JP2016531108A5 - - Google Patents

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Publication number
JP2016531108A5
JP2016531108A5 JP2016528587A JP2016528587A JP2016531108A5 JP 2016531108 A5 JP2016531108 A5 JP 2016531108A5 JP 2016528587 A JP2016528587 A JP 2016528587A JP 2016528587 A JP2016528587 A JP 2016528587A JP 2016531108 A5 JP2016531108 A5 JP 2016531108A5
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JP
Japan
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group
branched
linear
alkyl
compound
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JP2016528587A
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English (en)
Japanese (ja)
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JP6458028B2 (ja
JP2016531108A (ja
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Priority claimed from FR1357277A external-priority patent/FR3008978A1/fr
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Publication of JP2016531108A publication Critical patent/JP2016531108A/ja
Publication of JP2016531108A5 publication Critical patent/JP2016531108A5/ja
Application granted granted Critical
Publication of JP6458028B2 publication Critical patent/JP6458028B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2016528587A 2013-07-23 2014-07-22 インドール及びピロールの新規な誘導体、その製造方法及びそれを含む医薬組成物 Expired - Fee Related JP6458028B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR1357277A FR3008978A1 (fr) 2013-07-23 2013-07-23 "nouveaux derives d'indole et de pyrrole, leur procede de preparation et les compositions pharmaceutiques qui les contiennent"
FR13/57277 2013-07-23
PCT/FR2014/051884 WO2015011396A1 (fr) 2013-07-23 2014-07-22 Nouveaux derives d'indole et de pyrrole, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

Publications (3)

Publication Number Publication Date
JP2016531108A JP2016531108A (ja) 2016-10-06
JP2016531108A5 true JP2016531108A5 (enExample) 2017-08-24
JP6458028B2 JP6458028B2 (ja) 2019-01-23

Family

ID=49911607

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2016528587A Expired - Fee Related JP6458028B2 (ja) 2013-07-23 2014-07-22 インドール及びピロールの新規な誘導体、その製造方法及びそれを含む医薬組成物

Country Status (31)

Country Link
US (2) US9765056B2 (enExample)
EP (2) EP3168217A1 (enExample)
JP (1) JP6458028B2 (enExample)
KR (1) KR102337149B1 (enExample)
CN (1) CN105408321B (enExample)
AR (1) AR099914A1 (enExample)
AU (1) AU2014294866B2 (enExample)
BR (1) BR112016001333B1 (enExample)
CA (1) CA2917965C (enExample)
CY (1) CY1120475T1 (enExample)
DK (1) DK3027602T3 (enExample)
EA (1) EA028609B1 (enExample)
ES (1) ES2687475T3 (enExample)
FR (1) FR3008978A1 (enExample)
HK (1) HK1218753A1 (enExample)
HR (1) HRP20181333T1 (enExample)
HU (1) HUE039507T2 (enExample)
LT (1) LT3027602T (enExample)
MX (1) MX364479B (enExample)
NZ (1) NZ715847A (enExample)
PL (1) PL3027602T3 (enExample)
PT (1) PT3027602T (enExample)
RS (1) RS57545B1 (enExample)
RU (1) RU2693404C2 (enExample)
SG (1) SG11201600004SA (enExample)
SI (1) SI3027602T1 (enExample)
TW (1) TW201504224A (enExample)
UA (1) UA117020C2 (enExample)
UY (1) UY35653A (enExample)
WO (1) WO2015011396A1 (enExample)
ZA (1) ZA201600415B (enExample)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN105237509A (zh) * 2015-11-20 2016-01-13 江苏瑞邦农药厂有限公司 一种2,2-二氟-1,3-苯并二恶茂的合成方法
WO2017197051A1 (en) 2016-05-10 2017-11-16 C4 Therapeutics, Inc. Amine-linked c3-glutarimide degronimers for target protein degradation
WO2017197046A1 (en) 2016-05-10 2017-11-16 C4 Therapeutics, Inc. C3-carbon linked glutarimide degronimers for target protein degradation
ES2989988T3 (es) 2016-05-10 2024-11-28 C4 Therapeutics Inc Degronímeros heterorocíclicos para la degradación de proteínas diana
CN109562113A (zh) 2016-05-10 2019-04-02 C4医药公司 用于靶蛋白降解的螺环降解决定子体
KR102446529B1 (ko) * 2017-01-10 2022-09-23 에테하 취리히 세포 보호 화합물 및 이의 용도
JP6877722B2 (ja) 2017-03-31 2021-05-26 国立大学法人 東京大学 ノロウイルス抗体
CN110769822A (zh) 2017-06-20 2020-02-07 C4医药公司 用于蛋白降解的n/o-连接的降解决定子和降解决定子体
CN108409580A (zh) * 2018-02-01 2018-08-17 浙江工业大学 一种苄胺类化合物的合成方法
CN120698983A (zh) 2018-12-20 2025-09-26 C4医药公司 靶向蛋白降解
US20250387504A1 (en) 2022-05-20 2025-12-25 Novartis Ag Antibody-drug conjugates of antineoplastic compounds and methods of use thereof
TW202540185A (zh) 2023-11-22 2025-10-16 法商施維雅藥廠 抗cd74抗體藥物結合物及其使用方法
WO2025111431A1 (en) 2023-11-22 2025-05-30 Les Laboratoires Servier Anti-cd7 antibody-drug conjugates and methods of use thereof

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2005040128A1 (en) 2003-10-24 2005-05-06 Glaxo Group Limited Heterocyclyl compounds
TW200533398A (en) * 2004-03-29 2005-10-16 Bristol Myers Squibb Co Novel therapeutic agents for the treatment of migraine
CA2577752A1 (en) * 2004-08-20 2006-03-02 The Regents Of The University Of Michigan Small molecule inhibitors of anti-apoptotic bcl-2 family members and the uses thereof
GB0522908D0 (en) 2005-11-10 2005-12-21 Merck Sharp & Dohme Therapeutic agents
US9346795B2 (en) * 2011-05-25 2016-05-24 Bristol-Myers Squibb Company Substituted sulfonamides useful as antiapoptotic Bcl inhibitors
WO2013096055A1 (en) 2011-12-23 2013-06-27 Novartis Ag Compounds for inhibiting the interaction of bcl2 with binding partners
MX2014007731A (es) * 2011-12-23 2015-01-12 Novartis Ag Compuestos para inhibir la interaccion de bcl2 con los componentes de enlace.
CA2859873A1 (en) * 2011-12-23 2013-06-27 Novartis Ag Compounds for inhibiting the interaction of bcl2 with binding partners
CN104125955A (zh) * 2011-12-23 2014-10-29 诺华股份有限公司 用于抑制bcl2与结合配偶体相互作用的化合物
BR112014015322A8 (pt) * 2011-12-23 2017-06-13 Novartis Ag compostos e composições para inibir a interação de bcl2 com parceiros de ligação
FR2986002B1 (fr) 2012-01-24 2014-02-21 Servier Lab Nouveaux derives d'indolizine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

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