JP2012509846A5 - - Google Patents

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Publication number
JP2012509846A5
JP2012509846A5 JP2011532298A JP2011532298A JP2012509846A5 JP 2012509846 A5 JP2012509846 A5 JP 2012509846A5 JP 2011532298 A JP2011532298 A JP 2011532298A JP 2011532298 A JP2011532298 A JP 2011532298A JP 2012509846 A5 JP2012509846 A5 JP 2012509846A5
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JP
Japan
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substituted
pharmaceutical composition
group
amino acid
alkyl
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JP2011532298A
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English (en)
Japanese (ja)
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JP5706825B2 (ja
JP2012509846A (ja
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Priority claimed from PCT/US2009/061068 external-priority patent/WO2010045599A1/en
Publication of JP2012509846A publication Critical patent/JP2012509846A/ja
Publication of JP2012509846A5 publication Critical patent/JP2012509846A5/ja
Application granted granted Critical
Publication of JP5706825B2 publication Critical patent/JP5706825B2/ja
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JP2011532298A 2008-10-17 2009-10-16 フェノール性オピオイドの放出が減弱された医薬組成物 Active JP5706825B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US10640008P 2008-10-17 2008-10-17
US61/106,400 2008-10-17
PCT/US2009/061068 WO2010045599A1 (en) 2008-10-17 2009-10-16 Pharmaceutical compositions with attenuated release of phenolic opioids

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2015037724A Division JP2015129167A (ja) 2008-10-17 2015-02-27 フェノール性オピオイドの放出が減弱された医薬組成物

Publications (3)

Publication Number Publication Date
JP2012509846A JP2012509846A (ja) 2012-04-26
JP2012509846A5 true JP2012509846A5 (https=) 2012-12-06
JP5706825B2 JP5706825B2 (ja) 2015-04-22

Family

ID=41466912

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2011532298A Active JP5706825B2 (ja) 2008-10-17 2009-10-16 フェノール性オピオイドの放出が減弱された医薬組成物
JP2015037724A Pending JP2015129167A (ja) 2008-10-17 2015-02-27 フェノール性オピオイドの放出が減弱された医薬組成物

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2015037724A Pending JP2015129167A (ja) 2008-10-17 2015-02-27 フェノール性オピオイドの放出が減弱された医薬組成物

Country Status (12)

Country Link
US (2) US8802681B2 (https=)
EP (1) EP2349241B1 (https=)
JP (2) JP5706825B2 (https=)
KR (1) KR20110081852A (https=)
CN (1) CN102186467B (https=)
AU (1) AU2009305563C1 (https=)
CA (1) CA2739936C (https=)
IL (1) IL212081A (https=)
MX (1) MX2011004095A (https=)
RU (1) RU2562583C2 (https=)
WO (1) WO2010045599A1 (https=)
ZA (1) ZA201102361B (https=)

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US20110262359A1 (en) * 2010-04-21 2011-10-27 Jenkins Thomas E Compositions comprising enzyme-cleavable prodrugs of active agents and inhibitors thereof
US20130059914A1 (en) 2010-04-21 2013-03-07 Signature Therapeutics, Inc. Compositions Comprising Enzyme-Cleavable Amphetamine Prodrugs and Inhibitors Thereof
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US20110262355A1 (en) 2010-04-21 2011-10-27 Jenkins Thomas E Compositions comprising enzyme-cleavable opioid prodrugs and inhibitors thereof
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WO2012122420A2 (en) * 2011-03-09 2012-09-13 Pharmacofore, Inc. Opioid prodrugs with heterocyclic linkers
AU2012225337B2 (en) * 2011-03-09 2016-04-28 Signature Therapeutics, Inc. Active agent prodrugs with heterocyclic linkers
WO2016064914A1 (en) 2014-10-20 2016-04-28 Elysium Therapeutics, Inc. Diversion-resistant opioid formulations
US11634384B2 (en) 2014-11-25 2023-04-25 Concentric Analgesics, Inc. Prodrugs of phenolic TRPV1 agonists
US10335406B2 (en) * 2015-10-01 2019-07-02 Elysium Therapeutics, Inc. Opioid compositions resistant to overdose and abuse
JP2018534269A (ja) 2015-10-01 2018-11-22 エリージウム セラピューティクス， インコーポレイテッド 過剰摂取および乱用に抵抗性のポリサブユニットオピオイドプロドラッグ
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EP3595663A4 (en) * 2017-03-17 2021-01-13 Elysium Therapeutics, Inc. MULTIPLE SUBUNITY OPIOID PRODRUGS WITH RESISTANCE TO OVERDOSE AND ABUSE
US10717712B2 (en) 2018-07-27 2020-07-21 Concentric Analgesics, Inc. Pegylated prodrugs of phenolic TRPV1 agonists
US20220175699A1 (en) 2019-03-06 2022-06-09 Ensysce Biosciences, Inc. Compositions comprising enzyme-cleavable amphetamine prodrugs and inhibitors thereof
US12599578B2 (en) 2021-03-09 2026-04-14 Ensysce Biosciences Inc. Compositions comprising enzyme-cleavable prodrugs and controlled release nafamostat and methods of use thereof
MX2024003466A (es) 2021-09-29 2024-06-04 Ensysce Biosciences Inc Profarmacos de metadona escindibles por enzimas y metodos de uso de los mismos.

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