JP2011105738A5 - - Google Patents

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Publication number
JP2011105738A5
JP2011105738A5 JP2011010997A JP2011010997A JP2011105738A5 JP 2011105738 A5 JP2011105738 A5 JP 2011105738A5 JP 2011010997 A JP2011010997 A JP 2011010997A JP 2011010997 A JP2011010997 A JP 2011010997A JP 2011105738 A5 JP2011105738 A5 JP 2011105738A5
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JP
Japan
Prior art keywords
pharmaceutical composition
compound
pharmaceutically acceptable
acceptable salt
composition according
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JP2011010997A
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English (en)
Japanese (ja)
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JP5400812B2 (ja
JP2011105738A (ja
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Priority claimed from GBGB0412769.2A external-priority patent/GB0412769D0/en
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Publication of JP2011105738A publication Critical patent/JP2011105738A/ja
Publication of JP2011105738A5 publication Critical patent/JP2011105738A5/ja
Application granted granted Critical
Publication of JP5400812B2 publication Critical patent/JP5400812B2/ja
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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JP2011010997A 2004-06-08 2011-01-21 バニロイドアンタゴニストとして有用なキナゾリノン誘導体 Expired - Lifetime JP5400812B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB0412769.2 2004-06-08
GBGB0412769.2A GB0412769D0 (en) 2004-06-08 2004-06-08 Organic compounds

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2007526311A Division JP4703650B2 (ja) 2004-06-08 2005-06-08 バニロイドアンタゴニストとして有用なキナゾリノン誘導体

Publications (3)

Publication Number Publication Date
JP2011105738A JP2011105738A (ja) 2011-06-02
JP2011105738A5 true JP2011105738A5 (https=) 2012-03-08
JP5400812B2 JP5400812B2 (ja) 2014-01-29

Family

ID=32696854

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2007526311A Expired - Lifetime JP4703650B2 (ja) 2004-06-08 2005-06-08 バニロイドアンタゴニストとして有用なキナゾリノン誘導体
JP2011010997A Expired - Lifetime JP5400812B2 (ja) 2004-06-08 2011-01-21 バニロイドアンタゴニストとして有用なキナゾリノン誘導体

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2007526311A Expired - Lifetime JP4703650B2 (ja) 2004-06-08 2005-06-08 バニロイドアンタゴニストとして有用なキナゾリノン誘導体

Country Status (29)

Country Link
US (4) US7960399B2 (https=)
EP (1) EP1755606B2 (https=)
JP (2) JP4703650B2 (https=)
KR (2) KR20100101017A (https=)
CN (1) CN1956721B (https=)
AT (1) ATE376833T1 (https=)
AU (2) AU2005251476C1 (https=)
BR (1) BRPI0511933B8 (https=)
CA (1) CA2567821C (https=)
CY (1) CY1107846T1 (https=)
DE (1) DE602005003128T3 (https=)
DK (1) DK1755606T4 (https=)
EC (2) ECSP067067A (https=)
ES (1) ES2293584T5 (https=)
GB (1) GB0412769D0 (https=)
HR (1) HRP20070577T4 (https=)
IL (1) IL179532A (https=)
MA (1) MA28685B1 (https=)
MX (1) MXPA06014249A (https=)
NO (1) NO338181B1 (https=)
NZ (1) NZ551630A (https=)
PL (1) PL1755606T5 (https=)
PT (1) PT1755606E (https=)
RU (2) RU2449995C2 (https=)
SG (1) SG153811A1 (https=)
SI (1) SI1755606T2 (https=)
TN (1) TNSN06405A1 (https=)
WO (1) WO2005120510A1 (https=)
ZA (1) ZA200609634B (https=)

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US8349852B2 (en) 2009-01-13 2013-01-08 Novartis Ag Quinazolinone derivatives useful as vanilloid antagonists
JP2013518085A (ja) 2010-02-01 2013-05-20 ノバルティス アーゲー ＣＲＦ−１受容体アンタゴニストとしてのピラゾロ［５，１ｂ］オキサゾール誘導体
AR080056A1 (es) 2010-02-01 2012-03-07 Novartis Ag Derivados de ciclohexil-amida como antagonistas de los receptores de crf
JP5748777B2 (ja) 2010-02-02 2015-07-15 ノバルティス アーゲー Ｃｒｆ受容体アンタゴニストとしてのシクロヘキシルアミド誘導体
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CA2867043A1 (en) 2012-05-03 2013-11-07 Novartis Ag L-malate salt of 2,7-diaza-spiro[4.5]dec-7-yle derivatives and crystalline forms thereof as ghrelin receptor agonists
JP2016510749A (ja) 2013-03-05 2016-04-11 ユニヴァーシティー オブ ノートル ダム デュ ラック キナゾリノン抗生物質
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JP6994061B2 (ja) 2019-02-15 2022-01-14 ノバルティス アーゲー ４－（７－ヒドロキシ－２－イソプロピル－４－オキソ－４ｈ－キナゾリン－３－イル）－ベンゾニトリルの製剤
EP4431497A1 (en) 2019-02-15 2024-09-18 Bausch + Lomb Ireland Limited Crystalline forms of 4-(7-hydroxy-2-isopropyl-4-oxo-4h-quinazolin-3-yl)-benzonitrile and formulations thereof
EP3972695A1 (en) 2019-05-23 2022-03-30 Gilead Sciences, Inc. Substituted exo-methylene-oxindoles which are hpk1/map4k1 inhibitors
RU2755206C1 (ru) 2020-05-20 2021-09-14 Федеральное государственное бюджетное учреждение науки Тихоокеанский институт биоорганической химии им. Г.Б. Елякова Дальневосточного отделения Российской академии наук (ТИБОХ ДВО РАН) Средство пролонгированного анальгетического действия и лекарственный препарат на его основе
WO2022029656A1 (en) 2020-08-06 2022-02-10 Novartis Ag Crystalline forms of 4-(7-hydroxy-2-isopropyl-4-oxo-4h-quinazolin-3-yl)-benzonitrile and formulations thereof
WO2022105792A1 (zh) * 2020-11-17 2022-05-27 苏州晶云药物科技股份有限公司 一种喹唑啉酮衍生物的新晶型及其制备方法
UY39681A (es) 2021-03-26 2022-10-31 Novartis Ag Derivados de ciclobutilo 1,3–sustituidos y sus usos
JP2025531367A (ja) 2022-09-21 2025-09-19 ボシュ ＋ ロム アイルランド リミテッド Ｔｒｐｖ１アンタゴニストの結晶多形形態およびその製剤
KR20250030194A (ko) 2023-08-24 2025-03-05 코웨이 주식회사 출수 장치

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