JP2011046700A5 - - Google Patents

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JP2011046700A5
JP2011046700A5 JP2010171260A JP2010171260A JP2011046700A5 JP 2011046700 A5 JP2011046700 A5 JP 2011046700A5 JP 2010171260 A JP2010171260 A JP 2010171260A JP 2010171260 A JP2010171260 A JP 2010171260A JP 2011046700 A5 JP2011046700 A5 JP 2011046700A5
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solvate
pharmaceutically acceptable
acceptable salt
group
compound
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JP2010171260A
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JP2011046700A (ja
JP5520158B2 (ja
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JP2010171260A 2009-07-31 2010-07-30 含窒素スピロ環化合物及びその医薬用途 Active JP5520158B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2010171260A JP5520158B2 (ja) 2009-07-31 2010-07-30 含窒素スピロ環化合物及びその医薬用途

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2009179502 2009-07-31
JP2009179502 2009-07-31
JP2010171260A JP5520158B2 (ja) 2009-07-31 2010-07-30 含窒素スピロ環化合物及びその医薬用途

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2014077850A Division JP2014141516A (ja) 2009-07-31 2014-04-04 含窒素スピロ環化合物及びその医薬用途

Publications (3)

Publication Number Publication Date
JP2011046700A JP2011046700A (ja) 2011-03-10
JP2011046700A5 true JP2011046700A5 (enExample) 2014-02-13
JP5520158B2 JP5520158B2 (ja) 2014-06-11

Family

ID=43529436

Family Applications (9)

Application Number Title Priority Date Filing Date
JP2010171260A Active JP5520158B2 (ja) 2009-07-31 2010-07-30 含窒素スピロ環化合物及びその医薬用途
JP2014077850A Pending JP2014141516A (ja) 2009-07-31 2014-04-04 含窒素スピロ環化合物及びその医薬用途
JP2015224910A Ceased JP2016029104A (ja) 2009-07-31 2015-11-17 含窒素スピロ環化合物及びその医薬用途
JP2016214954A Ceased JP2017019877A (ja) 2009-07-31 2016-11-02 含窒素スピロ環化合物及びその医薬用途
JP2018028525A Ceased JP2018111701A (ja) 2009-07-31 2018-02-21 含窒素スピロ環化合物及びその医薬用途
JP2019219283A Withdrawn JP2020033384A (ja) 2009-07-31 2019-12-04 含窒素スピロ環化合物及びその医薬用途
JP2021144545A Withdrawn JP2021183653A (ja) 2009-07-31 2021-09-06 含窒素スピロ環化合物及びその医薬用途
JP2023128376A Withdrawn JP2023138641A (ja) 2009-07-31 2023-08-07 含窒素スピロ環化合物及びその医薬用途
JP2025077764A Pending JP2025109780A (ja) 2009-07-31 2025-05-08 含窒素スピロ環化合物及びその医薬用途

Family Applications After (8)

Application Number Title Priority Date Filing Date
JP2014077850A Pending JP2014141516A (ja) 2009-07-31 2014-04-04 含窒素スピロ環化合物及びその医薬用途
JP2015224910A Ceased JP2016029104A (ja) 2009-07-31 2015-11-17 含窒素スピロ環化合物及びその医薬用途
JP2016214954A Ceased JP2017019877A (ja) 2009-07-31 2016-11-02 含窒素スピロ環化合物及びその医薬用途
JP2018028525A Ceased JP2018111701A (ja) 2009-07-31 2018-02-21 含窒素スピロ環化合物及びその医薬用途
JP2019219283A Withdrawn JP2020033384A (ja) 2009-07-31 2019-12-04 含窒素スピロ環化合物及びその医薬用途
JP2021144545A Withdrawn JP2021183653A (ja) 2009-07-31 2021-09-06 含窒素スピロ環化合物及びその医薬用途
JP2023128376A Withdrawn JP2023138641A (ja) 2009-07-31 2023-08-07 含窒素スピロ環化合物及びその医薬用途
JP2025077764A Pending JP2025109780A (ja) 2009-07-31 2025-05-08 含窒素スピロ環化合物及びその医薬用途

Country Status (36)

Country Link
US (4) US8609647B2 (enExample)
EP (3) EP2460806B1 (enExample)
JP (9) JP5520158B2 (enExample)
KR (1) KR101773208B1 (enExample)
CN (1) CN102510865B (enExample)
AR (1) AR077497A1 (enExample)
AU (1) AU2010278066B2 (enExample)
BR (1) BR112012002157B1 (enExample)
CA (1) CA2767899C (enExample)
CO (1) CO6491052A2 (enExample)
CY (1) CY1118747T1 (enExample)
DK (1) DK2460806T3 (enExample)
ES (1) ES2616705T3 (enExample)
FI (1) FIC20250012I1 (enExample)
FR (1) FR25C1010I1 (enExample)
HR (1) HRP20170447T1 (enExample)
HU (2) HUE033070T2 (enExample)
IL (1) IL217048A (enExample)
LT (2) LT2460806T (enExample)
ME (1) ME02667B (enExample)
MX (1) MX2012001313A (enExample)
MY (1) MY163495A (enExample)
NL (1) NL301321I2 (enExample)
NO (1) NO2025014I1 (enExample)
NZ (1) NZ597994A (enExample)
PE (1) PE20121276A1 (enExample)
PL (1) PL2460806T3 (enExample)
PT (1) PT2460806T (enExample)
RS (1) RS55913B1 (enExample)
RU (1) RU2630694C2 (enExample)
SG (1) SG176918A1 (enExample)
SI (1) SI2460806T1 (enExample)
SM (1) SMT201700166T1 (enExample)
TW (1) TWI466885B (enExample)
WO (1) WO2011013785A1 (enExample)
ZA (1) ZA201200689B (enExample)

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CN117159553A (zh) 2016-01-21 2023-12-05 利奥制药有限公司 慢性手部湿疹的治疗
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US10851116B2 (en) 2017-01-20 2020-12-01 Leo Pharma A/S Bicyclic amines as novel JAK kinase inhibitors
WO2018141842A1 (en) * 2017-02-03 2018-08-09 Leo Pharma A/S 5-(7H-PYRROLO[2,3-d]PYRIMIDIN-4-YL)-5-AZASPIRO[2.5]OCTANE-8-CARBOXYLIC ACID DERIVATIVES AS NOVEL JAK KINASE INHIBITORS
JP2020536898A (ja) * 2017-10-10 2020-12-17 バイオジェン インコーポレイテッド スピロ誘導体を調製するためのプロセス
SG11202007251XA (en) * 2018-01-31 2020-08-28 Aptinyx Inc Spiro-lactam nmda receptor modulators and uses thereof
WO2020007698A1 (en) * 2018-07-06 2020-01-09 Leo Pharma A/S Novel amino-imidazopyrimidine derivatives as janus kinase inhibitors and pharmaceutical use thereof
WO2020092015A1 (en) 2018-11-02 2020-05-07 University Of Rochester Therapeutic mitigation of epithelial infection
MX2021012874A (es) 2019-05-15 2021-11-17 Leo Pharma As Tratamiento del lupus eritematoso cutaneo.
CN118903144A (zh) * 2019-08-07 2024-11-08 乐敦制药株式会社 泪液分泌促进用眼科组合物
CN119367282A (zh) * 2019-12-27 2025-01-28 乐敦制药株式会社 水性组合物
CN111560021B (zh) * 2020-06-30 2023-05-26 上海鲲博玖瑞医药科技发展有限公司 一种德高替尼中间体及其制备方法
CN111574540B (zh) * 2020-06-30 2023-08-29 云南华派医药科技有限公司 一种德高替尼的制备方法
CN111606929B (zh) * 2020-06-30 2023-07-07 中瀚(齐河县)生物医药科技有限公司 德高替尼的制备方法
CN114591321A (zh) * 2020-12-04 2022-06-07 广州费米子科技有限责任公司 氮杂并环化合物、其制备方法及其用途
TW202241439A (zh) * 2020-12-29 2022-11-01 大陸商上海岸闊醫藥科技有限公司 治療與抗腫瘤劑相關的皮膚疾病或病症的試劑和方法
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