JP2015501799A5 - - Google Patents

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JP2015501799A5
JP2015501799A5 JP2014541757A JP2014541757A JP2015501799A5 JP 2015501799 A5 JP2015501799 A5 JP 2015501799A5 JP 2014541757 A JP2014541757 A JP 2014541757A JP 2014541757 A JP2014541757 A JP 2014541757A JP 2015501799 A5 JP2015501799 A5 JP 2015501799A5
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JP
Japan
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compound
optionally substituted
ethyl
hydrocarbon group
fluorine
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JP2014541757A
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English (en)
Japanese (ja)
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JP2015501799A (ja
JP6083818B2 (ja
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Priority claimed from PCT/GB2012/052857 external-priority patent/WO2013072705A1/en
Publication of JP2015501799A publication Critical patent/JP2015501799A/ja
Publication of JP2015501799A5 publication Critical patent/JP2015501799A5/ja
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JP2014541757A 2011-11-18 2012-11-16 ムスカリンｍ１受容体アゴニスト Active JP6083818B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201161632813P 2011-11-18 2011-11-18
US61/632,813 2011-11-18
PCT/GB2012/052857 WO2013072705A1 (en) 2011-11-18 2012-11-16 Muscarinic m1 receptor agonists

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2017007283A Division JP6404374B2 (ja) 2011-11-18 2017-01-19 ムスカリンｍ１受容体アゴニスト

Publications (3)

Publication Number Publication Date
JP2015501799A JP2015501799A (ja) 2015-01-19
JP2015501799A5 true JP2015501799A5 (enExample) 2016-01-14
JP6083818B2 JP6083818B2 (ja) 2017-02-22

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ID=47278335

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2014541757A Active JP6083818B2 (ja) 2011-11-18 2012-11-16 ムスカリンｍ１受容体アゴニスト
JP2017007283A Active JP6404374B2 (ja) 2011-11-18 2017-01-19 ムスカリンｍ１受容体アゴニスト

Family Applications After (1)

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JP2017007283A Active JP6404374B2 (ja) 2011-11-18 2017-01-19 ムスカリンｍ１受容体アゴニスト

Country Status (16)

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US (6) US9187451B2 (enExample)
EP (1) EP2780015B1 (enExample)
JP (2) JP6083818B2 (enExample)
CN (2) CN104039321B (enExample)
AU (3) AU2012338581B2 (enExample)
BR (1) BR112014012056B1 (enExample)
CA (1) CA2856076C (enExample)
DK (1) DK2780015T3 (enExample)
ES (1) ES2619829T3 (enExample)
GB (1) GB2511685A (enExample)
HU (1) HUE033114T2 (enExample)
IN (1) IN2014KN01075A (enExample)
PL (1) PL2780015T3 (enExample)
PT (1) PT2780015T (enExample)
SG (1) SG11201402405QA (enExample)
WO (1) WO2013072705A1 (enExample)

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HUE033114T2 (en) 2011-11-18 2017-11-28 Heptares Therapeutics Ltd Muscarin M1 receptor agonists
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RS65894B1 (sr) * 2014-02-06 2024-09-30 Nxera Pharma Uk Ltd Biciklična aza jedinjenja kao agonisti muskarinskog receptora
GB201404922D0 (en) * 2014-03-19 2014-04-30 Heptares Therapeutics Ltd Pharmaceutical compounds
GB201504675D0 (en) * 2015-03-19 2015-05-06 Heptares Therapeutics Ltd Pharmaceutical compounds
GB201513740D0 (en) * 2015-08-03 2015-09-16 Heptares Therapeutics Ltd Muscarinic agonist
GB201513743D0 (en) 2015-08-03 2015-09-16 Heptares Therapeutics Ltd Muscarinic agonists
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GB201519352D0 (en) * 2015-11-02 2015-12-16 Heptares Therapeutics Ltd Pharmaceutical compounds
GB201617454D0 (en) 2016-10-14 2016-11-30 Heptares Therapeutics Limited Pharmaceutical compounds
CN108226319A (zh) * 2016-12-22 2018-06-29 亚宝药业集团股份有限公司 一种检测卡巴拉汀贴剂中光学异构体的方法
TW201922758A (zh) 2017-10-24 2019-06-16 美商歐樂根公司 烯胺及烯胺的非鏡像選擇性還原
JP6691928B2 (ja) * 2018-02-07 2020-05-13 株式会社ジンズホールディングス アイウエアセット及び信号処理ユニット
GB201810239D0 (en) 2018-06-22 2018-08-08 Heptares Therapeutics Ltd Pharmaceutical compounds
GB201819960D0 (en) 2018-12-07 2019-01-23 Heptares Therapeutics Ltd Pharmaceutical compounds
GB201819961D0 (en) 2018-12-07 2019-01-23 Heptares Therapeutics Ltd Pharmaceutical compounds
GB202020191D0 (en) 2020-12-18 2021-02-03 Heptares Therapeutics Ltd Pharmaceutical compounds
CN113121495A (zh) * 2020-01-10 2021-07-16 深圳市九明药业有限公司 一种地氯雷他定的制备方法
WO2025167860A1 (zh) * 2024-02-06 2025-08-14 南京迈诺威医药科技有限公司 一种含有占诺美林或其盐的药物组合物

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CA2883210C (en) 2012-09-18 2021-06-15 Heptares Therapeutics Limited Bicyclic aza compounds as muscarinic m1 receptor agonists
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RS65894B1 (sr) 2014-02-06 2024-09-30 Nxera Pharma Uk Ltd Biciklična aza jedinjenja kao agonisti muskarinskog receptora
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GB201513742D0 (en) 2015-08-03 2015-09-16 Heptares Therapeutics Ltd Muscarinic agonists
GB201513743D0 (en) 2015-08-03 2015-09-16 Heptares Therapeutics Ltd Muscarinic agonists
GB201519352D0 (en) 2015-11-02 2015-12-16 Heptares Therapeutics Ltd Pharmaceutical compounds
GB201617454D0 (en) 2016-10-14 2016-11-30 Heptares Therapeutics Limited Pharmaceutical compounds
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GB201709652D0 (en) 2017-06-16 2017-08-02 Heptares Therapeutics Ltd Pharmaceutical compounds
TW201922758A (zh) 2017-10-24 2019-06-16 美商歐樂根公司 烯胺及烯胺的非鏡像選擇性還原
GB201810239D0 (en) 2018-06-22 2018-08-08 Heptares Therapeutics Ltd Pharmaceutical compounds
GB201810245D0 (en) 2018-06-22 2018-08-08 Heptares Therapeutics Ltd Pharmaceutical compounds
GB201819960D0 (en) 2018-12-07 2019-01-23 Heptares Therapeutics Ltd Pharmaceutical compounds
GB201819961D0 (en) 2018-12-07 2019-01-23 Heptares Therapeutics Ltd Pharmaceutical compounds
GB202020191D0 (en) 2020-12-18 2021-02-03 Heptares Therapeutics Ltd Pharmaceutical compounds
GB202103211D0 (en) 2021-03-08 2021-04-21 Heptares Therapeutics Ltd Pharmaceutical compounds for use in therapy

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