2023-10-05 |
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Verfahren zur herstellung von cis-4-aminotetrahydrofuran-2-carbonsäureestern
|
|
US20250250230A1
(en)
|
2022-04-12 |
2025-08-07 |
Takeda Pharmaceutical Company Limited |
Heterocyclic compound
|
|
EP4543432A1
(en)
*
|
2022-06-21 |
2025-04-30 |
Alkermes, Inc. |
Substituted pyrrolidinyl and piperidinyl compounds and related methods of treatment
|
|
CA3260221A1
(en)
*
|
2022-06-21 |
2023-12-28 |
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Substituted Fused Bicyclic Compounds and Associated Treatment Processes
|
|
JP2025521504A
(ja)
*
|
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|
|
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(zh)
|
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|
|
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(zh)
*
|
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|
|
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(es)
|
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2025-01-29 |
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|
|
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(en)
|
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|
|
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|
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|
|
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|
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|
|
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|
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|
|
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|
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|