JP2011519871A5 - - Google Patents

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Publication number
JP2011519871A5
JP2011519871A5 JP2011507765A JP2011507765A JP2011519871A5 JP 2011519871 A5 JP2011519871 A5 JP 2011519871A5 JP 2011507765 A JP2011507765 A JP 2011507765A JP 2011507765 A JP2011507765 A JP 2011507765A JP 2011519871 A5 JP2011519871 A5 JP 2011519871A5
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JP
Japan
Prior art keywords
compound
pharmaceutically acceptable
acceptable salt
salt
pharmaceutically
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2011507765A
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English (en)
Japanese (ja)
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JP2011519871A (ja
JP4790871B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/CA2009/000611 external-priority patent/WO2009135299A1/en
Publication of JP2011519871A publication Critical patent/JP2011519871A/ja
Publication of JP2011519871A5 publication Critical patent/JP2011519871A5/ja
Application granted granted Critical
Publication of JP4790871B2 publication Critical patent/JP4790871B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2011507765A 2008-05-05 2009-05-04 レニン阻害剤としての3,4−置換ピペリジン誘導体 Expired - Fee Related JP4790871B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US12652908P 2008-05-05 2008-05-05
US61/126,529 2008-05-05
US18830308P 2008-08-07 2008-08-07
US61/188,303 2008-08-07
PCT/CA2009/000611 WO2009135299A1 (en) 2008-05-05 2009-05-04 3, 4 - substituted piperidine derivatives as renin inhibitors

Related Child Applications (2)

Application Number Title Priority Date Filing Date
JP2011123057A Division JP5653842B2 (ja) 2008-05-05 2011-06-01 レニン阻害剤としての3,4−置換ピペリジン誘導体
JP2011123054A Division JP5587246B2 (ja) 2008-05-05 2011-06-01 レニン阻害剤としての3,4−置換ピペリジン誘導体

Publications (3)

Publication Number Publication Date
JP2011519871A JP2011519871A (ja) 2011-07-14
JP2011519871A5 true JP2011519871A5 (https=) 2011-08-25
JP4790871B2 JP4790871B2 (ja) 2011-10-12

Family

ID=41264366

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2011507765A Expired - Fee Related JP4790871B2 (ja) 2008-05-05 2009-05-04 レニン阻害剤としての3,4−置換ピペリジン誘導体
JP2011123057A Expired - Fee Related JP5653842B2 (ja) 2008-05-05 2011-06-01 レニン阻害剤としての3,4−置換ピペリジン誘導体
JP2011123054A Expired - Fee Related JP5587246B2 (ja) 2008-05-05 2011-06-01 レニン阻害剤としての3,4−置換ピペリジン誘導体

Family Applications After (2)

Application Number Title Priority Date Filing Date
JP2011123057A Expired - Fee Related JP5653842B2 (ja) 2008-05-05 2011-06-01 レニン阻害剤としての3,4−置換ピペリジン誘導体
JP2011123054A Expired - Fee Related JP5587246B2 (ja) 2008-05-05 2011-06-01 レニン阻害剤としての3,4−置換ピペリジン誘導体

Country Status (23)

Country Link
US (1) US8889714B2 (https=)
EP (1) EP2274295B1 (https=)
JP (3) JP4790871B2 (https=)
KR (2) KR101403311B1 (https=)
CN (1) CN102015682B (https=)
AU (1) AU2009243875B2 (https=)
BR (1) BRPI0912388A2 (https=)
CA (1) CA2722734C (https=)
CO (1) CO6311081A2 (https=)
CR (1) CR11809A (https=)
DO (1) DOP2010000329A (https=)
EA (1) EA020853B1 (https=)
ES (1) ES2548134T3 (https=)
IL (1) IL208467A (https=)
MA (1) MA32296B1 (https=)
MX (1) MX2010012067A (https=)
MY (1) MY152042A (https=)
NI (1) NI201000188A (https=)
NZ (1) NZ589019A (https=)
PL (1) PL2274295T3 (https=)
SG (1) SG192543A1 (https=)
SV (1) SV2010003723A (https=)
WO (1) WO2009135299A1 (https=)

Families Citing this family (10)

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CN102099036B (zh) 2008-06-03 2015-05-27 英特芒尼公司 用于治疗炎性疾患和纤维化疾患的化合物和方法
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TWI562977B (en) * 2010-11-05 2016-12-21 Bayer Ip Gmbh Process for the preparation of substituted n-(benzyl)cyclopropanamines by imine hydrogenation
UA112897C2 (uk) * 2012-05-09 2016-11-10 Байєр Фарма Акцієнгезелльшафт Біциклічно заміщені урацили та їх застосування для лікування і/або профілактики захворювань
AR092742A1 (es) 2012-10-02 2015-04-29 Intermune Inc Piridinonas antifibroticas
MX382781B (es) 2014-04-02 2025-03-13 Intermune Inc Piridinonas anti-fibroticas.
CN107602381B (zh) * 2017-09-11 2021-03-16 陕西莱特光电材料股份有限公司 一种萘甲酸酯类衍生物及其制备方法
CN108033876A (zh) * 2017-12-20 2018-05-15 江汉大学 一种5-溴-2-氯苯甲醛的制备方法
US12459934B2 (en) 2018-11-28 2025-11-04 Basf Se Pesticidal compounds
WO2021219513A1 (en) 2020-04-28 2021-11-04 Basf Se Pesticidal compounds

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