JP2010539095A5 - - Google Patents
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- JP2010539095A5 JP2010539095A5 JP2010524243A JP2010524243A JP2010539095A5 JP 2010539095 A5 JP2010539095 A5 JP 2010539095A5 JP 2010524243 A JP2010524243 A JP 2010524243A JP 2010524243 A JP2010524243 A JP 2010524243A JP 2010539095 A5 JP2010539095 A5 JP 2010539095A5
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- substituted
- aryl
- cycloalkyl
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Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US97114407P | 2007-09-10 | 2007-09-10 | |
| US60/971,144 | 2007-09-10 | ||
| US1337207P | 2007-12-13 | 2007-12-13 | |
| US61/013,372 | 2007-12-13 | ||
| PCT/US2008/075848 WO2009036059A2 (en) | 2007-09-10 | 2008-09-10 | Novel stat3 pathway inhibitors and cancer stem cell inhibitors |
Related Child Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2014232396A Division JP6106149B2 (ja) | 2007-09-10 | 2014-11-17 | 新規のStat3経路阻害剤及び癌幹細胞阻害剤 |
| JP2014232397A Division JP2015034179A (ja) | 2007-09-10 | 2014-11-17 | 新規のStat3経路阻害剤及び癌幹細胞阻害剤 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2010539095A JP2010539095A (ja) | 2010-12-16 |
| JP2010539095A5 true JP2010539095A5 (enExample) | 2012-09-27 |
| JP5688840B2 JP5688840B2 (ja) | 2015-03-25 |
Family
ID=40452461
Family Applications (16)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010524251A Expired - Fee Related JP5872160B2 (ja) | 2007-09-10 | 2008-09-10 | 癌治療のための新規の組成物および方法 |
| JP2010524243A Expired - Fee Related JP5688840B2 (ja) | 2007-09-10 | 2008-09-10 | 新規のStat3経路阻害剤及び癌幹細胞阻害剤 |
| JP2010524249A Expired - Fee Related JP5701603B2 (ja) | 2007-09-10 | 2008-09-10 | Stat3経路阻害剤および癌幹細胞経路阻害剤の新規のグループ |
| JP2014177908A Expired - Fee Related JP5925849B2 (ja) | 2007-09-10 | 2014-09-02 | Stat3経路阻害剤および癌幹細胞経路阻害剤の新規のグループ |
| JP2014177915A Expired - Fee Related JP5938072B2 (ja) | 2007-09-10 | 2014-09-02 | 癌治療のための新規の組成物および方法 |
| JP2014232397A Withdrawn JP2015034179A (ja) | 2007-09-10 | 2014-11-17 | 新規のStat3経路阻害剤及び癌幹細胞阻害剤 |
| JP2014232396A Expired - Fee Related JP6106149B2 (ja) | 2007-09-10 | 2014-11-17 | 新規のStat3経路阻害剤及び癌幹細胞阻害剤 |
| JP2015230291A Expired - Fee Related JP6358659B2 (ja) | 2007-09-10 | 2015-11-26 | Stat3経路阻害剤および癌幹細胞経路阻害剤の新規のグループ |
| JP2016004076A Expired - Fee Related JP6347795B2 (ja) | 2007-09-10 | 2016-01-13 | 癌治療のための新規の組成物および方法 |
| JP2016016973A Expired - Fee Related JP6346628B2 (ja) | 2007-09-10 | 2016-02-01 | Stat3経路阻害剤および癌幹細胞経路阻害剤の新規のグループ |
| JP2016097607A Withdrawn JP2016147906A (ja) | 2007-09-10 | 2016-05-16 | 新規のStat3経路阻害剤及び癌幹細胞阻害剤 |
| JP2017242778A Withdrawn JP2018076349A (ja) | 2007-09-10 | 2017-12-19 | Stat3経路阻害剤および癌幹細胞経路阻害剤の新規のグループ |
| JP2018102234A Withdrawn JP2018131464A (ja) | 2007-09-10 | 2018-05-29 | 癌治療のための新規の組成物および方法 |
| JP2019029436A Pending JP2019073560A (ja) | 2007-09-10 | 2019-02-21 | 新規のStat3経路阻害剤及び癌幹細胞阻害剤 |
| JP2020085065A Pending JP2020117547A (ja) | 2007-09-10 | 2020-05-14 | 癌治療のための新規の組成物および方法 |
| JP2020091326A Pending JP2020143135A (ja) | 2007-09-10 | 2020-05-26 | Stat3経路阻害剤および癌幹細胞経路阻害剤の新規のグループ |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010524251A Expired - Fee Related JP5872160B2 (ja) | 2007-09-10 | 2008-09-10 | 癌治療のための新規の組成物および方法 |
Family Applications After (14)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010524249A Expired - Fee Related JP5701603B2 (ja) | 2007-09-10 | 2008-09-10 | Stat3経路阻害剤および癌幹細胞経路阻害剤の新規のグループ |
| JP2014177908A Expired - Fee Related JP5925849B2 (ja) | 2007-09-10 | 2014-09-02 | Stat3経路阻害剤および癌幹細胞経路阻害剤の新規のグループ |
| JP2014177915A Expired - Fee Related JP5938072B2 (ja) | 2007-09-10 | 2014-09-02 | 癌治療のための新規の組成物および方法 |
| JP2014232397A Withdrawn JP2015034179A (ja) | 2007-09-10 | 2014-11-17 | 新規のStat3経路阻害剤及び癌幹細胞阻害剤 |
| JP2014232396A Expired - Fee Related JP6106149B2 (ja) | 2007-09-10 | 2014-11-17 | 新規のStat3経路阻害剤及び癌幹細胞阻害剤 |
| JP2015230291A Expired - Fee Related JP6358659B2 (ja) | 2007-09-10 | 2015-11-26 | Stat3経路阻害剤および癌幹細胞経路阻害剤の新規のグループ |
| JP2016004076A Expired - Fee Related JP6347795B2 (ja) | 2007-09-10 | 2016-01-13 | 癌治療のための新規の組成物および方法 |
| JP2016016973A Expired - Fee Related JP6346628B2 (ja) | 2007-09-10 | 2016-02-01 | Stat3経路阻害剤および癌幹細胞経路阻害剤の新規のグループ |
| JP2016097607A Withdrawn JP2016147906A (ja) | 2007-09-10 | 2016-05-16 | 新規のStat3経路阻害剤及び癌幹細胞阻害剤 |
| JP2017242778A Withdrawn JP2018076349A (ja) | 2007-09-10 | 2017-12-19 | Stat3経路阻害剤および癌幹細胞経路阻害剤の新規のグループ |
| JP2018102234A Withdrawn JP2018131464A (ja) | 2007-09-10 | 2018-05-29 | 癌治療のための新規の組成物および方法 |
| JP2019029436A Pending JP2019073560A (ja) | 2007-09-10 | 2019-02-21 | 新規のStat3経路阻害剤及び癌幹細胞阻害剤 |
| JP2020085065A Pending JP2020117547A (ja) | 2007-09-10 | 2020-05-14 | 癌治療のための新規の組成物および方法 |
| JP2020091326A Pending JP2020143135A (ja) | 2007-09-10 | 2020-05-26 | Stat3経路阻害剤および癌幹細胞経路阻害剤の新規のグループ |
Country Status (14)
| Country | Link |
|---|---|
| US (12) | US9745278B2 (enExample) |
| EP (6) | EP2190429B1 (enExample) |
| JP (16) | JP5872160B2 (enExample) |
| CN (6) | CN101854930B (enExample) |
| CA (4) | CA2911990C (enExample) |
| CY (3) | CY1117604T1 (enExample) |
| DK (4) | DK3050566T3 (enExample) |
| ES (3) | ES2569215T3 (enExample) |
| HR (3) | HRP20160430T1 (enExample) |
| HU (3) | HUE027657T2 (enExample) |
| PL (4) | PL2190429T3 (enExample) |
| PT (2) | PT2200431T (enExample) |
| SI (3) | SI2194987T1 (enExample) |
| WO (3) | WO2009036099A1 (enExample) |
Families Citing this family (131)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SI1848414T1 (sl) | 2005-02-03 | 2011-08-31 | Gen Hospital Corp | Postopek za zdravljenje raka, odpornega na gefitinib |
| RU2451524C2 (ru) | 2005-11-04 | 2012-05-27 | Вайет | Противоопухолевые комбинации с ингибиторами mtor, герцептином и/или hki-272 |
| HRP20160430T1 (hr) * | 2007-09-10 | 2016-05-20 | Boston Biomedical, Inc. | Nova grupa inhibitora stat3 puta i inhibitora puta matičnih stanica karcinoma |
| US8022216B2 (en) | 2007-10-17 | 2011-09-20 | Wyeth Llc | Maleate salts of (E)-N-{4-[3-chloro-4-(2-pyridinylmethoxy)anilino]-3-cyano-7-ethoxy-6-quinolinyl}-4-(dimethylamino)-2-butenamide and crystalline forms thereof |
| US20130331294A1 (en) | 2007-11-09 | 2013-12-12 | Fox Chase Cancer Center | Egfr/nedd9/tgf-beta interactome and methods of use thereof for the identification of agents having efficacy in the treatment of hyperproliferative disorders |
| WO2009062199A1 (en) * | 2007-11-09 | 2009-05-14 | Fox Chase Cancer Center | EGFR/NEDD9/TGF-β LNTERACTOME AND METHODS OF USE THEREOF FOR THE IDENTIFICATION OF AGENTS HAVING EFFICACY IN THE TREATMENT OF HYPERPROLIFERATIVE DISORDERS |
| UY31800A (es) * | 2008-05-05 | 2009-11-10 | Smithkline Beckman Corp | Metodo de tratamiento de cancer usando un inhibidor de cmet y axl y un inhibidor de erbb |
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| EA020766B1 (ru) | 2008-07-08 | 2015-01-30 | Борд Оф Риджентс, Дзе Юниверсити Оф Техас Систем | Ингибиторы пролиферации и активации переносчика сигнала и активатора транскрипции (stats) |
| KR101434009B1 (ko) | 2008-08-04 | 2014-08-25 | 와이어쓰 엘엘씨 | 4-아닐리노-3-사이아노퀴놀린과 카페시타빈의 항신생물성 조합물 |
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